All Products

Displaying Products by Catalog Number (5100 - 5199)

Cat. No. Product Name / Activity
5101 PD 90780
Inhibits NGF binding to p75NTR
5106 GSK 2193874
Potent and selective TRPV4 antagonist; orally active
5107 GSK 2606414
Potent and selective PERK inhibitor; orally bioavailable
5108 TFC 007
Potent hematopoietic prostaglandin D synthase (H-PGDS) inhibitor
5110 GSK 1562590 hydrochloride
High affinity, selective urotensin II (UT) receptor antagonist
5111 GSK 1838705
Potent IR and IGF1R inhibitor; also inhibits anaplastic lymphoma kinase (ALK)
5112 NS 9283
Positive allosteric modulator of α4β2 nAChRs
5113 AbK
Photo-crosslinking probe; unnatural amino acid
5114 K34c
Potent and selective α5β1 integrin inhibitor
5115 OXA (17-33)
Potent and selective peptide OX1 agonist
5116 PACMA 31
Irreversible protein disulfide isomerase (PDI) inhibitor
5117 Hoechst 33342
Blue-fluorescent dye for DNA staining. Cell permeable. Used for: nuclear counterstain, apoptosis analysis, fixed and live-cell staining. Application: flow cytometry, confocal microscopy
5118 SynaptoRedTM C2
Fluorescent dye; stains synaptic vesicles
5119 Calcein AM
Cell permeable compound; hydrolyzed to become fluorescent in living cells
5121 3PO
PFKFB3 inhibitor
5123 BMX-IN-1
Potent and irreversible BMX inhibitor
5126 iMDK
Suppressor of MDK expression; inhibits PI 3-K signaling
5127 P1
Protein disulfide isomerase (PDI) inhibitor
5129 TC-G 1005
Potent and selective GPBA receptor (TGR5) agonist
5130 CTCE 9908
CXCR4 antagonist; antitumor
5131 NAB 2
Protects against α-synuclein toxicity; promotes Rsp5/Nedd4-dependent endosomal transport
5132 UNC 0642
Potent and selective G9a and GLP inhibitor
5133 GKA 50
Glucokinase activator
5134 MRT 67307 dihydrochloride
Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor
5135 Propidium iodide
Red-fluorescent DNA stain; membrane impermeant to live cells. PI staining differentiates live and dead cells
5140 GSK 2830371
Potent and selective allosteric inhibitor of Wip1 phosphatase
5141 AZD 5582 dihydrochloride
Dimeric Smac mimetic; potent IAP inhibitor
5142 Mps1-IN-1 dihydrochloride
Selective Mps1 kinase inhibitor
5143 Ononetin
TRPM3 blocker
5146 Sulforhodamine 101
Red fluorescent dye; selective astrocyte marker
5147 Istradefylline
Potent and selective A2A antagonist
5148 Wnt-C59
Highly potent PORCN inhibitor
5149 CX 614
Positive allosteric modulator of AMPA receptors
5150 NCL 00017509
Potent and reversible NIMA related kinase 2 (Nek2) inhibitor
5151 Prosaptide TX14(A)
Potent GPR37 and GPR37L1 agonist
5153 ML 240
ATP-competitive inhibitor of p97 ATPase
5155 SGI 1027
DNA methyltransferase inhibitor
5157 DMNPE-caged ATP diammonium salt
Caged ATP
5158 Morphine hydrochloride
Narcotic opioid analgesic
5160 Medetomidine hydrochloride
Potent and highly selective α2 agonist
5161 ML 154
Potent Neuropeptide S receptor antagonist
5163 A 366
Potent and selective G9a/GLP inhibitor
5164 CVT 10216
Potent and selective ALDH2 inhibitor
5166 Perhexiline maleate
Carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor
5169 Noradrenaline bitartrate
Endogenous adrenergic hormone and neurotransmitter
5171 NBOH-2C-CN hydrochloride
High affinity and selective 5-HT2A agonist
5173 MS 436
Potent and selective BRD4(1) inhibitor
5175 AEBSF
Broad spectrum, irreversible inhibitor of serine proteases
5177 WZ 4003
Potent and selective NUAK1/2 inhibitor
5178 ASP 7663
Selective TRPA1 activator
5179 TCID
Selective ubiquitin C-terminal hydrolase-L3 (UCH-L3) inhibitor
5180 Ferrostatin 1
Selective inhibitor of erastin induced ferroptosis
5181 Tolvaptan
Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active
5182 OXA 06 dihydrochloride
Potent ROCK inhibitor
5183 ETP 45835 dihydrochloride
Mnk1 and Mnk2 inhibitor
5185 JTE 607 dihydrochloride
Active metabolite binds CPSF3; Pro-drug
5186 Neuropathiazol
Selective inducer of neuronal differentiation in hippocampal neural progenitors
5188 S 07662
Constitutive androstane receptor (CAR) inverse agonist
5189 GSK 2837808A
Potent and selective LDHA inhibitor
5190 FRAX 486
Potent PAK inhibitor; brain penetrant and orally bioavailable
5191 PTC 209
Bmi-1 inhibitor; antitumor
5192 NBI 31772
High affinity insulin-like growth factor-I binding protein IGFBP inhibitor
5193 Remodelin
N-acetyltransferase 10 (NAT10) inhibitor
5196 PMX 205
Potent C5a receptor peptide antagonist
5197 Spautin 1
USP10 and USP13 inhibitor; inhibits autophagy
5198 AZ 20
Potent and selective ATR kinase inhibitor; antitumor
5199 AZD 7762 hydrochloride
Potent and selective ATP-competitive inhibitor of Chk1 and Chk2; also enhances CRISPR-Cpf1-mediated genome editing

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