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Displaying Products by Catalog Number (5100 - 5199)

Cat. No. Product Name / Activity
5100 TC-T 6000
Potent equilibrative nucleoside transporter 4 (ENT4) inhibitor
5101 PD 90780
Inhibits NGF binding to p75NTR
5102 PLX 647 dihydrochloride
Potent dual Fms/KIT inhibitor
5103 Lys-CoA
Selective p300 inhibitor
5106 GSK 2193874
Potent and selective TRPV4 antagonist; orally active
5107 GSK 2606414
Potent and selective PERK inhibitor; orally bioavailable
5108 TFC 007
Potent hematopoietic prostaglandin D synthase (H-PGDS) inhibitor
5109 SB 743921 hydrochloride
Potent kinesin spindle protein (KSP) inhibitor
5110 GSK 1562590 hydrochloride
High affinity, selective urotensin II (UT) receptor antagonist
5111 GSK 1838705
Potent IR and IGF1R inhibitor; also inhibits anaplastic lymphoma kinase (ALK)
5112 NS 9283
Positive allosteric modulator of α4β2 nAChRs
5113 AbK
Photo-crosslinking probe; unnatural amino acid
5115 OXA (17-33)
Potent and selective peptide OX1 agonist
5116 PACMA 31
Irreversible protein disulfide isomerase (PDI) inhibitor
5117 Hoechst 33342
Fluorescent dye for labeling DNA
5118 SynaptoRedTM C2
Fluorescent dye; stains synaptic vesicles
5119 Calcein AM
Cell permeable compound; hydrolyzed to become fluorescent in living cells
5121 3PO
PFKFB3 inhibitor
5122 Dansyl-NECA
Potent and selective fluorescent adenosine A1 agonist
5123 BMX-IN-1
Potent and irreversible BMX inhibitor
5124 PD 404182
High affinity inhibitor of KDO 8-P synthase; also DDAH1 inhibitor
5125 CKD 602
Topoisomerase I inhibitor
5126 iMDK
Suppressor of MDK expression; inhibits PI 3-K signaling
5127 P1
Protein disulfide isomerase (PDI) inhibitor
5128 C 21
Selective PRMT1 inhibitor
5129 TC-G 1005
Potent and selective GPBA receptor (TGR5) agonist
5130 CTCE 9908
CXCR4 antagonist; antitumor
5131 NAB 2
Protects against α-synuclein toxicity; promotes Rsp5/Nedd4-dependent endosomal transport
5132 UNC 0642
Potent and selective G9a and GLP inhibitor
5133 GKA 50
Glucokinase activator
5134 MRT 67307 dihydrochloride
Salt inducible kinase (SIK) inhibitor
5135 Propidium iodide
Red-fluorescent DNA stain; membrane impermeant to live cells. Pi staining differentiates live and dead cells
5136 Rizatriptan benzoate
Potent 5-HT1B and 5-HT1D agonist
5138 RSVA 405
AMPK activator; also STAT3 inhibitor
5139 Telmisartan
AT1 antagonist; PPARγ partial agonist
5140 GSK 2830371
Potent and selective allosteric inhibitor of Wip1 phosphatase
5141 AZD 5582 dihydrochloride
Dimeric Smac mimetic; potent IAP inhibitor
5142 Mps1-IN-1 dihydrochloride
Selective Mps1 kinase inhibitor
5143 Ononetin
TRPM3 blocker
5144 CFM 4
CARP-1 mimetic; proapoptotic
5145 AI-3
ARE activator; induces Nrf2-ARE-dependent transcription
5146 Sulforhodamine 101
Red fluorescent dye; selective astrocyte marker
5147 Istradefylline
Potent and selective A2A antagonist
5148 Wnt-C59
Highly potent PORCN inhibitor
5149 CX 614
Positive allosteric modulator of AMPA receptors
5150 NCL 00017509
Potent and reversible NIMA related kinase 2 (Nek2) inhibitor
5151 Prosaptide TX14(A)
Potent GPR37 and GPR37L1 agonist
5153 ML 240
ATP-competitive inhibitor of p97 ATPase
5154 HNGF6A
Humanin analog; increases insulin sensitivity
5155 SGI 1027
DNA methyltransferase inhibitor
5157 DMNPE-caged ATP diammonium salt
Caged ATP
5158 Morphine hydrochloride
Narcotic opioid analgesic
5160 Medetomidine hydrochloride
Potent and highly selective α2 agonist
5161 ML 154
Potent Neuropeptide S receptor antagonist
5163 A 366
Potent and selective G9a/GLP inhibitor
5164 CVT 10216
Potent and selective ALDH2 inhibitor
5166 Perhexiline maleate
Carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor
5167 Congo Red
Amyloid fibril binding dye; also a VGlut inhibitor
5168 Rose Bengal
Stains exposed epithelium in eye. Also VGlut and VMAT inhibitor
5169 Noradrenaline bitartrate
Endogenous adrenergic hormone and neurotransmitter
5171 NBOH-2C-CN hydrochloride
High affinity and selective 5-HT2A agonist
5172 FLI 06
Inhibitor of Notch signaling; disrupts Notch trafficking and processing
5173 MS 436
Potent and selective BRD4(1) inhibitor
5175 AEBSF
Broad spectrum, irreversible inhibitor of serine proteases
5177 WZ 4003
Potent and selective NUAK1/2 inhibitor
5178 ASP 7663
Selective TRPA1 activator
5179 TCID
Selective ubiquitin C-terminal hydrolase-L3 (UCH-L3) inhibitor
5180 Ferrostatin 1
Selective inhibitor of erastin induced ferroptosis
5181 Tolvaptan
Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active
5182 OXA 06 dihydrochloride
Potent ROCK inhibitor
5183 ETP 45835 dihydrochloride
Mnk1 and Mnk2 inhibitor
5184 BDS I
Potent and reversible Kv3.4 potassium channel blocker; neuroprotective
5185 JTE 607 dihydrochloride
Cytokine release inhibitor; anti-inflammatory
5186 Neuropathiazol
Selective inducer of neuronal differentiation in hippocampal neural progenitors
5188 S 07662
Constitutive androstane receptor (CAR) inverse agonist
5189 GSK 2837808A
Potent, selective LDHA inhibitor
5190 FRAX 486
Potent PAK inhibitor; brain penetrant and orally bioavailable
5191 PTC 209
Bmi-1 inhibitor; antitumor
5192 NBI 31772
High affinity insulin-like growth factor-I binding protein IGFBP inhibitor
5193 Remodelin
N-acetyltransferase 10 (NAT10) inhibitor
5195 Agitoxin 2
Potent Shaker K+ channel blocker
5196 PMX 205
Potent C5a receptor peptide antagonist
5197 Spautin 1
USP10 and USP13 inhibitor; inhibits autophagy
5198 AZ 20
Potent and selective ATR kinase inhibitor; antitumor
5199 AZD 7762 hydrochloride
Potent and selective ATP-competitive inhibitor of Chk1 and Chk2; also enhances CRISPR-Cpf1-mediated genome editing

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