All Products

Displaying Products Alphabetically by Name (T)

Cat. No. Product Name / Activity
1676 T 0156 hydrochloride
Highly potent, selective PDE5 inhibitor
2373 T 0901317
Potent liver X receptor (LXR) agonist; also CAR inverse agonist
6134 T 26c disodium salt
Highly potent and selective MMP13 inhibitor
6106 T 3364366
Potent and reversible fatty acid desaturase 1 inhibitor; orally bioavailable
5269 T 5601640
Selective LIMK2 inhibitor; antitumor
2519 T 98475
GnRH receptor antagonist
6726 T-peptide
Cytotoxic Tau peptide; cell permeable
2301 T 0070907
Highly potent and selective covalent PPARγ antagonist
4538 T16Ainh - A01
Ca2+-activated Cl- channel transmembrane protein 16A (TMEM16A) inhibitor
4723 T2AA
PCNA inhibitor
6666 T3
Thyroid hormone; also promotes differentiation of oligodendroglial precursor cells
0181 TACA
GABAA agonist; also GABA-T substrate and GABA uptake inhibitor
3599 TAK 165
Potent and selective ErbB2 inhibitor
5209 TAK 21d
Potent FAAH inhibitor
6587 TAK 242
TLR4 signaling inhibitor
6777 TAK 375
Very high affinity and selective melatonin receptor agonist
4254 TAK 715
Potent p38 MAPK inhibitor; anti-inflammatory
5403 TAK 960 hydrochloride
Potent and selective PLK1 inhibitor
4506 TAME hydrochloride
Ubiquitin ligase APC/C inhibitor; promotes Cdc20 autoubiquitination
6729 TAN 452
Potent and selective peripherally acting δ opioid antagonist; antianalgesic.
5523 TAPI 0
ADAM-17 (TACE) and MMP inhibitor
6162 TAPI 1
ADAM-17 (TACE) and MMP inhibitor
6013 TAPI 2
ADAM-17 (TACE) and MMP inhibitor
4521 TAS 301
Inhibitor of smooth muscle cell migration and proliferation
5729 TASP 0390325
Potent and selective V1B receptor antagonist; orally bioavailable
5362 TASP 0433864
Selective positive allosteric modulator of mGlu2 receptors
4811 TAT 14
Nrf2 pathway activator; blocks Nrf2/Keap1 interaction
6227 TAT-Gap19
Cx43 hemichannel blocker
6847 TAT-GluA2 3Y
Inhibitor of AMPA receptor endocytosis
2905 TB 21007
α5-selective GABAA inverse agonist
2275 TBB
Selective cell-permeable CK2 inhibitor
2825 TBCA
Selective CK2 inhibitor
7259 TBK1 PROTAC® 3i
Potent TANK-binding kinase 1 (TBK1) Degrader
7260 TBK1 control PROTAC® 4
Negative control for TBK1 PROTAC® 3i (Cat. No. 7259)
1223 DL-TBOA
Selective non-transportable inhibitor of EAATs
2669 TC 1
High affinity σ1 ligand
4300 TC 14012
CXCR4 antagonist; ACKR3 (CXCR7) agonist
2518 TC 1698 dihydrochloride
α7-selective agonist
2737 TC 2559 difumarate
Selective α4β2 nAChR partial agonist
6105 TC AC 28
High affinity BET bromodomain ligand
5412 TC AQP1 1
Aquaporin 1 (AQP1) channel blocker
4825 TC ASK 10
Potent and selective ASK1 inhibitor; orally bioavailable
6466 TC E3 5031
Carboxylic acid-functionalized Thalidomide; cereblon ligand for PROTACs
6628 TC E3 5032
Precursor to Pomalidomide-based PROTACs
4575 TC HSD 21
Potent and selective 17β-hydroxysteroid dehydrogenase type 3 inhibitor
6125 TC JL 37
Potent TYK2 inhibitor
6079 TC KHNS 11
Potent and selective PI 3-kinase δ inhibitor; orally bioavailable
4708 TC LPA5 4
LPA5 receptor antagonist
4750 TC Mps1 12
Potent and selective Mps1 kinase inhibitor
5087 TC NTR1 17
Selective NTS1 partial agonist
4625 TC OT 39
Potent non-peptide oxytocin receptor partial agonist; also V1a receptor antagonist
6884 TC SL C5
Metastasis-associated lung adenocarcinoma transcript 1 (Malat1) RNA inhibitor
