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Displaying Products by Catalog Number (4800 - 4899)

Cat. No. Product Name / Activity
4800 4EGI-1
Inhibits eIF4E:eIF4G subunit interaction
4801 QNZ 46
Non-competitive and GluN2C/GluN2D-selective NMDA antagonist
4803 CRANAD 2
Near-infrared probe that detects Aβ40 aggregates
4804 APETx2
ASIC3 channel blocker
4805 TCS HDAC6 20b
Selective HDAC6 inhibitor
4806 BMS 345541
Selective allosteric inhibitor of IKK; anti-inflammatory
4808 FK 866 hydrochloride
Potent and non-competitive NAMPT inhibitor; induces apoptosis and autophagy
4809 DSR 6434
Potent TLR7 agonist
4810 BAM 7
Selective Bax activator; induces Bax-mediated apoptosis
4811 TAT 14
Nrf2 pathway activator; blocks Nrf2/Keap1 interaction
4812 ADWX 1
Potent and selective KV1.3 channel blocker
4813 Paprotrain
Reversible inhibitor of MKLP-2
4814 Methoxyresorufin
Fluorometric CYP450 substrate
4815 3-Cyano-7-ethoxycoumarin
Fluorescent cytochrome P450 substrate
4816 Pentoxyresorufin
Fluorometric cytochrome P450 substrate
4817 SKPin C1
Inhibits Skp2-mediated p27 degradation; induces cell cycle arrest
4818 PF 04418948
Potent and selective EP2 receptor antagonist
4819 Methylprednisolone
Glucocorticoid receptor agonist
4820 PF 04691502
Potent and selective dual PI 3-K/mTOR inhibitor
4821 PF 03814735
Aurora kinase A and B inhibitor
4822 Clindamycin hydrochloride
Antibiotic; inhibits protein synthesis
4823 PF 05212384
Potent and selective dual PI 3-K/mTOR inhibitor
4824 PD 334581
MEK1 inhibitor
4825 TC ASK 10
Potent and selective ASK1 inhibitor; orally bioavailable
4826 SUN 11602
Basic fibroblast growth factor (bFGF) mimetic; neuroprotective
4828 LDN 209929 dihydrochloride
Potent and selective haspin inhibitor
4829 ML 239
Breast cancer stem cell inhibitor
4830 LMK 235
Selective HDAC4/HDAC5 inhibitor
4831 NS 3861
α3β2 full agonist; also α3β4 partial agonist
4832 AZ 12216052
Positive allosteric modulator of mGlu8 receptors
4833 Levonorgestrel
Synthetic progesterone analog
4835 GPP 78 hydrochloride
NAMPT inhibitor; also induces autophagy
4836 AZ 628
Potent Raf kinase inhibitor
4837 AZD 3988
Potent and selective DGAT-1 inhibitor
4838 AZ 12080282 dihydrochloride
Inhibitor of Hedgehog (Hh) signaling
4839 AZD 6482
Potent and selective PI 3-Kβ inhibitor
4840 KU 0060648
Dual DNA-PK and PI 3-K inhibitor
4842 BIX 02189
Selective MEK5 and ERK5 inhibitor
4844 HJC 0350
Selective Epac2 inhibitor
4845 A 939572
Potent SCD-1 inhibitor
4847 PluriSln 1
SCD-1 inhibitor
4848 MI 2 (MALT1 inhibitor)
MALT1 inhibitor
4849 3-Nitropropionic acid
Irreversible mitochondrial respiratory complex II inhibitor
4852 Carbetocin
Oxytocin analog
4853 8-pCPT-2-O-Me-cAMP-AM
Selective Epac activator; cell-permeable analog of 8CPT-2Me-cAMP (Cat. No. 1645)
4854 ML 00253764 hydrochloride
Melanocortin MC4 receptor antagonist; brain penetrant
4855 WIKI4
Potent tankyrase inhibitor
4857 Amlexanox
Selective inhibitor of TBK
4858 NSC 697923
Selective UBE2N inhibitor
4860 ML 193
Potent, selective GPR55 antagonist
4862 PPTN hydrochloride
High affinity and selective P2Y14 antagonist
4863 CA 074
Selective cathepsin B inhibitor
4864 NS 6180
Potent KCa3.1 channel blocker
4865 APY 29
Inhibits IRE1α autophosphorylation; activates IRE1α endoribonuclease activity
4866 ML 190
Selective κ opioid receptor antagonist
4868 SR 1001
RORα/γ inverse agonist
4869 SR 2211
Selective RORγ inverse agonist
4870 H2L 5765834
LPA1,3,5 antagonist
4872 KML 29
Highly potent and selective MAGL inhibitor
4874 SR 1078
RORα/γ agonist
4875 Senexin A
Cdk8 inhibitor
4876 Eact
Activator of Ca2+-activated Cl- channel transmembrane protein 16A (TMEM16A)
4877 CaCCinh-A01
Calcium-activated chloride channel (CaCC) inhibitor
4878 H2L5186303
Potent and selective LPA2 receptor antagonist
4879 TC-G 1001
GPR35 agonist; more potent than zaprinast (Cat. No. 0947)
4880 ML 281
STK33 inhibitor
4881 LUF 6283
HCA2 (GPR109A) partial agonist
4883 CU CPT 4a
Selective TLR3 inhibitor
4884 CU CPT 22
Selective TLR1/2 inhibitor
4885 R 1530
Multi-RTK inhibitor; inhibits angiogenesis
4886 RU-SKI 43 hydrochloride
Hedgehog acyltransferase (Hhat) inhibitor; cell permeable
4887 OAC-1
Oct4 activator; enhances iPSC reprogramming efficiency
4888 KHS 101 hydrochloride
Selective inducer of neuronal differentiation in hippocampal neural progenitors
4889 SGC-CBP30
Potent CBP/p300 BRD inhibitor
4890 AR-C 118925XX
Selective and competitive P2Y2 antagonist
4891 I-CBP 112
Selective CBP/p300 BRD inhibitor
4892 (R)-PFI 2 hydrochloride
Potent and selective SETD7 inhibitor
4893 XL 388
Potent and selective mTOR inhibitor; antitumor
4895 ML 298 hydrochloride
Selective PLD2 inhibitor
4896 LH 846
Selective casein kinase 1δ inhibitor
4897 CYM 5541
Selective S1P3 receptor allosteric agonist
4898 TC-E 5006
γ-secretase modulator; reduces Aβ42 levels
4899 ML 120B dihydrochloride
Novel IKK2-selective inhibitor

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