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Displaying Products by Catalog Number (3200 - 3299)

Cat. No. Product Name / Activity
3200 XAC
Adenosine receptor antagonist
3201 Dimebon dihydrochloride
Neuroprotectant; protects against β-amyloid neurotoxicity
3202 Echistatin, α1 isoform
αVβ3 and glycoprotein IIb/IIIa (integrin αIIbβ3) inhibitor
3203 Celastrol
Inhibits TNF-α-induced NF-κB activation
3206 Doxercalciferol
Vitamin D2 analog, VDR agonist
3207 Kifunensine
Inhibitor of class I α-mannosidases
3208 Swainsonine
Inhibitor of α-mannosidase II
3209 α,β-Methyleneadenosine 5'-triphosphate trisodium salt
Non-selective P2 agonist
3211 SB 525334
Selective inhibitor of TGF-βRI
3212 CP 376395 hydrochloride
Potent and selective CRF1 antagonist; binds at an allosteric site
3213 Methylene Blue
Biological stain
3214 RETRA hydrochloride
Antitumor agent; suppresses mutant p53-bearing cancer cells
3215 ZIP (Scrambled)
Control peptide for ZIP (Cat. No. 2549)
3219 CGP 36216 hydrochloride
GABAB antagonist; displays activity at presynaptic receptors
3220 ShK-Dap22
Extremely potent and selective KV1.3 blocker; suppresses T cell activation in vitro
3221 bPiDDB
Orthosteric neuronal nAChR antagonist
3222 TCS JNK 6o
Selective JNK inhibitor
3225 Lys-[Des-Arg9]Bradykinin
Selective B1 agonist
3226 R 892
Potent and selective B1 antagonist
3228 [Lys5,MeLeu9,Nle10]-NKA(4-10)
Selective NK2 agonist
3229 [Phe8Ψ(CH-NH)-Arg9]-Bradykinin
Selective B2 agonist
3230 Sar-[D-Phe8]-des-Arg9-Bradykinin
Potent and selective B1 agonist
3231 Ac9-25
Annexin I N-terminal peptide; acts as a FPR1 ligand
3233 AGK 2
Selective SIRT2 inhibitor
3235 CDPPB
Positive allosteric modulator of mGlu5 receptors
3236 PACAP 6-38
Potent PAC1 receptor antagonist
3237 BIM 23042
Selective neuromedin B receptor antagonist (NMB-R, BB1)
3238 TCS PrP Inhibitor 13
Antiprion agent; inhibits PrPSc accumulation
3239 PF 573228
Potent and selective FAK inhibitor
3240 SCH 221510
Potent and selective NOP agonist
3241 Ko 143
Potent and selective BCRP inhibitor
3242 BMS 193885
Potent, competitive NPY Y1 receptor antagonist
3245 ATP disodium salt
P2 agonist
3246 LY 354740
Potent and highly selective group II mGlu agonist
3248 VU 0155041
Potent positive allosteric modulator of mGlu4 receptors
3249 Z-Cyclopentyl-AP4
Group III mGlu agonist (mGlu4 > mGlu8 > mGlu7)
3250 L-838,417
GABAA partial agonist; displays subtype selectivity
3251 KC 12291 hydrochloride
Orally active atypical Na+ channel blocker; cardioprotective
3252 WWL 70
Potent ABHD6 inhibitor
3253 Triptolide
Inhibits RNAPII-mediated transcription; antitumor, anti-inflammatory and immunosuppressive
3254 Ro 61-8048
Potent kynurenine 3-monooxygenase (KMO) inhibitor
3255 PJ 34 hydrochloride
Potent PARP inhibitor
3256 Metoprolol tartrate
Selective β1 antagonist
3257 5-Fluorouracil
Thymidylate synthetase inhibitor
3258 Mitomycin C
DNA cross-linking antitumor agent
3259 Gemcitabine hydrochloride
DNA synthesis inhibitor
3260 Epirubicin hydrochloride
Inhibits DNA synthesis and function. Inhibits DNA topoisomerase II
3262 JNJ 1661010
Selective, reversible FAAH inhibitor
3263 SB 505124
Selective inhibitor of TGF-βRI, ALK4 and ALK7
3264 GW 788388
Potent and selective inhibitor of TGF-βRI
3265 SB 452533
Potent TRPV1 receptor antagonist
3266 GLP-1 (9-36) amide
Metabolite of GLP-1-(7-36) (Cat. No. 2082)
3267 Thiostrepton
Antibiotic, inhibits protein synthesis
3268 Minocycline hydrochloride
Antibiotic. Displays neuroprotective effects
3269 SD 208
Potent ATP-competitive TGF-βRI inhibitor
3270 GIT 27
Immunomodulator; reduces production of pro-inflammatory cytokines
3271 Compound 401
Selective DNA-PK and mTOR inhibitor
3272 (±)-LY 395756
Mixed mGlu2 agonist/ mGlu3 antagonist
3276 Mephenytoin
CYP2C19 substrate. Anticonvulsant
3277 Pentamidine isethionate
NMDA antagonist: antimicrobial
3278 YM 511
Potent aromatase (CYP19) inhibitor
3279 UTPγS trisodium salt
Selective P2Y2/4 agonist
3280 2-ThioUTP tetrasodium salt
Potent and selective P2Y2 agonist
3281 Canrenone
Mineralocorticoid receptor antagonist
3282 NAD 299 hydrochloride
Selective, high affinity 5-HT1A antagonist
3283 LY 487379 hydrochloride
Selective positive allosteric modulator of mGlu2 receptors
3284 Rec 15/2615 dihydrochloride
Selective α1B antagonist
3285 NPS ALX Compound 4a dihydrochloride
Potent and selective 5-HT6 antagonist
3286 Milnacipran hydrochloride
5-HT and NA reuptake inhibitor (SNRI)
3287 Prochlorperazine dimaleate
D2 receptor antagonist; also 5-HT3 and nAChR antagonist
3290 ZIP, Biotinylated
Biotinylated peptide for ZIP (Cat. No. 2549)
3291 PF 915275
Potent and selective 11β-hydroxysteroid dehydrogenase inhibitor
3292 Metyrapone
11-β hydroxylase inhibitor
3293 Finasteride
Type II 5α-reductase inhibitor
3295 RG 108
Non-nucleoside DNA methyltransferase inhibitor
3296 AP 18
Reversible TRPA1 channel blocker
3297 SSR 146977 hydrochloride
Potent and selective NK3 antagonist
3298 NGD 94-1
Selective D4 receptor ligand
3299 AMD 3100 octahydrochloride
Highly selective CXCR4 antagonist

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