All Products

Displaying Products by Catalog Number (2000 - 2099)

Cat. No. Product Name / Activity
2000 XE 991 dihydrochloride
Potent, selective KV7 (KCNQ) channel blocker; blocks M-currents
2001 GS 39783
Positive allosteric modulator of GABAB receptors
2002 Ro 31-8220 mesylate
Protein kinase inhibitor
2004 Isradipine
CaV1.x blocker
2005 Ro 04-5595 hydrochloride
GluN2B-selective NMDA antagonist
2006 Paxilline
SERCA ATPase blocker. Also potent BKCa channel blocker
2007 Fluticasone propionate
Selective high affinity glucocorticoid receptor agonist
2008 SKF 86002 dihydrochloride
p38 MAPK inhibitor; anti-inflammatory agent
2009 PSB 1115
Selective human A2B antagonist; water-soluble
2010 PSB 10 hydrochloride
Potent, highly selective hA3 receptor antagonist/inverse agonist
2011 Tomoxetine hydrochloride
Potent and selective noradrenalin re-uptake inhibitor
2012 PSB 11 hydrochloride
Potent, selective hA3 receptor antagonist/inverse agonist
2013 Guggulsterone
Broad spectrum steroid receptor ligand. Antagonizes FXR and displays hypolipidemic activity
2018 Mirtazapine
Potent 5-HT2 antagonist; also 5-HT3, H1 and α2 antagonist; antidepressant
2019 PSB 36
Potent and selective A1 antagonist
2020 Ch 55
Potent RAR agonist
2021 LE 135
Selective RARβ antagonist
2022 SR 202
Selective PPARγ antagonist; antidiabetic and antiobesity agent
2024 PL 017
Selective μ agonist
2025 Cinalukast
Potent, selective CysLT1 (LTD4) antagonist; orally active
2033 Pentostatin
Adenosine deaminase inhibitor
2034 ROS 234 dioxalate
Potent H3 antagonist
2037 SDZ 205-557 hydrochloride
5-HT3 and 5-HT4 antagonist
2038 Iloprost
Prostacyclin (PGI2) analog
2067 187-1, N-WASP inhibitor
N-WASP inhibitor; inhibits actin assembly
2070 K 41498
Highly selective and potent CRF2 antagonist
2071 Antisauvagine-30
Potent, selective and competitive CRF2 antagonist
2072 Aminopurvalanol A
Selective cdk inhibitor; potently inhibits cdk1, cdk2 and cdk5
2073 (R)-(-)-Apomorphine hydrochloride
Dopamine agonist; non-subtype-selective
2074 SKF 83959 hydrobromide
D1-like partial agonist
2075 SKF 83822 hydrobromide
Selective D1-like agonist
2076 Y-26763
Kir6 (KATP) channel opener
2077 Y-27152
Prodrug of Kir6 (KATP) channel opener Y-26763 (Cat. No. 2076); orally active in vivo
2078 UBP 296
Potent and selective kainate antagonist; selective for GluK1-containing receptors
2079 UBP 302
Potent and selective kainate antagonist; active enantiomer of UBP 296 (Cat. No. 2078)
2080 PHM 27 (human)
Potent calcitonin agonist; endogenous analog of human VIP
2081 Exendin-3 (9-39) amide
Potent GLP-1 receptor antagonist
2082 Glucagon-like peptide 1 (7-36) amide (human, rat)
Potent insulinotropic peptide
2084 GIP (human)
Potent insulinotropic gut hormone; GIP agonist
2085 Galnon
Non-selective galanin receptor agonist
2086 GTP 14564
Class III receptor tyrosine kinase (RTK) inhibitor
2087 NTR 368
p75NTR fragment; induces apoptosis
2088 DMNB
DNA-PK inhibitor
2089 RS 102895 hydrochloride
CCR2b chemokine receptor antagonist
2090 CALP1
Cell-permeable calmodulin agonist
2092 Ionomycin free acid
Calcium ionophore
2094 Oxyntomodulin (porcine, bovine)
GLP-1 receptor agonist; endogenous preproglucagon derived peptide; modulates feeding and metabolism
2095 PNU 37883 hydrochloride
Vascular Kir6 (KATP) channel blocker
2096 DAU 5884 hydrochloride
M3 receptor antagonist
2097 SKI II
Selective non-lipid inhibitor of sphingosine kinase
2098 Apoptosis Activator 2
Promotes apoptosome formation and activates caspase-9/caspase-3 pathway. Selectively induces tumor cell apoptosis

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