4066 TC-A 2317 hydrochloride
Potent, selective Aurora kinase A inhibitor
4345 TC-C 14G
High affinity and potent CB1 inverse agonist
4301 TC-DAPK 6
Potent and selective inhibitor of DAPK1
5049 TC-E 5001
Potent tankyrase inhibitor
5089 TC-E 5002
Selective KDM2/7 inhibitor
5099 TC-E 5003
Selective PRMT1 inhibitor
4572 TC-E 5005
Potent and selective PDE10A inhibitor
4898 TC-E 5006
γ-secretase modulator; reduces Aβ42 levels
5244 TC-E 5008
Selective mutant isocitrate dehydrogenase 1 (mIDH1) inhibitor; phenotypically lethal
4355 TC-F 2
Potent, reversible and selective FAAH inhibitor
4624 TC-FPR 43
Potent FPR2 agonist
5021 TC-G 1000
Potent and selective α2D agonist
4879 TC-G 1001
GPR35 agonist; more potent than zaprinast (Cat. No. 0947)
5080 TC-G 1003
High affinity somatostatin sst2 agonist
4407 TC-G 1004
Potent and selective A2A antagonist
5129 TC-G 1005
Potent and selective GPBA receptor (TGR5) agonist
4747 TC-G 1006
Potent and selective sphingosine-1-phosphate receptor 1 (S1P1) agonist
5355 TC-G 1008
Potent and selective GPR39 agonist
4353 TC-G 24
Potent and selective GSK-3β inhibitor
4270 TC-H 106
Class I histone deacetylase inhibitor
4527 TC-I 15
Potent α2β1 inhibitor; displays antithrombotic activity in vivo
4632 TC-I 2000
TRPM8 blocker
5410 TC-I 2014
Potent TRPM8 antagonist
4365 TC-MCH 7c
Selective melanin-concentrating hormone receptor 1 (MCH1R) antagonist
4435 TC-N 1752
NaV channel blocker
4370 TC-N 22A
Potent and selective positive allosteric modulator of mGlu4 receptors
4255 TC-O 9311
Potent and selective GPR139 agonist
4386 TC-P 262
Selective P2X3 and P2X2/3 antagonist
4961 TC-S 7001
Potent and highly selective ROCK inhibitor; orally active
3567 TC-S 7003
Potent Lck inhibitor
5088 TC-S 7004
Potent and selective DYRK1A/B inhibitor
4459 TC-S 7005
Potent and selective PLK2 inhibitor
5240 TC-S 7006
Potent and selective Tpl2 (Cot; MAP3K8) inhibitor
5243 TC-S 7009
High affinity and selective HIF-2α inhibitor
5286 TC-S 7010
Potent and selective Aurora kinase A inhibitor
4363 TC-SP 14
Potent S1P1 receptor agonist
5100 TC-T 6000
Potent equilibrative nucleoside transporter 4 (ENT4) inhibitor
2592 TCB-2
High affinity and potent 5-HT2A agonist
5179 TCID
Selective ubiquitin C-terminal hydrolase-L3 (UCH-L3) inhibitor
4154 TCN 201
GluN1/GluN2A-selective NMDA antagonist
4163 TCN 213
NMDA antagonist; selective for GluN2A over GluN2B containing receptors
4072 TCN 237 dihydrochloride
Highly potent and selective GluN2B NMDA antagonist
4259 TCN 238
Positive allosteric modulator of mGlu4 receptors
Constitutive androstane receptor agonist
3818 TCS 1102
Potent, dual orexin receptor antagonist
3942 TCS 1105
GABAA α2 benzodiazepine agonist
2236 TCS 183
Fragment 1-13 of GSK-3β sequence
2320 TCS 184
Scrambled control peptide for use with TCS 183 (Cat. No. 2236)
3869 TCS 2002
Potent GSK-3β inhibitor
4221 TCS 21311
Potent JAK3 inhibitor. Also inhibits GSK-3β and PKC
3877 TCS 2210
Inducer of neuronal differentiation in MSCs
3038 TCS 2312
Potent Chk1 inhibitor
3900 TCS 2314
α4β1 (VLA-4) antagonist
4069 TCS 2510
Selective EP4 agonist
4244 TCS 3035
GPR35 agonist
2591 TCS 359
Potent FLT3 inhibitor
2754 TCS 401
Selective inhibitor of PTP1B
2782 TCS 46b
GluN1A/GluN2B-selective NMDA antagonist; orally bioavailable
3938 TCS 5861528
TRPA1 blocker
4465 TCS ERK 11e
Potent and selective ERK2 inhibitor
4805 TCS HDAC6 20b
