All Products

Displaying Products by Catalog Number (4600 - 4699)

Cat. No. Product Name / Activity
4600 Auranofin
Thioredoxin reductase inhibitor; induces MPT
4601 TUG 891
Potent and selective FFA4 (GPR120) agonist
4602 LDN 27219
Transglutaminase 2 (TG2) inhibitor; reversible
4603 LUF 5834
Potent adenosine A2A and A2B receptor partial agonist
4604 PTIQ
Potent MMP-3 expression inhibitor; neuroprotective
4605 (±)-SLV 319
High affinity and selective CB1 antagonist
4606 CYM 9484
Potent NPY Y2 receptor antagonist
4607 LM 22A4
Potent TrkB agonist
4608 BIIB 021
Selective Hsp90 inhibitor
4609 BMS 303141
ATP citrate lyase inhibitor; orally bioavailable
4611 PBP 10
Selective FPR2 antagonist; cell permeable
4612 URB 597
Potent and selective FAAH inhibitor
4613 Tegaserod maleate
5-HT4 partial agonist
4615 MEDICA 16
FFA1 (GPR40) agonist; also inhibits ATP citrate lyase
4616 Olmesartan
Potent AT1 antagonist
4617 Penitrem A
Potent and selective BKCa (KCa1.1) channel blocker
4618 GW 6471
PPARα antagonist
4619 Melphalan
DNA alkylating agent; cytotoxic and antineoplastic
4621 MKT 077
Binds mot-2; selectively cytotoxic in cancer cells
4622 MK 1903
Potent and selective GPR109A (HCA2) agonist
4624 TC-FPR 43
Potent FPR2 agonist
4625 TC OT 39
Potent non-peptide oxytocin receptor partial agonist; also V1a receptor antagonist
4626 Andrographolide
Inhibits NFκB; blocks androgen receptor (AR) expression
4627 Phlorizin
Na+-glucose cotransporter (SGLT) inhibitor
4628 DiMNF
Selective aryl hydrocarbon receptor modulator (SAhRM)
4629 GSK2578215A
Potent, selective LRRK2 inhibitor; brain penetrant
4630 SB 747651A dihydrochloride
Potent MSK1 inhibitor; also inhibits other AGC group kinases
4632 TC-I 2000
TRPM8 blocker
4633 Pam3CSK4
TLR1/2 agonist; induces cytokine production
4635 SC 79
Akt activator
4637 Pam2CSK4
TLR2/6 agonist; induces TNF-α production
4638 Pam2CSK4 Biotin
Biotinylated Pam2CSK4 (Cat. No. 4637)
4639 TT 232
sst1 and sst4 agonist
4640 N,N-Dimethylsphingosine
Sphingosine kinase inhibitor
4641 BI 6015
Hepatocyte nuclear factor 4α (HNF4α) antagonist
4642 4-CMTB
FFA2 agonist; also exhibits positive allosteric modulatory activity
4643 PCI 34051
Potent and selective HDAC8 inhibitor
4644 CID 2011756
Pan protein kinase D (PKD) inhibitor; cell permeable
4645 Z-VRPR-FMK trifluoroacetate salt
Irreversible MALT1 inhibitor
4646 Elacridar hydrochloride
P-gp inhibitor
4647 GR 203040
Potent and selective NK1 antagonist
4650 I-BET 151 dihydrochloride
BET bromodomain inhibitor; also promotes differentiation of hiPSCs into megakaryocytes
4651 JW 67
Wnt pathway inhibitor; induces degradation of active β-catenin
4652 SAHA
Class I and II HDAC inhibitor
4653 ML 171
Selective NADPH oxidase 1 (NOX1) inhibitor
4655 NSC 74859
Selective STAT3 inhibitor
4656 (D)-(+)-Neopterin
Stimulated by IFN-γ; marker of immune activation
4657 Zolmitriptan
Potent 5-HT1B/1D/1F agonist
4659 Floxuridine
Thymidylate synthetase inhibitor
4660 KB SRC 4
Potent and selective c-Src inhibitor
4662 SMANT hydrochloride
Inhibits Smoothened (Smo) accumulation
4663 Apocynin
NADPH-oxidase inhibitor
4664 Obtustatin
Potent and selective α1β1 inhibitor
4665 ProTx I
CaV3.1 blocker; also inhibits NaV1.8 and KV2.1
4666 UNC 1215
Potent inhibitor of L3MBTL3 Kme reader domain; cell permeable
4667 SB 706375
High affinity, non-peptide UT receptor antagonist
4668 GW 627368
Selective EP4 receptor competitive antagonist
4670 SB 611812
Urotensin-II (UT) antagonist; attenuates cardiac dysfunction
4672 SB 223412
Potent, selective non-peptide NK3 antagonist. Brain penetrant
4673 SB 674042
Potent and selective non-peptide OX1 antagonist
4674 CZC 24832
Selective inhibitor of PI 3-kinase γ
4675 CCT 031374 hydrobromide
Inhibits TCF-dependent transcription; lowers β-catenin levels
4676 ARRY 520 trifluoroacetate
Potent and selective kinesin spindle protein (KSP) inhibitor; induces Mcl-1 degradation
4677 CYM 50260
Potent and selective S1P4 agonist
4678 CYM 50308
Potent and selective S1P4 agonist
4679 CYM 50358 hydrochloride
Potent and selective S1P4 antagonist
4683 RFRP 3 (human)
NPFF1 agonist; GnIH homolog
4684 Daminozide
Selective KDM2/7 inhibitor
4685 KL 001
Cryptochrome protein stabilizer; lengthens circadian period
4686 Xanthohumol
p97 ATPase (VCP) inhibitor
4688 GSK J2
Inactive isomer of GSK J1 (Cat. No. 4593)
4690 Fmk
Irreversible ribosomal S6 kinase 1/2 inhibitor
4691 NAV 26
Selective Nav1.7 channel blocker
4694 Ro 5-3335
Core binding factor inhibitor; attenuates hematopoiesis
4695 Ischemin sodium salt
CBP inhibitor; cell permeable
4697 A 331440 dihydrochloride
Selective H3 antagonist

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