Cat. No. | Product Name / Activity |
---|---|
4601 | TUG 891 |
Potent and selective FFA4 (GPR120) agonist | |
4602 | LDN 27219 |
Transglutaminase 2 (TG2) inhibitor; reversible | |
4603 | LUF 5834 |
Potent adenosine A2A and A2B receptor partial agonist | |
4606 | CYM 9484 |
Potent NPY Y2 receptor antagonist | |
4607 | LM 22A4 |
Potent TrkB agonist | |
4609 | BMS 303141 |
ATP citrate lyase inhibitor; orally bioavailable | |
4611 | PBP 10 |
Selective FPR2 antagonist; cell permeable | |
4612 | URB 597 |
Potent and selective FAAH inhibitor | |
4616 | Olmesartan |
Potent AT1 antagonist | |
4617 | Penitrem A |
Potent and selective KCa1.1 (BK) channel blocker | |
4618 | GW 6471 |
PPARα antagonist | |
4619 | Melphalan |
DNA alkylating agent; cytotoxic and antineoplastic | |
4621 | MKT 077 |
Binds mot-2; selectively cytotoxic in cancer cells | |
4622 | MK 1903 |
Potent and selective GPR109A (HCA2) agonist | |
4624 | TC-FPR 43 |
Potent FPR2 agonist | |
4625 | TC OT 39 |
Potent non-peptide oxytocin receptor partial agonist; also V1a receptor antagonist | |
4629 | GSK2578215A |
Potent, selective LRRK2 inhibitor; brain penetrant | |
4630 | SB 747651A dihydrochloride |
Potent MSK1 inhibitor; also inhibits other AGC group kinases | |
4632 | TC-I 2000 |
TRPM8 blocker | |
4633 | Pam3CSK4 |
TLR1/2 agonist; induces cytokine production | |
4635 | SC 79 |
Akt activator | |
4637 | Pam2CSK4 |
TLR2/6 agonist; induces TNF-α production | |
4641 | BI 6015 |
Hepatocyte nuclear factor 4α (HNF4α) antagonist | |
4642 | 4-CMTB |
FFA2 agonist; also exhibits positive allosteric modulatory activity | |
4643 | PCI 34051 |
Potent and selective HDAC8 inhibitor | |
4645 | Z-VRPR-FMK trifluoroacetate salt |
Irreversible MALT1 inhibitor | |
4646 | Elacridar hydrochloride |
P-gp and BCRP inhibitor | |
4647 | GR 203040 |
Potent and selective NK1 antagonist | |
4650 | I-BET 151 dihydrochloride |
BET bromodomain inhibitor; also promotes differentiation of hiPSCs into megakaryocytes | |
4651 | JW 67 |
Wnt pathway inhibitor; induces degradation of active β-catenin | |
4652 | SAHA |
Class I and II HDAC inhibitor | |
4655 | NSC 74859 |
Selective STAT3 inhibitor | |
4656 | (D)-(+)-Neopterin |
Stimulated by IFN-γ; marker of immune activation | |
4657 | Zolmitriptan |
Potent 5-HT1B/1D/1F agonist | |
4660 | KB SRC 4 |
Potent and selective c-Src inhibitor | |
4663 | Apocynin |
NADPH-oxidase inhibitor | |
4664 | Obtustatin |
Potent and selective α1β1 inhibitor | |
4673 | SB 674042 |
Potent and selective non-peptide OX1 antagonist | |
4676 | ARRY 520 trifluoroacetate |
Potent and selective kinesin spindle protein (KSP) inhibitor; induces Mcl-1 degradation | |
4677 | CYM 50260 |
Potent and selective S1P4 agonist | |
4678 | CYM 50308 |
Potent and selective S1P4 agonist | |
4679 | CYM 50358 hydrochloride |
Potent and selective S1P4 antagonist | |
4683 | RFRP 3 (human) |
NPFF1 agonist; GnIH homolog | |
4685 | KL 001 |
Cryptochrome protein stabilizer; lengthens circadian period | |
4686 | Xanthohumol |
p97 ATPase (VCP) inhibitor | |
4687 | ML 252 |
Potent and selective KV7.2 inhibitor; brain penetrant | |
4688 | GSK J2 |
Inactive isomer of GSK J1 (Cat. No. 4593) | |
4690 | Fmk |
Irreversible ribosomal S6 kinase 1/2 inhibitor | |
4691 | NAV 26 |
Selective Nav1.7 channel blocker | |
4694 | Ro 5-3335 |
Core binding factor inhibitor; attenuates hematopoiesis | |
4695 | Ischemin sodium salt |
CBP inhibitor; cell permeable |