Selective HDAC6 inhibitor
2827 TCS JNK 5a
Selective inhibitor of JNK2 and JNK3
3222 TCS JNK 6o
Selective JNK inhibitor
3371 TCS OX2 29
Potent and selective OX2 antagonist
2979 TCS PIM-1 1
Selective, ATP-competitive Pim-1 kinase inhibitor
3238 TCS PrP Inhibitor 13
Antiprion agent; inhibits PrPSc accumulation
6092 TDZD 8
Selective non-ATP competitive inhibitor of GSK 3β
0645 2-TEDC
5-, 12-, 15-Lipoxygenase inhibitor
5891 TES, free acid
Buffering agent; pKa at physiolgical pH (7.4) at 25°C
6619 TFAX 488, SE
Green fluorescent dye; amine reactive
6621 TFAX 488, TFP
Green fluorescent dye; amine reactive
6623 TFAX 546, SE
Yellow fluorescent dye; amine reactive
6624 TFAX 568, SE
Orange fluorescent dye; amine reactive
6625 TFAX 594, SE
Red fluorescent dye; amine reactive
High affinity EAAT1 and EAAT2 blocker
5108 TFC 007
Potent hematopoietic prostaglandin D synthase (H-PGDS) inhibitor
1464 TFLLR-NH2
PAR1-activating peptide
3813 TFM-4AS-1
Selective androgen receptor modulator (SARM)
4336 TG 003
Potent inhibitor of Clk-family kinases; also inhibits DYRK1A/B
5052 TG 4-155
High affinity and selective EP2 receptor antagonist
5425 TGN 020
Aquaporin 4 (AQP4) channel blocker
5832 TGX 221
Potent and selective PI 3-kinase β inhibitor
6191 TH 1020
Toll-like receptor (TLR) 5/Flagellin complex antagonist
6522 TH 1217
Potent dCTP pyrophosphatase 1 inhibitor
6899 TH 257
Potent and selective allosteric LIMK 1/2 inhibitor
6534 TH 5427 hydrochloride
Potent NUDT5 inhibitor
6749 TH 5487
Selective 8-oxoguanine DNA glycosylase 1 (OGG1) inhibitor
5334 TH 588
Potent MTH1 inhibitor
6532 THAL SNS 032
Potent and selective Cdk9 degrading PROTAC
1990 (R,R)-THC
Potent subtype-selective ligand; ERα agonist/ERβ antagonist
6334 THDOC
Positive modulator of GABAA receptors; endogenous neurosteroid
0807 THIP hydrochloride
GABAA agonist
3032 THIQ
Potent and selective MC4 receptor agonist
6017 THPN
Nur77 agonist; induces autophagy in melanoma cell lines
6981 TL 0259
Selective and highly potent Fgr and Lyn kinase inhibitor; orally bioavailable
6524 TL 12-186
Multikinase degrading PROTAC
6746 TL 13-110
Negative control for TL 13-112 (Cat. No. 6745)
6745 TL 13-112
Selective ALK Degrader
6744 TL 13-12
Selective ALK degrader
6747 TL 13-22
Negative control for TL 13-12 (Cat. No. 6744)
6525 TL 13-27
Negative control for TL 12-186 (Cat. No. 6524)
5910 TL4-12
Potent MAP4K2 (GCK) inhibitor
3051 TLQP 21
VGF-derived peptide
7131 TM 38837
Highly potent CB1 inverse agonist; peripherally restricted
5769 TM 5275 sodium salt
Plasminogen activator inhibitor-1 (PAI-1) inhibitor; orally bioavailable
6194 TM 5441
Plasminogen activator inhibitor-1 (PAI-1) inhibitor
6325 TM N1324
Potent and selective GPR39 agonist; orally bioavailable
3675 TMCB
Dual-kinase inhibitor; inhibits CK2 and ERK8
5960 TMI 1
Adam 17 (TACE) and MMP inhibitor; orally bioavailable
4152 TMN 355
Cyclophilin A inhibitor
2438 TMPH hydrochloride
Neuronal nAChR antagonist
4253 TMPyP4 tosylate
Inhibitor of human telomerase
6802 6 TMR Tre
Fluorescent trehalose; selectively labels mycobacterial cell envelope
3946 TNP
Inhibitor of IP6K; also inhibits IP3K
2464 TNP-ATP triethylammonium salt
Potent and selective P2X antagonist
4414 TP 003
GABAA partial agonist; acts at benzodiazepine site
6008 TP 064
Potent and selective PRMT 4 inhibitor
6670 TP 238
CECR2 and BPTF/FALZ inhibitor
