All ProductsDisplaying Products by Catalog Number (5000 - 5099)
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| Cat. No. | Product Name / Activity |
|---|---|
| 5000 | FTIDC |
| Potent and selective negative allosteric modulator of mGlu1 receptors; also mGlu1 inverse agonist | |
| 5003 | Rhosin hydrochloride |
| Rho inhibitor | |
| 5005 | DR 4485 hydrochloride |
| High affinity and selective 5-HT7 antagonist; orally bioavailable | |
| 5011 | HMR 1556 |
| Potent and selective Iks channel blocker | |
| 5012 | PCI 29732 |
| Potent BTK inhibitor | |
| 5013 | AC 710 |
| Potent and selective PDGFR family inhibitor | |
| 5015 | 5-BrdU |
| Synthetic thymidine analog; used for cell proliferation assays | |
| 5016 | Fisetin |
| Naturally occuring flavonoid and antioxidant; neuroprotective | |
| 5018 | PEAQX tetrasodium salt |
| Potent and GluN2A-selective NMDA antagonist | |
| 5025 | Necrosulfonamide |
| Necroptosis inhibitor; also inhibits pyroptosis | |
| 5026 | KYT 0353 |
| Potent and selective inhibitor of L-type amino acid transporter 1 (LAT1); active in vivo | |
| 5027 | BCH |
| LAT1 inhibitor | |
| 5029 | CHC |
| MCT inhibitor; decreases glycoloysis | |
| 5031 | Pramlintide |
| Synthetic version of amylin (Cat. No. 3418) | |
| 5032 | Talampanel |
| Non-competitive non-NMDA iGluR antagonist | |
| 5037 | Nepicastat hydrochloride |
| Potent and selective dopamine β-hydroxylase (DBH) inhibitor; orally bioavailable | |
| 5040 | SB 706504 |
| p38 MAPK inhibitor | |
| 5042 | Psalmotoxin 1 |
| Potent and selective ASIC1a channel blocker | |
| 5043 | FFN 206 dihydrochloride |
| Fluorescent VMAT2 substrate | |
| 5044 | SR 3576 |
| Highly potent and selective JNK3 inhibitor | |
| 5047 | PRT 4165 |
| Inhibitor of Bmi1/Ring1A; blocks histone H2A ubiquitination | |
| 5050 | CASIN |
| Cdc42 inhibitor | |
| 5051 | BIO 5192 |
| Highly potent and selective inhibitor of integrin α4β1 (VLA-4) | |
| 5053 | AC 186 |
| Potent and selective ERβ agonist; neuroprotective | |
| 5061 | RKI 1447 dihydrochloride |
| Potent and selective ROCK inhibitor; antitumor | |
| 5062 | Cyclotraxin B |
| TrkB receptor antagonist | |
| 5064 | LY 379268 disodium salt |
| Selective group II mGlu agonist; sodium salt of LY 379268 (Cat. No. 2453) | |
| 5066 | ICA 121431 |
| Potent and selective NaV1.3 and NaV1.1 channel blocker | |
| 5067 | MRT 68601 hydrochloride |
| Potent TBK inhibitor | |
| 5069 | Teriflunomide |
| Inhibitor of DHODH; active metabolite of Leflunomide | |
| 5071 | NKY 80 |
| Adenylyl cyclase inhibitor | |
| 5072 | PFI 3 |
| Potent and selective SMARCA2/4 and polybromo 1 inhibitor | |
| 5075 | Harmine |
| Potent and selective DYRK1A inhibitor | |
| 5076 | SZL P1-41 |
| Selective Skp2 inhibitor; suppresses E3 ligase activity | |
| 5077 | DDR1-IN-1 dihydrochloride |
| Selective DDR1 inhibitor | |
| 5079 | ABT 089 dihydrochloride |
| High affinity and selective α4β2 nAChR partial agonist | |
| 5081 | J 147 |
| Neuroprotective and neurotrophic compound; reduces Aβ40 and Aβ42 levels | |
| 5083 | QO 58 |
| Kv7 channel opener | |
| 5085 | L 012 sodium salt |
| Chemiluminescent ROS and RNS indicator | |
| 5087 | TC NTR1 17 |
| Selective NTS1 partial agonist | |
| 5088 | TC-S 7004 |
| Potent and selective DYRK1A/B inhibitor | |
| 5089 | TC-E 5002 |
| Selective KDM2/7 inhibitor | |
| 5092 | Acridine Orange hydrochloride |
| Nucleic acid binding dye. Cell permeable. Used for: cell cycle and apoptosis determination. Application: flow cytometry, fluorescence microscopy | |
| 5095 | DBM 1285 dihydrochloride |
| p38 MAPK inhibitor; anti-inflammatory | |
| 5096 | AdipoRon hydrochloride |
| Orally active AdipoR1 and AdipoR2 agonist; antidiabetic | |
| 5097 | A12B4C3 |
| Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor |