Cat. No. | Product Name / Activity |
---|---|
5101 | PD 90780 |
Inhibits NGF binding to p75NTR | |
5106 | GSK 2193874 |
Potent and selective TRPV4 antagonist; orally active | |
5107 | GSK 2606414 |
Potent and selective PERK inhibitor; orally bioavailable | |
5108 | TFC 007 |
Potent hematopoietic prostaglandin D synthase (H-PGDS) inhibitor | |
5110 | GSK 1562590 hydrochloride |
High affinity, selective urotensin II (UT) receptor antagonist | |
5111 | GSK 1838705 |
Potent IR and IGF1R inhibitor; also inhibits anaplastic lymphoma kinase (ALK) | |
5112 | NS 9283 |
Positive allosteric modulator of α4β2 nAChRs | |
5113 | AbK |
Photo-crosslinking probe; unnatural amino acid | |
5114 | K34c |
Potent and selective α5β1 integrin inhibitor | |
5115 | OXA (17-33) |
Potent and selective peptide OX1 agonist | |
5116 | PACMA 31 |
Irreversible protein disulfide isomerase (PDI) inhibitor | |
5117 | Hoechst 33342 |
Fluorescent dye for staining DNA | |
5118 | SynaptoRedTM C2 |
Fluorescent dye; stains synaptic vesicles | |
5119 | Calcein AM |
Cell permeable compound; hydrolyzed to become fluorescent in living cells | |
5121 | 3PO |
PFKFB3 inhibitor | |
5123 | BMX-IN-1 |
Potent and irreversible BMX inhibitor | |
5126 | iMDK |
Suppressor of MDK expression; inhibits PI 3-K signaling | |
5127 | P1 |
Protein disulfide isomerase (PDI) inhibitor | |
5128 | C 21 |
Selective PRMT1 inhibitor | |
5129 | TC-G 1005 |
Potent and selective GPBA receptor (TGR5) agonist | |
5130 | CTCE 9908 |
CXCR4 antagonist; antitumor | |
5131 | NAB 2 |
Protects against α-synuclein toxicity; promotes Rsp5/Nedd4-dependent endosomal transport | |
5132 | UNC 0642 |
Potent and selective G9a and GLP inhibitor | |
5133 | GKA 50 |
Glucokinase activator | |
5134 | MRT 67307 dihydrochloride |
Salt inducible kinase (SIK) inhibitor | |
5135 | Propidium iodide |
Red-fluorescent DNA stain; membrane impermeant to live cells. Pi staining differentiates live and dead cells | |
5136 | Rizatriptan benzoate |
Potent 5-HT1B and 5-HT1D agonist | |
5139 | Telmisartan |
AT1 antagonist; PPARγ partial agonist | |
5140 | GSK 2830371 |
Potent and selective allosteric inhibitor of Wip1 phosphatase | |
5141 | AZD 5582 dihydrochloride |
Dimeric Smac mimetic; potent IAP inhibitor | |
5142 | Mps1-IN-1 dihydrochloride |
Selective Mps1 kinase inhibitor | |
5143 | Ononetin |
TRPM3 blocker | |
5146 | Sulforhodamine 101 |
Red fluorescent dye; selective astrocyte marker | |
5147 | Istradefylline |
Potent and selective A2A antagonist | |
5148 | Wnt-C59 |
Highly potent PORCN inhibitor | |
5149 | CX 614 |
Positive allosteric modulator of AMPA receptors | |
5150 | NCL 00017509 |
Potent and reversible NIMA related kinase 2 (Nek2) inhibitor | |
5151 | Prosaptide TX14(A) |
Potent GPR37 and GPR37L1 agonist | |
5153 | ML 240 |
ATP-competitive inhibitor of p97 ATPase | |
5155 | SGI 1027 |
DNA methyltransferase inhibitor | |
5157 | DMNPE-caged ATP diammonium salt |
Caged ATP | |
5158 | Morphine hydrochloride |
Narcotic opioid analgesic | |
5160 | Medetomidine hydrochloride |
Potent and highly selective α2 agonist | |
5161 | ML 154 |
Potent Neuropeptide S receptor antagonist | |
5163 | A 366 |
Potent and selective G9a/GLP inhibitor | |
5164 | CVT 10216 |
Potent and selective ALDH2 inhibitor | |
5166 | Perhexiline maleate |
Carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor | |
5167 | Congo Red |
Amyloid fibril binding dye; also a VGlut inhibitor | |
5168 | Rose Bengal |
Stains exposed epithelium in eye. Also VGlut and VMAT inhibitor | |
5169 | Noradrenaline bitartrate |
Endogenous adrenergic hormone and neurotransmitter | |
5171 | NBOH-2C-CN hydrochloride |
High affinity and selective 5-HT2A agonist | |
5172 | FLI 06 |
Inhibitor of Notch signaling; disrupts Notch trafficking and processing | |
5173 | MS 436 |
Potent and selective BRD4(1) inhibitor | |
5175 | AEBSF |
Broad spectrum, irreversible inhibitor of serine proteases | |
5177 | WZ 4003 |
Potent and selective NUAK1/2 inhibitor | |
5178 | ASP 7663 |
Selective TRPA1 activator | |
5179 | TCID |
Selective ubiquitin C-terminal hydrolase-L3 (UCH-L3) inhibitor | |
5180 | Ferrostatin 1 |
Selective inhibitor of erastin induced ferroptosis | |
5181 | Tolvaptan |
Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active | |
5182 | OXA 06 dihydrochloride |
Potent ROCK inhibitor | |
5183 | ETP 45835 dihydrochloride |
Mnk1 and Mnk2 inhibitor | |
5185 | JTE 607 dihydrochloride |
Active metabolite binds CPSF3; Pro-drug | |
5186 | Neuropathiazol |
Selective inducer of neuronal differentiation in hippocampal neural progenitors | |
5188 | S 07662 |
Constitutive androstane receptor (CAR) inverse agonist | |
5189 | GSK 2837808A |
Potent and selective LDHA inhibitor | |
5190 | FRAX 486 |
Potent PAK inhibitor; brain penetrant and orally bioavailable | |
5191 | PTC 209 |
Bmi-1 inhibitor; antitumor | |
5192 | NBI 31772 |
High affinity insulin-like growth factor-I binding protein IGFBP inhibitor | |
5193 | Remodelin |
N-acetyltransferase 10 (NAT10) inhibitor | |
5196 | PMX 205 |
Potent C5a receptor peptide antagonist | |
5197 | Spautin 1 |
USP10 and USP13 inhibitor; inhibits autophagy | |
5198 | AZ 20 |
Potent and selective ATR kinase inhibitor; antitumor | |
5199 | AZD 7762 hydrochloride |
Potent and selective ATP-competitive inhibitor of Chk1 and Chk2; also enhances CRISPR-Cpf1-mediated genome editing |