6000 TP 472
Potent BRD9/7 inhibitor
5999 TP 472N
Negative control for TP 472
2559 TPCA-1
Potent, selective inhibitor of IKKβ
4309 TPEN
Cell-permeable Zn2+ chelator; also inhibits RNA binding protein Lin28
1040 TPMPA
Selective GABAA-ρ antagonist
5343 TPPB
High affinity PKC activator; also APP modulator
5918 TPPU
Potent soluble epoxide hydrolase inhibitor; orally bioavailable and brain penetrant
4233 TQS
Positive allosteric modulator of α7 nAChRs
6908 TR 14035
Potent integrin α4β7 and α4β1 (VLA-4) antagonist; orally bioavailable
2946 TRAM 34
Potent and highly selective KCa3.1 (IK) channel blocker
4952 TRAM 39
Potent KCa3.1 (IK) blocker
3497 TRAP-6
PAR1 peptide fragment (residues 42-47); acts as a PAR1 agonist
4734 TRC 051384
Inducer of heat shock protein Hsp70
3164 TRIS hydrochloride
Commonly used laboratory reagent; used to make TBS, TAE and TBE buffers
3163 TRIS base
Commonly used laboratory reagent; used to make TBS, TAE and TBE buffers
2906 TRO 19622
Binds voltage-dependent anion channel (VDAC)
6875 TRPC6-PAM-C20
Selective TRPC6 positive allosteric modulator
6831 TRPV3 74a
Selective TRPV3 antagonist; brain penetrant
4639 TT 232
sst1 and sst4 agonist
0761 TTNPB
Retinoic acid analog; RAR agonist
4432 TTP 22
High affinity, selective CK2 inhibitor
4601 TUG 891
Potent and selective FFA4 (GPR120) agonist
4038 TW 37
Bcl-2 inhibitor; induces apoptosis
3835 TWS 119
GSK-3β inhibitor; induces neuronal differentiation in ESCs
5328 TY 52156
S1P3 receptor antagonist
2308 Tabimorelin hemifumarate
Potent, orally active ghrelin receptor agonist
4157 Tacalcitol
Synthetic vitamin D3 (Cat. No. 4156) analog
0965 Tacrine hydrochloride
Cholinesterase inhibitor
6311 Tadalafil
Potent and highly selective PDE5 inhibitor; orally bioavailable
6427 Tafluprost
Very high affinity FP receptor agonist
6430 Takinib
Potent and selective TAK1/MAP3K7 kinase inhibitor
3719 Talabostat mesylate
Potent DPP IV inhibitor; activates NLRP1b inflammasome
5032 Talampanel
Non-competitive non-NMDA iGluR antagonist
2510 Talniflumate
CaCC blocker and Cl-/HCO3- exchange inhibitor
3145 Talopram hydrochloride
Potent, selective inhibitor of noradrenalin transporters
4352 Talsupram hydrochloride
Selective inhibitor of noradrenalin transporters
2672 Taltirelin
Synthetic thyrotropin-releasing hormone analog
6342 Tamoxifen
Estrogen receptor partial agonist/antagonist
0999 Tamoxifen citrate
Estrogen receptor partial agonist/antagonist
3050 Tamsulosin hydrochloride
Selective α1A antagonist
2854 Tandospirone hydrochloride
Selective 5-HT1A partial agonist
4426 Tanshinone IIA
Inhibits NF-κB and AP-1 DNA binding. Displays antioxidant properties
6586 Targapremir 210
Inhibits formation of miR-210
5757 Tariquidar dihydrochloride
Potent P-glycoprotein (P-gp) inhibitor
7051 Tasquinimod
High affinity HDAC4 negative allosteric modulator; also binds S100A9; antiangiogenic
0209 Taurine
Non-selective, endogenous glycine receptor partial agonist
2305 Tautomycetin
Selective PP1 inhibitor
1097 Taxol
Promotes assembly and inhibits disassembly of microtubules
6267 Taxol Janelia Fluor ® 549
Yellow fluorescent taxol derivative; probe for microtubule staining
6266 Taxol Janelia Fluor® 646
Red fluorescent taxol derivative; probe for microtubule staining; protocol available
3997 Tazarotene
Receptor-selective retinoid; binds RAR-β and -γ
