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Displaying Products by Catalog Number (2500 - 2599)

Cat. No. Product Name / Activity
2500 Bay 59-3074
CB1/CB2 receptor partial agonist
2501 Bay 36-7620
mGlu1 inverse agonist
2502 MRS 2693 trisodium salt
Selective P2Y6 agonist
2503 (-)-Bicuculline methiodide
GABAA antagonist; more water soluble version of (+)-bicuculline (Cat. No. 0130)
2504 Irsogladine maleate
PDE4 inhibitor; antiulcer agent
2505 Nonactin
Monovalent cation ionophore
2506 SSR 69071
Potent, orally active human leukocyte elastase inhibitor
2507 J 104129 fumarate
Potent and selective M3 antagonist
2508 Trap 101
Potent and selective NOP antagonist; active in vivo
2509 Cardamonin
Inhibitor of NF-κB activation; anti-inflammatory
2510 Talniflumate
CaCC blocker and Cl-/HCO3- exchange inhibitor
2511 APC 366
Tryptase inhibitor
2512 CGS 35066
Endothelin-converting enzyme (ECE) inhibitor
2513 Acyclovir
Inhibits viral DNA polymerase; antiherpetic agent
2514 L-161,982
Selective EP4 receptor antagonist
2517 RS 504393
Highly selective CCR2 chemokine receptor antagonist
2518 TC 1698 dihydrochloride
α7-selective agonist
2519 T 98475
GnRH receptor antagonist
2520 PD 166793
Broad spectrum MMP inhibitor
2521 NSC 3852
Histone deacetylase inhibitor
2522 YM 26734
Secretory phospholipase A2 (sPLA2) inhibitor
2524 A 205804
Selective inhibitor of E-selectin and ICAM-1 expression
2529 UFP 803
Urotensin-II (UT) antagonist
2530 PPDA
GluN2C/GluN2D-selective NMDA antagonist
2531 Ganaxolone
Potent positive allosteric modulator of GABAA receptors
2532 TFB-TBOA
High affinity EAAT1 and EAAT2 blocker
2533 DPO-1
Blocker of KV1.5 channel and IKur current
2536 Domperidone
Peripheral D2-like antagonist
2538 L-BMAA hydrochloride
Neurotoxic amino acid
2539 IKK 16
Selective inhibitor of IKK
2540 Tocrifluor T1117
Novel fluorescent cannabinoid ligand; fluorescent form of AM 251 (Cat. No. 1117)
2542 Ki 8751
Potent, selective VEGFR-2 inhibitor
2544 Nafarelin
GnRH receptor agonist
2545 Lofepramine
5-HT and NA reuptake inhibitor (SNRI)
2546 PKI 14-22 amide, myristoylated
Cell-permeable protein kinase A inhibitor
2547 6-Hydroxydopamine hydrobromide
Selective catecholaminergic neurotoxin
2548 NF 110
Potent P2X3 antagonist
2549 ZIP
Cell-permeable inhibitor of atypical PKC isozyme PKMζ
2550 SUN-B 8155
Non-peptide calcitonin agonist
2551 Calcitriol
Vitamin D receptor (VDR) agonist
2554 CD 1530
Potent and selective RARγ agonist
2555 GYKI 53655 hydrochloride
Non-competitive non-NMDA iGluR antagonist
2557 Phencyclidine hydrochloride
Non-competitive NMDA antagonist
2558 10-DEBC hydrochloride
Selective Akt/PKB inhibitor
2559 TPCA-1
Potent, selective inhibitor of IKKβ
2560 SB 218078
Chk1 inhibitor
2561 Calmidazolium chloride
Calmodulin antagonist
2562 PB 28 dihydrochloride
High affinity σ2 agonist
2563 Fexaramine
Potent, selective farnesoid X receptor (FXR) agonist
2564 AM 114
20S proteasome inhibitor
2565 ZK 756326
Selective, non-peptide CCR8 agonist
2566 Melanotan II
High affinity melanocortin receptor agonist
2567 PLP (139-151)
Encephalitogenic myelin proteolipid fragment
2568 MOG (35-55)
Encephalitogenic myelin oligodendrocyte glycoprotein fragment
2569 CGP 42112
Selective, high affinity AT2 ligand
2570 Kisspeptin 10 (human)
Endogenous ligand for kisspeptin receptor
2571 Amlodipine besylate
CaV1.x blocker
2573 PSB 069
Non-selective NTPDase inhibitor
2574 PSB 06126
NTPDase 3 inhibitor
2576 Hemokinin 1 (human)
Endogenous and selective NK1 agonist
2577 Cetirizine dihydrochloride
Selective H1 antagonist
2578 Benazepril hydrochloride
Angiotensin-converting enzyme (ACE) inhibitor
2580 Tenidap
NSAID, cyclooxygenase (COX-1) inhibitor. Also opener of KIR2.3
2581 PAC 1
Activator of procaspase-3; pro-apoptotic
2582 Lansoprazole
H+,K+-ATPase inhibitor
2583 Omeprazole
H+,K+-ATPase inhibitor
2584 α-MSH
Endogenous melanocortin receptor agonist
2585 Compstatin
C3-binding peptide; inhibits complement activation
2587 Neuropeptide S (human)
Endogenous Neuropeptide S receptor agonist
2591 TCS 359
Potent FLT3 inhibitor
2592 TCB-2
High affinity and potent 5-HT2A agonist
2595 J 113863
Potent CCR1 chemokine receptor antagonist
2596 Mexiletine hydrochloride
Na+ channel blocker; antiarrhythmic agent
2598 (±)-J 113397
Potent and selective NOP antagonist
2599 OSU 6162 hydrochloride
Dopamine stabilizer

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