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Displaying Products by Catalog Number (5900 - 5999)

Cat. No. Product Name / Activity
5900 c-Di-GMP sodium salt
Endogenous STING and DDX41 agonist; activates STING-dependent signaling
5901 c-Di-AMP sodium salt
Endogenous STING and DDX41 agonist; activates STING-dependent signaling
5902 Tiotropium bromide
Potent muscarinic receptor antagonist
5903 CATPB
FFA2 (GPR43) inverse agonist
5904 Montelukast sodium
CysLT1 and GPR17 antagonist
5906 Imatinib mesylate
Potent and selective v-Abl tyrosine kinase inhibitor; also inhibits PDGFR and c-kit
5907 VX 680
High affinity and selective Aurora kinase inhibitor
5908 Bis-ANS
Fluorescent probe for nonpolar cavities in proteins; used to detect Aβ fibres
5909 RMM 46
MSK/RSK family kinase inhibitor
5910 TL4-12
Potent MAP4K2 (GCK) inhibitor
5911 FFN 200 dihydrochloride
Selective fluorescent VMAT2 substrate
5913 Ro 6842262
Potent LPA1 antagonist
5914 AM 0902
Potent and selective TRPA1 antagonist
5915 PF 04449613
Potent PDE9 inhibitor; brain penetrant
5916 Canertinib dihydrochloride
Potent EGFR kinase inhibitor
5917 PF 9184
Potent microsomal prostaglandin E synthase 1 (mPGES-1) inhibitor
5918 TPPU
Potent soluble epoxide hydrolase inhibitor; orally bioavailable and brain penetrant
5919 PI 3065
Potent and selective PI 3-kinase p110δ inhibitor
5920 LG 100268
Potent and selective RXR agonist; also activates RXR/PPARγ heterodimers
5921 D9
Potent thioredoxin reductase (TrxR) inhibitor
5922 CRT 0066854 hydrochloride
PKCι and PKCζ inhibitor
5924 ER 819762
Potent EP4 receptor antagonist; orally bioavailable
5928 RS 09
TLR4 peptide agonist; acts as an adjuvant in vivo
5929 BeKm 1
Potent and selective KV11.1 (hERG) channel blocker
5930 PBIT
JARID1 (Jumonji AT-Rich Interactive Domain 1) inhibitor
5931 PF 05089771
Potent and selective Nav1.7 channel blocker
5934 NCT 501 hydrochloride
Potent and selective ALDH1A1 inhibitor
5935 H2DCFDA
Fluorescent ROS indicator; cell permeable
5937 A 779
Selective Mas receptor (Ang-(1-7) receptor) antagonist
5938 Mambalgin 1
Selective ASIC1a inhibitor; analgesic
5939 PF 6274484
High affinity and potent covalent EGFR kinase inhibitor
5940 AdTx1
Selective, high affinity, non-competitive α1A adrenoceptor antagonist
5941 OD1
Potent hNav1.4, rNav1.6 and rNav1.7 channel activator
5943 ML 339
Potent and selective hCXCR6 antagonist
5944 G10
Activator of STING-dependent signaling
5945 2',3'-cGAMP sodium salt
Endogenous high affinity STING agonist
5946 3',3'-cGAMP sodium salt
STING agonist
5948 DMNPE-4 AM-caged-calcium
Caged calcium; cell permeable
5951 WAY 252623
Potent LXR agonist
5952 PDD 00017273
Potent and selective PARG inhibitor; cell permeable
5953 Adaptaquin
HIF-prolyl hydroxylase-2 (PHD2) inhibitor; antioxidant
5954 MSG 606
Potent human MC1 receptor antagonist; also MC3 and MC5 partial agonist
5955 eCF 309
Potent mTOR inhibitor
5956 NF 1819
Potent and selective irreversible MAGL inhibitor; membrane permeable and brain penetrant
5957 C3
Selective microsomal prostaglandin E synthase 1 (mPGES-1) inhibitor
5958 Desloratadine
High affinity H1 antagonist; anti-inflammatory
5959 Autocamtide-2-related inhibitory peptide, myristoylated
CaM kinase II inhibitor; enhanced cell permeable derivative of Autocamtide-2-related inhibitory peptide
5960 TMI 1
Adam 17 (TACE) and MMP inhibitor; orally bioavailable
5961 HIOC
Selective TrkB receptor agonist; neuroprotectant
5962 3-AP
Ribonucleotide reductase inhibitor; also an iron chelator
5963 CMPI hydrochloride
Potent positive allosteric modulator of α4β2 nAChRs; also inhibitor of (α4)2(β2)3, muscle-type and Torpedo nAChRs
5964 SI-2 hydrochloride
Steroid receptor coactivator 3 (SRC-3) inhibitor
5965 ISAM 140
High affinity A2B receptor antagonist
5966 ML 233
Non-peptide apelin agonist
5968 Ro 3280
Potent and selective PLK1 inhibitor
5969 (R)-CE3F4
Epac inhibitor; R-enantiomer of CE3F4 (Cat. No. 4793)
5970 BAY 299
Potent and selective BRD1 and TAF1 inhibitor
5973 CP 724714
Potent and selective ErbB2 inhibitor
5976 Ned K
NAADP signaling inhibitor
5978 WL 47 - dimer
High affinity caveolin-1 ligand
5979 Eicosapentaenoic Acid
Endogenous polyunsaturated fatty acid; stimulates ERK1/2 phosphorylation
5981 Itraconazole
SMO antagonist; acts at different binding site to cyclopamine (Cat No. 1623)
5982 cis-6-Hydroxynorketamine hydrochloride
Enhances AMPA currents: antidepressant
5983 BMS 986187
Potent positive allosteric modulator of δ receptors
5984 LY 2955303
High affinity and selective RARγ antagonist
5986 NAV 2729
Selective ARF6 inhibitor
5987 (±)-ML 209
RORγt inverse agonist; suppresses Th17 cell differentiation
5989 BIRB 796
High affinity and selective p38 kinase inhibitor
5991 BAY 598
Potent and selective SMYD2 inhibitor
5992 MM 54
Potent apelin antagonist
5993 CP 673451
Potent and selective PDGFR inhibitor
5994 Enzastaurin
Potent PKCβ inhibitor
5995 AMG 517
Potent TRPV1 antagonist
5996 (R)-Norketamine hydrochloride
NMDA receptor modulator; analgesic
5999 TP 472N
Negative control for TP 472

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