4613 Tegaserod maleate
5-HT4 partial agonist
3664 Teijin compound 1
Potent CCR2b antagonist
6658 Telaprevir
Hepatitis C virus (HCV) protease NS3/4A inhibitor
1122 Telenzepine dihydrochloride
Potent, selective M1 antagonist
5139 Telmisartan
AT1 antagonist; PPARγ partial agonist
2706 Temozolomide
DNA-methylating antitumor agent
3082 Tempol
Superoxide scavenger; antioxidant
5264 Temsirolimus
mTOR inhibitor; antitumor
2580 Tenidap
NSAID, cyclooxygenase (COX-1) inhibitor. Also opener of KIR2.3
3666 Tenofovir
Reverse transcriptase inhibitor
3365 Tenovin-1
Protects against MDM2-mediated p53 degradation
1506 Terazosin hydrochloride
α1 and α2B antagonist (α1 > α2B). Orally active
6484 Terbinafine hydrochloride
Selective K2P9.1 (TASK-3) activator; also inhibits fungal squalene epoxidase
3948 Terfenadine
H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker
5069 Teriflunomide
Inhibitor of DHODH; active metabolite of Leflunomide
1405 (-)-Terreic acid
Selective inhibitor of BTK
4339 Tertiapin LQ
Selective Kir1.1 blocker; derivative of tertiapin-Q (Cat. No. 1316)
1316 Tertiapin-Q
Selective blocker of inward-rectifier K+ channels
3965 Tesaglitazar
PPARα/γ agonist
2822 Testosterone
Endogenous androgen receptor agonist
2175 Tetrabenazine
Potent inhibitor of vesicular monoamine transport
3068 Tetraethylammonium chloride
Non-selective K+ channel blocker
0312 (RS)-(Tetrazol-5-yl)glycine
Highly potent NMDA agonist
0723 Tetrindole mesylate
MAO-A inhibitor
1078 Tetrodotoxin
Na+ channel blocker
1069 Tetrodotoxin citrate
Na+ channel blocker; citrate salt of tetrodotoxin (Cat. No. 1078)
0652 Thalidomide
Binds cereblon; also TNF-α synthesis inhibitor
6686 Thalidomide 4'-ether-PEG2-alkyne
Cereblon ligand with PEG linker and terminal alkyne for onward chemistry
6950 Thalidomide 4'-ether-PEG3-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6951 Thalidomide 4'-ether-PEG5-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
7329 Thalidomide 4'-ether-alkylC2-acid
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
6850 Thalidomide 4'-ether-alkylC2-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
7330 Thalidomide 4'-ether-alkylC3-acid
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7331 Thalidomide 4'-ether-alkylC4-acid
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
6917 Thalidomide 4'-ether-alkylC4-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
7332 Thalidomide 4'-ether-alkylC5-acid
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7333 Thalidomide 4'-ether-alkylC6-acid
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
6627 Thalidomide 4'-ether-alkylC6-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
7334 Thalidomide 4'-ether-alkylC7-acid
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7335 Thalidomide 4'-ether-alkylC8-acid
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
6966 Thalidomide 4'-oxyacetamide-PEG1-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6967 Thalidomide 4'-oxyacetamide-PEG2-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6467 Thalidomide 4'-oxyacetamide-PEG3-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6468 Thalidomide 4'-oxyacetamide-PEG4-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6913 Thalidomide 4'-oxyacetamide-alkylC1-PEG3-alkylC3-amine
Cereblon ligand with alkyl-PEG-alkyl linker and terminal amine for onward chemistry
