All Products

Displaying Products by Catalog Number (5000 - 5099)

Cat. No. Product Name / Activity
5000 FTIDC
Potent and selective negative allosteric modulator of mGlu1 receptors; also mGlu1 inverse agonist
5003 Rhosin hydrochloride
Rho inhibitor
5005 DR 4485 hydrochloride
High affinity and selective 5-HT7 antagonist; orally bioavailable
5011 HMR 1556
Potent and selective Iks channel blocker
5012 PCI 29732
Potent BTK inhibitor
5013 AC 710
Potent and selective PDGFR family inhibitor
5015 5-BrdU
Synthetic thymidine analog; used for cell proliferation assays
5016 Fisetin
Naturally occuring flavonoid and antioxidant; neuroprotective
5017 A 85380 dihydrochloride
High affinity and selective α4β2 nAChR agonist
5018 PEAQX tetrasodium salt
Potent and GluN2A-selective NMDA antagonist
5020 SF 1670
PTPN2 and PTEN inhibitor
5025 Necrosulfonamide
Necroptosis inhibitor; also inhibits pyroptosis
5026 KYT 0353
Potent and selective inhibitor of L-type amino acid transporter 1 (LAT1); active in vivo
5027 BCH
LAT1 inhibitor
5029 CHC
MCT inhibitor; decreases glycoloysis
5031 Pramlintide
Synthetic version of amylin (Cat. No. 3418)
5032 Talampanel
Non-competitive non-NMDA iGluR antagonist
5037 Nepicastat hydrochloride
Potent and selective dopamine β-hydroxylase (DBH) inhibitor; orally bioavailable
5040 SB 706504
p38 MAPK inhibitor
5042 Psalmotoxin 1
Potent and selective ASIC1a channel blocker
5043 FFN 206 dihydrochloride
Fluorescent VMAT2 substrate
5044 SR 3576
Highly potent and selective JNK3 inhibitor
5046 LM11A 31 dihydrochloride
Nonpeptide p75NTR ligand; neuroprotective
5047 PRT 4165
Inhibitor of Bmi1/Ring1A; blocks histone H2A ubiquitination
5050 CASIN
Cdc42 inhibitor
5051 BIO 5192
Highly potent and selective inhibitor of integrin α4β1 (VLA-4)
5053 AC 186
Potent and selective ERβ agonist; neuroprotective
5056 Ki 16425
LPA1 and LPA3 receptor antagonist
5057 UNC 2327
Allosteric inhibitor of PRMT3
5061 RKI 1447 dihydrochloride
Potent and selective ROCK inhibitor; antitumor
5062 Cyclotraxin B
TrkB receptor antagonist
5064 LY 379268 disodium salt
Selective group II mGlu agonist; sodium salt of LY 379268 (Cat. No. 2453)
5066 ICA 121431
Potent and selective NaV1.3 and NaV1.1 channel blocker
5067 MRT 68601 hydrochloride
Potent TBK inhibitor
5068 ITD 1
Selective inhibitor of TGF-β signaling; induces cardiomyocyte differentiation in ESCs
5069 Teriflunomide
Inhibitor of DHODH; active metabolite of Leflunomide
5071 NKY 80
Adenylyl cyclase inhibitor
5072 PFI 3
Potent and selective SMARCA2/4 and polybromo 1 inhibitor
5075 Harmine
Potent and selective DYRK1A inhibitor
5076 SZL P1-41
Selective Skp2 inhibitor; suppresses E3 ligase activity
5077 DDR1-IN-1 dihydrochloride
Selective DDR1 inhibitor
5079 ABT 089 dihydrochloride
High affinity and selective α4β2 nAChR partial agonist
5081 J 147
Neuroprotective and neurotrophic compound; reduces Aβ40 and Aβ42 levels
5083 QO 58
Kv7 channel opener
5085 L 012 sodium salt
Chemiluminescent ROS and RNS indicator
5086 PA 452
RXR antagonist
5087 TC NTR1 17
Selective NTS1 partial agonist
5088 TC-S 7004
Potent and selective DYRK1A/B inhibitor
5089 TC-E 5002
Selective KDM2/7 inhibitor
5092 Acridine Orange hydrochloride
Nucleic acid binding dye
5095 DBM 1285 dihydrochloride
p38 MAPK inhibitor; anti-inflammatory
5096 AdipoRon hydrochloride
Orally active AdipoR1 and AdipoR2 agonist; antidiabetic
5097 A12B4C3
Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor
5098 KRCA 0008
Potent Ack1 and ALK dual inhibitor; orally bioavailable

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