All Products

Displaying Products by Catalog Number (5100 - 5199)

Cat. No. Product Name / Activity
5106 GSK 2193874
Potent and selective TRPV4 antagonist; orally active
5107 GSK 2606414
Potent and selective PERK inhibitor; orally bioavailable
5108 TFC 007
Potent hematopoietic prostaglandin D synthase (H-PGDS) inhibitor
5109 SB 743921 hydrochloride
Potent kinesin spindle protein (KSP) inhibitor
5110 GSK 1562590 hydrochloride
High affinity, selective urotensin II (UT) receptor antagonist
5111 GSK 1838705
Potent IR and IGF1R inhibitor; also inhibits anaplastic lymphoma kinase (ALK)
5112 NS 9283
Positive allosteric modulator of α4β2 nAChRs
5113 AbK
Photo-crosslinking probe; unnatural amino acid
5114 K34c
Potent and selective α5β1 integrin inhibitor
5115 OXA (17-33)
Potent and selective peptide OX1 agonist
5116 PACMA 31
Irreversible protein disulfide isomerase (PDI) inhibitor
5117 Hoechst 33342
Blue-fluorescent dye for DNA staining. Cell permeable. Used for: nuclear counterstain, apoptosis analysis, fixed and live-cell staining. Application: flow cytometry, confocal microscopy
5118 SynaptoRedTM C2
Fluorescent dye. Used for: synaptic vesicles staining. Application: fluorescence microscopy
5119 Calcein AM
Cell permeable non-fluorescent compound; green-fluorescent in living cells once hydrolyzed. Used for: cell tracing and cell viability monitoring. Application: fluorescent microscopy and flow cytometry
5121 3PO
PFKFB3 inhibitor
5126 iMDK
Suppressor of MDK expression; inhibits PI 3-K signaling
5129 TC-G 1005
Potent and selective GPBA receptor (TGR5) agonist
5130 CTCE 9908
CXCR4 antagonist; antitumor
5132 UNC 0642
Potent and selective G9a and GLP inhibitor
5133 GKA 50
Glucokinase activator
5134 MRT 67307 dihydrochloride
Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor
5135 Propidium iodide
Red-fluorescent DNA stain, membrane impermeant to live cells. Used for: apoptosis detection, nuclear counterstaining, viability staining. Application: flow cytometry, confocal microscopy, fluorescence microscopy
5140 GSK 2830371
Potent and selective allosteric inhibitor of Wip1 phosphatase
5141 AZD 5582 dihydrochloride
Dimeric Smac mimetic; potent IAP inhibitor
5143 Ononetin
TRPM3 blocker
5146 Sulforhodamine 101
Red fluorescent dye; selective astrocyte marker
5147 Istradefylline
Potent and selective A2A antagonist
5148 Wnt-C59
Highly potent PORCN inhibitor
5149 CX 614
Positive allosteric modulator of AMPA receptors
5150 NCL 00017509
Potent and reversible NIMA related kinase 2 (Nek2) inhibitor
5151 Prosaptide TX14(A)
Potent GPR37 and GPR37L1 agonist
5153 ML 240
ATP-competitive inhibitor of p97 ATPase
5157 DMNPE-caged ATP diammonium salt
Caged ATP
5158 Morphine hydrochloride
Narcotic opioid analgesic
5160 Medetomidine hydrochloride
Potent and highly selective α2 agonist
5163 A 366
Potent and selective G9a/GLP inhibitor
5164 CVT 10216
Potent and selective ALDH2 inhibitor
5166 Perhexiline maleate
Carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor
5169 Noradrenaline bitartrate
Endogenous adrenergic hormone and neurotransmitter
5171 NBOH-2C-CN hydrochloride
High affinity and selective 5-HT2A agonist
5175 AEBSF
Broad spectrum, irreversible inhibitor of serine proteases
5177 WZ 4003
Potent and selective NUAK1/2 inhibitor
5178 ASP 7663
Selective TRPA1 activator
5180 Ferrostatin 1
Selective inhibitor of erastin induced ferroptosis
5181 Tolvaptan
Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active
5182 OXA 06 dihydrochloride
Potent ROCK inhibitor
5185 JTE 607 dihydrochloride
Active metabolite binds CPSF3; Pro-drug
5189 GSK 2837808A
Potent and selective LDHA inhibitor
5190 FRAX 486
Potent PAK inhibitor; brain penetrant and orally bioavailable
5192 NBI 31772
High affinity insulin-like growth factor-I binding protein IGFBP inhibitor
5193 Remodelin
N-acetyltransferase 10 (NAT10) inhibitor
5196 PMX 205
Potent C5a receptor peptide antagonist
5197 Spautin 1
USP10 and USP13 inhibitor; inhibits autophagy
5198 AZ 20
Potent and selective ATR kinase inhibitor; antitumor
5199 AZD 7762 hydrochloride
Potent and selective ATP-competitive inhibitor of Chk1 and Chk2; also enhances CRISPR-Cpf1-mediated genome editing

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