6949 Thalidomide 4'-oxyacetamide-alkylC2-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
6469 Thalidomide 4'-oxyacetamide-alkylC4-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
6300 Thalidomide 4'-oxyacetamide-alkylC4-azide
Cereblon ligand with alkyl linker and terminal azide for onward chemistry
6968 Thalidomide 4'-oxyacetamide-alkylC6-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
6946 Thalidomide 4'-oxyacetamide-alkylC8-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
6685 Thalidomide, propargyl
Alkyne-functionalized Thalidomide; 'click' cereblon ligand for PROTACs
7288 Thalidomide-Cyanine 5
Fluorescent cereblon probe
1138 Thapsigargin
Potent inhibitor of SERCA ATPase
2795 Theophylline
Adenosine receptor antagonist; bronchodilator
4390 Thiamet G
Potent O-GlcNAcase inhibitor
3845 Thiazovivin
ROCK inhibitor ; improves the efficiency of fibroblast reprogramming and induction of iPSCs
3280 2-ThioUTP tetrasodium salt
Potent and selective P2Y2 agonist
4061 6-Thioguanine
Anticancer and immunosuppressive agent
1567 Thiolutin
Bacterial RNA polymerase inhibitor
0644 Thioperamide
H3 antagonist; also H4 inverse agonist
3070 Thioridazine hydrochloride
Dopamine receptor antagonist; antipsychotic
3267 Thiostrepton
Antibiotic, inhibits protein synthesis
7005 4-Thiouridine
Photoreactive uridine analog for RNA sequencing
1185 Thrombin Receptor Agonist Peptide
Causes platelet aggregation and secretion
3390 Thymosin β4
Potent actin polymerization regulator
4256 Tiagabine hydrochloride
Selective GAT-1 inhibitor; anticonvulsant
1972 Tianeptine sodium salt
Selective facilitator of 5-HT uptake; antidepressant
6864 Ticagrelor
High affinity and reversible P2Y12 antagonist; displays inverse agonism in vitro; also inhibits ENT1
5579 Tilfrinib
Potent and selective breast tumor kinase (Brk) inhibitor
0649 (S)-Timolol maleate
β1 antagonist
0747 Tin protoporphyrin IX dichloride
Heme oxygenase inhibitor
0826 Tiotidine
Potent and selective H2 antagonist
5902 Tiotropium bromide
Potent muscarinic receptor antagonist
6410 Tipifarnib
Potent farnesyltransferase inhibitor; orally bioavailable
5565 Tiplaxtinin
Plasminogen activator inhibitor-1 (PAI-1) inhibitor
3609 Tizanidine hydrochloride
α2 agonist
5390 Tobramycin
Aminoglycoside antibiotic
3909 Toceranib
Potent PDGFR and VEGFR inhibitor
2540 Tocrifluor T1117
Novel fluorescent cannabinoid ligand; fluorescent form of AM 251 (Cat. No. 1117)
7150 Tocriscreen 2.0 Max
Bioactive compound library for high-throughput screening, high-content screening and chemical biology applications; comprised of 1280 biologically active compounds (250 μL 10 mM DMSO solutions)
7152 Tocriscreen 2.0 Micro
Bioactive compound library for high-throughput screening, high-content screening and chemical biology applications; comprised of 1280 biologically active compounds (15 μL 10 mM DMSO solutions)
7151 Tocriscreen 2.0 Mini
Bioactive compound library for high-throughput screening, high-content screening and chemical biology applications; comprised of 1280 compounds (50 μL 10 mM DMSO solutions)
7350 Tocriscreen Antiviral Library
Antiviral compound library for high throughput screening, chemical biology applications and drug repurposing; contains 240 bioactive compounds (100 μL 10 mM DMSO solutions)
6801 Tocriscreen Epigenetics Library
