All Products

Displaying Products by Catalog Number (2000 - 2099)

Cat. No. Product Name / Activity
2000 XE 991 dihydrochloride
Potent, selective KV7 (KCNQ) channel blocker; blocks M-currents
2001 GS 39783
Positive allosteric modulator of GABAB receptors
2002 Ro 31-8220 mesylate
Protein kinase inhibitor
2004 Isradipine
CaV1.x blocker
2006 Paxilline
SERCA ATPase blocker. Also potent BKCa channel blocker
2007 Fluticasone propionate
Selective high affinity glucocorticoid receptor agonist
2009 PSB 1115
Selective human A2B antagonist; water-soluble
2010 PSB 10 hydrochloride
Potent, highly selective hA3 receptor antagonist/inverse agonist
2011 Tomoxetine hydrochloride
Potent and selective noradrenalin re-uptake inhibitor
2018 Mirtazapine
Potent 5-HT2 antagonist; also 5-HT3, H1 and α2 antagonist; antidepressant
2020 Ch 55
Potent RAR agonist
2021 LE 135
Selective RARβ antagonist
2022 SR 202
Selective PPARγ antagonist; antidiabetic and antiobesity agent
2033 Pentostatin
Adenosine deaminase inhibitor
2070 K 41498
Highly selective and potent CRF2 antagonist
2072 Aminopurvalanol A
Selective cdk inhibitor; potently inhibits cdk1, cdk2 and cdk5
2073 (R)-(-)-Apomorphine hydrochloride
Dopamine agonist; non-subtype-selective
2074 SKF 83959 hydrobromide
D1-like partial agonist
2075 SKF 83822 hydrobromide
Selective D1-like agonist
2076 Y-26763
Kir6 (KATP) channel opener
2078 UBP 296
Potent and selective kainate antagonist; selective for GluK1-containing receptors
2079 UBP 302
Potent and selective kainate antagonist; active enantiomer of UBP 296 (Cat. No. 2078)
2081 Exendin-3 (9-39) amide
Potent GLP-1 receptor antagonist
2082 Glucagon-like peptide 1 (7-36) amide (human, rat)
Potent insulinotropic peptide
2084 GIP (human)
Potent insulinotropic gut hormone; GIP agonist
2089 RS 102895 hydrochloride
CCR2b chemokine receptor antagonist
2090 CALP1
Cell-permeable calmodulin agonist
2092 Ionomycin free acid
Calcium ionophore
2094 Oxyntomodulin (porcine, bovine)
GLP-1 receptor agonist; endogenous preproglucagon derived peptide; modulates feeding and metabolism
2095 PNU 37883 hydrochloride
Vascular Kir6 (KATP) channel blocker
2096 DAU 5884 hydrochloride
M3 receptor antagonist
2097 SKI II
Selective non-lipid inhibitor of sphingosine kinase
2098 Apoptosis Activator 2
Promotes apoptosome formation and activates caspase-9/caspase-3 pathway. Selectively induces tumor cell apoptosis

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