All Products

Displaying Products by Catalog Number (5000 - 5099)

Cat. No. Product Name / Activity
5000 FTIDC
Potent and selective negative allosteric modulator of mGlu1 receptors; also mGlu1 inverse agonist
5003 Rhosin hydrochloride
Rho inhibitor
5005 DR 4485 hydrochloride
High affinity and selective 5-HT7 antagonist; orally bioavailable
5009 BMS 509744
Potent and selective ITK inhibitor
5011 HMR 1556
Potent and selective Iks channel blocker
5012 PCI 29732
Potent BTK inhibitor
5013 AC 710
Potent and selective PDGFR family inhibitor
5015 5-BrdU
Synthetic thymidine analog; used for cell proliferation assays
5016 Fisetin
Naturally occuring flavonoid and antioxidant; neuroprotective
5017 A 85380 dihydrochloride
High affinity and selective α4β2 nAChR agonist
5018 PEAQX tetrasodium salt
Potent and GluN2A-selective NMDA antagonist
5020 SF 1670
PTPN2 and PTEN inhibitor
5021 TC-G 1000
Potent and selective α2D agonist
5022 BMS 599626 dihydrochloride
Potent, selective EGFR and ErbB2 inhibitor
5025 Necrosulfonamide
Necroptosis inhibitor; also inhibits pyroptosis
5026 KYT 0353
Potent and selective inhibitor of L-type amino acid transporter 1 (LAT1); active in vivo
5027 BCH
LAT1 inhibitor
5028 GMQ hydrochloride
Selective ASIC3 opener
5029 CHC
MCT inhibitor; decreases glycoloysis
5031 Pramlintide
Synthetic version of amylin (Cat. No. 3418)
5032 Talampanel
Non-competitive non-NMDA iGluR antagonist
5033 2-MPPA
Selective glutamate carboxypeptidase II (GCP II) inhibitor; orally bioavailable
5035 AS 2034178
Selective FFA1 (GPR40) agonist
5037 Nepicastat hydrochloride
Potent and selective dopamine β-hydroxylase (DBH) inhibitor; orally bioavailable
5038 ABT
Cytochrome P450 inhibitor; inhibits 20-HETE synthesis
5039 SR 144528
High affinity and selective CB2 inverse agonist
5040 SB 706504
p38 MAPK inhibitor
5041 PAOPA
Allosteric modulator of D2 receptors
5042 Psalmotoxin 1
Potent and selective ASIC1a channel blocker
5043 FFN 206 dihydrochloride
Fluorescent VMAT2 substrate
5044 SR 3576
Highly potent and selective JNK3 inhibitor
5045 L002
p300 inhibitor
5046 LM11A 31 dihydrochloride
Nonpeptide p75NTR ligand; neuroprotective
5047 PRT 4165
Inhibitor of Bmi1/Ring1A; blocks histone H2A ubiquitination
5048 YZ9
PFKFB3 inhibitor
5049 TC-E 5001
Potent tankyrase inhibitor
5050 CASIN
Cdc42 inhibitor
5051 BIO 5192
Highly potent and selective inhibitor of integrin α4β1 (VLA-4)
5052 TG 4-155
High affinity and selective EP2 receptor antagonist
5053 AC 186
Potent and selective ERβ agonist; neuroprotective
5054 ME 0328
Selective PARP-3 inhibitor
5055 Qc 1
Threonine dehydrogenase inhibitor
5056 Ki 16425
LPA1 and LPA3 receptor antagonist
5057 UNC 2327
Allosteric inhibitor of PRMT3
5061 RKI 1447 dihydrochloride
Potent and selective ROCK inhibitor; antitumor
5062 Cyclotraxin B
TrkB receptor antagonist
5063 SRPIN340
Selective SRPK1 inhibitor
5064 LY 379268 disodium salt
Selective group II mGlu agonist; sodium salt of LY 379268 (Cat. No. 2453)
5065 NSC 319726
Reactivator of mutant p53
5066 ICA 121431
Potent and selective NaV1.3 and NaV1.1 channel blocker
5067 MRT 68601 hydrochloride
Potent TBK inhibitor
5068 ITD 1
Selective inhibitor of TGF-β signaling; induces cardiomyocyte differentiation in ESCs
5069 Teriflunomide
Inhibitor of DHODH; active metabolite of Leflunomide
5071 NKY 80
Adenylyl cyclase inhibitor
5072 PFI 3
Potent and selective SMARCA2/4 and polybromo 1 inhibitor
5074 ANQ 11125
Selective motilin receptor antagonist
5075 Harmine
Potent and selective DYRK1A inhibitor
5076 SZL P1-41
Selective Skp2 inhibitor; suppresses E3 ligase activity
5077 DDR1-IN-1 dihydrochloride
Selective DDR1 inhibitor
5079 ABT 089 dihydrochloride
High affinity and selective α4β2 nAChR partial agonist
5080 TC-G 1003
High affinity somatostatin sst2 agonist
5081 J 147
Neuroprotective and neurotrophic compound; reduces Aβ40 and Aβ42 levels
5082 LDN 212320
Increases EAAT2 expression; neuroprotective
5083 QO 58
Kv7 channel opener
5084 MN 64
Potent and selective tankyrase inhibitor
5085 L 012 sodium salt
Chemiluminescent ROS and RNS indicator
5086 PA 452
RXR antagonist
5087 TC NTR1 17
Selective NTS1 partial agonist
5088 TC-S 7004
Potent and selective DYRK1A/B inhibitor
5089 TC-E 5002
Selective KDM2/7 inhibitor
5092 Acridine Orange hydrochloride
Nucleic acid binding dye
5094 PG 931
Potent and selective MC4 receptor agonist
5095 DBM 1285 dihydrochloride
p38 MAPK inhibitor; anti-inflammatory
5096 AdipoRon hydrochloride
Orally active AdipoR1 and AdipoR2 agonist; antidiabetic
5097 A12B4C3
Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor
5098 KRCA 0008
Potent Ack1 and ALK dual inhibitor; orally bioavailable
5099 TC-E 5003
Selective PRMT1 inhibitor

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