A library of 101 epigenetic compounds (250 μL, 10 mM DMSO solutions) for high throughput screening, high content screening and chemical biology applications
7200 Tocriscreen FDA-Approved Drugs Library
Drug repurposing library; a library of 190 compounds equivalent to active components of drug formulations approved by the FDA (100 μL 10 mM DMSO solutions)
6268 Tocriscreen Kinase Inhibitor Library
A bioactive compound library of 160 kinase inhibitors (250 μL 10 mM DMSO solutions) for high-throughput screening, high-content screening and chemical biology applications
6555 TokeOni
NIR-emission luciferin analog; ideal for deep tissue applications; orally bioavailable and brain penetrant
5864 Tolcapone
COMT inhibitor; also inhibits transthyretin aggregation
5181 Tolvaptan
Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active
2011 Tomoxetine hydrochloride
Potent and selective noradrenalin re-uptake inhibitor
3620 Topiramate
GluK1 antagonist; inhibits carbonic anhydrase (CA) II and IV; also positive allosteric modulator of GABAA receptors
4562 Topotecan hydrochloride
DNA topoisomerase I inhibitor; Camptothecin (Cat. No. 1100) analog
4184 Torcetrapib
Inhibitor of cholesteryl ester transfer protein (CETP)
4247 Torin 1
Potent and selective mTOR inhibitor
4248 Torin 2
Potent and selective mTOR inhibitor
5270 Toyocamycin
Adenosine analog; antifungal antibiotic
1558 Tracazolate hydrochloride
Allosteric modulator of GABAA receptors
3619 Tramiprosate
Targets soluble Aβ to decrease amyloid plaque deposition. Also GABA analog
1098 Tranilast
Antiallergic; inhibits inflammatory mediator release from mast cells
3852 Tranylcypromine hydrochloride
Irreversible inhibitor of LSD1; also inhibits MAO
2508 Trap 101
Potent and selective NOP antagonist; active in vivo
4218 Travaprost
Potent and selective FP prostaglandin receptor agonist
6336 Trazodone hydrochloride
5-HT2A and α1 adrenoceptor antagonist; also enhances neural differentiation; antidepressant and neuroprotectant
5349 Treprostinil
Potent prostacyclin (PGI2) analog
2337 Trequinsin hydrochloride
Highly potent PDE3 inhibitor
2472 Triacsin C
Inhibitor of acyl-CoA synthetase
1406 Trichostatin A
Potent histone deacetylase inhibitor
4460 Trifluorothymidine
Thymidylate synthetase inhibitor
3859 6,2',4'-Trimethoxyflavone
Aryl hydrocarbon receptor antagonist
0662 trans-Triprolidine hydrochloride
Highly potent H1 antagonist
3253 Triptolide
Inhibits RNAPII-mediated transcription; antitumor, anti-inflammatory and immunosuppressive
2191 S-Trityl-L-cysteine
Potent, selective inhibitor of mitotic kinesin Eg5
3114 Troglitazone
Selective PPARγ agonist; antidiabetic agent
6002 Trolox
Antifade reagent; antioxidant vitamin E derivative; cell permeable and water soluble
0641 Tropanyl-3,5-dimethylbenzoate
5-HT3 antagonist
0909 Tropicamide
Selective M4 antagonist
2459 Tropisetron hydrochloride
Potent 5-HT3 antagonist; also α7 nAChR partial agonist
3863 Trovafloxacin mesylate
Antibiotic; inhibits bacterial DNA synthesis
3402 Tubacin
HDAC6 inhibitor; inhibits a-tubulin deacetylation
6270 Tubastatin A hydrochloride
Potent HDAC6 inhibitor
2820 (+)-Tubocurarine chloride
nAChR antagonist
3516 Tunicamycin
Antibiotic; GlcNAc phosphotransferase inhibitor
0579 Tyrphostin B44, (+) enantiomer
EGFR-kinase inhibitor

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