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Displaying Products by Catalog Number (1900 - 1999)

Cat. No. Product Name / Activity
1900 [Ala107]-MBP (104-118)
Protein kinase C inhibitor
1901 [Ala113]-MBP (104-118)
Protein kinase C inhibitor
1902 [Ala92]-p16 (84-103)
Cdk inhibitor
1904 PKA inhibitor fragment (6-22) amide
Potent protein kinase A inhibitor
1905 VIP (6-28) (human, rat, porcine, bovine)
VIP receptor antagonist
1906 Atrial natriuretic factor (1-28) (human, porcine)
Endogenous peptide regulating blood pressure
1907 Neuromedin N (rat, mouse, porcine, canine)
Neurotensin-like peptide
1908 Neuromedin B (porcine)
Mammalian bombesin-like peptide
1909 Neurotensin
Endogenous neurotransmitter and endocrine modulator
1910 Oxytocin
Involved in uterine contraction and lactation
1911 VIP (human, rat, mouse, rabbit, canine, porcine)
Involved in neurotransmission and smooth muscle relaxation
1912 Atrial natriuretic factor (1-28) (rat)
Endogenous peptide regulating blood pressure
1914 Eledoisin
Potent tachykinin receptor ligand
1915 Kinetensin (human)
Neurotensin-like peptide
1916 Litorin
Amphibian bombesin-like peptide
1917 Neuromedin U (rat)
Endogenous modulator of blood pressure and flow, gut ion transport, feeding and body temperature
1918 Secretin (human)
Gastrointestinal peptide
1919 Secretin (rat)
Gastrointestinal peptide
1920 Eledoisin-Related Peptide
Tachykinin receptor ligand
1921 N-Formyl-Met-Leu-Phe
Endogenous FPR1 agonist
1922 [D-Lys3]-GHRP-6
Ghrelin receptor antagonist
1923 pp60 c-src (521-533) (phosphorylated)
Inhibits tyrosine kinase activity of pp60c-src and pp60v-src
1927 N-Acetyl-O-phosphono-Tyr-Glu-Glu-Ile-Glu
Phosphopeptide ligand for src SH2 domain
1928 Neuropeptide AF (human)
Endogenous NPFF1 and NPFF2 agonist; antiopioid neuropeptide and MRGPRA agonist
1929 Melanocyte-stimulating hormone release inhibiting factor
Inhibitor of α-MSH release; inhibits opioid effects in vivo
1930 N-Acetyl-O-phosphono-Tyr-Glu Dipentylamide
Phosphopeptide ligand for src SH2 domain
1931 G-Protein antagonist peptide
Inhibits G protein activation by GPCRs
1932 U 46619
Potent, stable thromboxane A2 (TP) receptor agonist
1933 Exendin-4
Potent GLP-1 receptor agonist
1935 Caffeic acid-pYEEIE
Phosphopeptide ligand for src SH2 domain
1936 Damnacanthal
Potent, selective p56lck inhibitor; also LIMK1/2 inhibitor
1937 NSC 693868
Cdk inhibitor; also inhibits GSK-3
1938 Amyloid β-Peptide (1-43) (human)
Amyloid β-protein fragment
1939 C14TKL-1
Endogenous NK1 agonist
1941 m-3M3FBS
Phospholipase C activator
1942 o-3M3FBS
Inactive analog of m-3M3FBS (Cat. No. 1941)
1944 Loratidine
Peripheral H1 antagonist; antiallergic agent
1946 [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
Potent ghrelin receptor inverse agonist; Antagonist at other neuropeptide receptors
1947 PR 39 (porcine)
IκBα inhibitor
1949 L-670,596
Potent, selective thromboxane A2/prostaglandin endoperoxide antagonist
1950 Gap 26
Gap junction blocker; inhibits smooth muscle contraction and IP3-mediated ATP release
1952 DCB
Allosteric modulator of mGlu5 receptors
1953 DMeOB
Negative allosteric modulator of mGlu5 receptors
1954 Antagonist G
Broad spectrum neuropeptide receptor antagonist
1955 Ritanserin
Potent 5-HT2 antagonist
1956 Bestatin
Aminopeptidase inhibitor
1957 GR 79236
A1 agonist
1960 SB 334867
Selective non-peptide OX1 antagonist
1961 SB 258585 hydrochloride
Potent, selective 5-HT6 antagonist
1962 SB 239063
Potent, selective p38 MAPK inhibitor; orally active
1963 SB 408124
Selective non-peptide OX1 antagonist
1964 Gossypol
Proapoptotic; downregulates Bcl-2 and Bcl-XL
1965 Simvastatin
HMG-CoA reductase inhibitor
1966 UCM 707
Potent anandamide transport inhibitor
1967 Ranitidine hydrochloride
Selective H2 antagonist
1968 AS 19
Potent 5-HT7 agonist
1969 SL 327
Selective inhibitor of MEK1 and MEK2; brain penetrant
1970 Norketamine hydrochloride
Potent non-competitive NMDA antagonist; antinociceptive
1971 (+)-Anabasine hydrochloride
High affinity nAChR partial agonist
1972 Tianeptine sodium salt
Selective facilitator of 5-HT uptake; antidepressant
1974 SANT-1
Inhibitor of hedgehog (Hh) signaling; antagonizes smoothened activity
1975 6-Iodonordihydrocapsaicin
Potent, competitive vanilloid receptor antagonist
1979 L-803,087 trifluoroacetate
Potent and selective sst4 agonist
1980 L-817,818
Potent and selective sst5 agonist
1982 Reboxetine mesylate
Potent and selective noradrenalin uptake inhibitor; orally active
1983 740 Y-P
Cell-permeable PI 3-kinase activator
1984 Nogo-66 (1-40)
Competitive antagonist for Nogo-66 receptor; promotes neuron regeneration
1985 PNU 142633
Highly selective 5-HT1D agonist
1987 Leptomycin B
Inhibits nuclear export of proteins; antitumor
1989 c-JUN peptide
Peptide inhibitor of JNK/c-Jun interaction
1990 (R,R)-THC
Potent subtype-selective ligand; ERα agonist/ERβ antagonist
1991 MPP dihydrochloride
Highly selective ERα antagonist
1992 Nomifensine
Potent noradrenalin and dopamine uptake inhibitor. Antidepressant
1993 Halofuginone hydrobromide
High affinity competitive prolyl-tRNA synthetase inhibitor
1994 ZK 93423 hydrochloride
Potent benzodiazepine agonist
1995 Ro 19-4603
Benzodiazepine inverse agonist
1996 ZK 93426 hydrochloride
Potent and competitive benzodiazepine antagonist
1997 Ro 15-4513
Benzodiazepine partial inverse agonist
1998 JMV 449
Potent neurotensin receptor agonist
1999 Linopirdine dihydrochloride
KV7 (KCNQ) channel blocker

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