All ProductsDisplaying Products by Catalog Number (5100 - 5199)
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| Cat. No. | Product Name / Activity |
|---|---|
| 5101 | PD 90780 |
| Inhibits NGF binding to p75NTR | |
| 5106 | GSK 2193874 |
| Potent and selective TRPV4 antagonist; orally active | |
| 5107 | GSK 2606414 |
| Potent and selective PERK inhibitor; orally bioavailable | |
| 5108 | TFC 007 |
| Potent hematopoietic prostaglandin D synthase (H-PGDS) inhibitor | |
| 5110 | GSK 1562590 hydrochloride |
| High affinity, selective urotensin II (UT) receptor antagonist | |
| 5111 | GSK 1838705 |
| Potent IR and IGF1R inhibitor; also inhibits anaplastic lymphoma kinase (ALK) | |
| 5112 | NS 9283 |
| Positive allosteric modulator of α4β2 nAChRs | |
| 5113 | AbK |
| Photo-crosslinking probe; unnatural amino acid | |
| 5114 | K34c |
| Potent and selective α5β1 integrin inhibitor | |
| 5115 | OXA (17-33) |
| Potent and selective peptide OX1 agonist | |
| 5116 | PACMA 31 |
| Irreversible protein disulfide isomerase (PDI) inhibitor | |
| 5117 | Hoechst 33342 |
| Fluorescent dye for staining DNA | |
| 5118 | SynaptoRedTM C2 |
| Fluorescent dye; stains synaptic vesicles | |
| 5119 | Calcein AM |
| Cell permeable compound; hydrolyzed to become fluorescent in living cells | |
| 5121 | 3PO |
| PFKFB3 inhibitor | |
| 5123 | BMX-IN-1 |
| Potent and irreversible BMX inhibitor | |
| 5126 | iMDK |
| Suppressor of MDK expression; inhibits PI 3-K signaling | |
| 5127 | P1 |
| Protein disulfide isomerase (PDI) inhibitor | |
| 5128 | C 21 |
| Selective PRMT1 inhibitor | |
| 5129 | TC-G 1005 |
| Potent and selective GPBA receptor (TGR5) agonist | |
| 5130 | CTCE 9908 |
| CXCR4 antagonist; antitumor | |
| 5131 | NAB 2 |
| Protects against α-synuclein toxicity; promotes Rsp5/Nedd4-dependent endosomal transport | |
| 5132 | UNC 0642 |
| Potent and selective G9a and GLP inhibitor | |
| 5133 | GKA 50 |
| Glucokinase activator | |
| 5134 | MRT 67307 dihydrochloride |
| Salt inducible kinase (SIK) inhibitor | |
| 5135 | Propidium iodide |
| Red-fluorescent DNA stain; membrane impermeant to live cells. Pi staining differentiates live and dead cells | |
| 5136 | Rizatriptan benzoate |
| Potent 5-HT1B and 5-HT1D agonist | |
| 5139 | Telmisartan |
| AT1 antagonist; PPARγ partial agonist | |
| 5140 | GSK 2830371 |
| Potent and selective allosteric inhibitor of Wip1 phosphatase | |
| 5141 | AZD 5582 dihydrochloride |
| Dimeric Smac mimetic; potent IAP inhibitor | |
| 5142 | Mps1-IN-1 dihydrochloride |
| Selective Mps1 kinase inhibitor | |
| 5143 | Ononetin |
| TRPM3 blocker | |
| 5146 | Sulforhodamine 101 |
| Red fluorescent dye; selective astrocyte marker | |
| 5147 | Istradefylline |
| Potent and selective A2A antagonist | |
| 5148 | Wnt-C59 |
| Highly potent PORCN inhibitor | |
| 5149 | CX 614 |
| Positive allosteric modulator of AMPA receptors | |
| 5150 | NCL 00017509 |
| Potent and reversible NIMA related kinase 2 (Nek2) inhibitor | |
| 5151 | Prosaptide TX14(A) |
| Potent GPR37 and GPR37L1 agonist | |
| 5153 | ML 240 |
| ATP-competitive inhibitor of p97 ATPase | |
| 5155 | SGI 1027 |
| DNA methyltransferase inhibitor | |
| 5157 | DMNPE-caged ATP diammonium salt |
| Caged ATP | |
| 5158 | Morphine hydrochloride |
| Narcotic opioid analgesic | |
| 5160 | Medetomidine hydrochloride |
| Potent and highly selective α2 agonist | |
| 5161 | ML 154 |
| Potent Neuropeptide S receptor antagonist | |
| 5163 | A 366 |
| Potent and selective G9a/GLP inhibitor | |
| 5164 | CVT 10216 |
| Potent and selective ALDH2 inhibitor | |
| 5166 | Perhexiline maleate |
| Carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor | |
| 5167 | Congo Red |
| Amyloid fibril binding dye; also a VGlut inhibitor | |
| 5168 | Rose Bengal |
| Stains exposed epithelium in eye. Also VGlut and VMAT inhibitor | |
| 5169 | Noradrenaline bitartrate |
| Endogenous adrenergic hormone and neurotransmitter | |
| 5171 | NBOH-2C-CN hydrochloride |
| High affinity and selective 5-HT2A agonist | |
| 5172 | FLI 06 |
| Inhibitor of Notch signaling; disrupts Notch trafficking and processing | |
| 5173 | MS 436 |
| Potent and selective BRD4(1) inhibitor | |
| 5175 | AEBSF |
| Broad spectrum, irreversible inhibitor of serine proteases | |
| 5177 | WZ 4003 |
| Potent and selective NUAK1/2 inhibitor | |
| 5178 | ASP 7663 |
| Selective TRPA1 activator | |
| 5179 | TCID |
| Selective ubiquitin C-terminal hydrolase-L3 (UCH-L3) inhibitor | |
| 5180 | Ferrostatin 1 |
| Selective inhibitor of erastin induced ferroptosis | |
| 5181 | Tolvaptan |
| Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active | |
| 5182 | OXA 06 dihydrochloride |
| Potent ROCK inhibitor | |
| 5183 | ETP 45835 dihydrochloride |
| Mnk1 and Mnk2 inhibitor | |
| 5185 | JTE 607 dihydrochloride |
| Active metabolite binds CPSF3; Pro-drug | |
| 5186 | Neuropathiazol |
| Selective inducer of neuronal differentiation in hippocampal neural progenitors | |
| 5188 | S 07662 |
| Constitutive androstane receptor (CAR) inverse agonist | |
| 5189 | GSK 2837808A |
| Potent and selective LDHA inhibitor | |
| 5190 | FRAX 486 |
| Potent PAK inhibitor; brain penetrant and orally bioavailable | |
| 5191 | PTC 209 |
| Bmi-1 inhibitor; antitumor | |
| 5192 | NBI 31772 |
| High affinity insulin-like growth factor-I binding protein IGFBP inhibitor | |
| 5193 | Remodelin |
| N-acetyltransferase 10 (NAT10) inhibitor | |
| 5196 | PMX 205 |
| Potent C5a receptor peptide antagonist | |
| 5197 | Spautin 1 |
| USP10 and USP13 inhibitor; inhibits autophagy | |
| 5198 | AZ 20 |
| Potent and selective ATR kinase inhibitor; antitumor | |
| 5199 | AZD 7762 hydrochloride |
| Potent and selective ATP-competitive inhibitor of Chk1 and Chk2; also enhances CRISPR-Cpf1-mediated genome editing |