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Displaying Products by Catalog Number (1200 - 1299)

Cat. No. Product Name / Activity
1200 Nω-Propyl-L-arginine hydrochloride
Highly selective inhibitor of nNOS
1201 Phorbol 12-myristate 13-acetate
Protein kinase C activator
1202 SB 203580
Selective inhibitor of p38 MAPK
1203 MRS 2219
Potentiates P2X1-mediated responses
1205 SR 57227 hydrochloride
Potent and selective 5-HT3 agonist
1206 SC 19220
Selective EP1 receptor antagonist
1207 BRL 15572 hydrochloride
Selective h5-HT1D antagonist
1208 (2R,4R)-APDC
Highly selective group II agonist
1209 LY 341495
Highly potent and selective group II mGlu antagonist
1210 FR 139317
Highly potent, selective ETA antagonist
1211 ZD 7155 hydrochloride
Selective non-peptide AT1 antagonist
1212 MPEP hydrochloride
Potent mGlu5 antagonist; also positive allosteric modulator of mGlu4 receptors
1213 PD 98059
MEK inhibitor
1214 SIB 1893
mGlu5 antagonist; also positive allosteric modulator at mGlu4 receptors
1215 SIB 1757
Highly selective mGlu5 antagonist
1217 MRS 1220
Highly potent and selective hA3 antagonist
1218 DH 97
MT2 receptor antagonist
1219 IDRA 21
Inhibits AMPA desensitization
1220 (RS)-PPG
Potent and selective mGlu8 agonist
1221 SB 224289 hydrochloride
Selective 5-HT1B antagonist
1222 DMPQ dihydrochloride
Potent, selective inhibitor of PDGFRβ
1223 DL-TBOA
Selective non-transportable inhibitor of EAATs
1224 2-APB
IP3 receptor antagonist. Also TRP channel modulator
1225 TCPOBOP
Constitutive androstane receptor agonist
1226 Etoposide
Topoisomerase II inhibitor
1227 Apigenin
Protein kinase inhibitor
1228 Nocodazole
Microtubule inhibitor
1229 Actinomycin D
Inhibits RNA polymerase
1230 Methotrexate
Cytotoxic agent
1231 Brefeldin A
Disrupts protein translocation to Golgi
1232 Wortmannin
Potent, irreversible inhibitor of PI 3-kinase. Also inhibitor of PLK1
1233 Cytochalasin D
Disrupts actin filament function
1234 A23187, free acid
Calcium ionophore
1235 Cyclopiazonic acid
Inhibitor of SERCA ATPase
1236 BHQ
Inhibitor of SERCA ATPase
1237 LY 367385
Selective mGlu1a antagonist
1238 CCMQ
Used to characterize GluN2B-containing NMDA receptors
1239 Ac-RYYRIK-NH2
High affinity NOP ligand
1240 NF 023
Selective, competitive P2X1 antagonist
1241 CGS 19755
Potent competitive NMDA antagonist
1242 SB 216641 hydrochloride
Selective h5-HT1B antagonist
1243 (+)-PD 128907 hydrochloride
High affinity D3 agonist (D3 ≥ D2 > D4)
1244 KB-R7943 mesylate
Na+/Ca2+ exchange inhibitor (reverse mode)
1245 CGP 35348
Selective GABAB antagonist; brain penetrant
1246 CGP 52432
Potent and selective GABAB antagonist
1247 CGP 46381
Selective GABAB antagonist; brain penetrant
1248 CGP 55845 hydrochloride
Potent and selective GABAB antagonist
1249 CY 208-243
Selective D1-like agonist
1250 SDZ 220-581
Competitive NMDA antagonist
1251 SDZ 220-040
Potent competitive NMDA antagonist
1253 (S)-WAY 100135 dihydrochloride
Potent and selective 5-HT1A antagonist
1254 Y-27632 dihydrochloride
Selective ROCK inhibitor; inhibits ROCK1 (p160 ROCK) and ROCK2; stem cell freezing (cryopreservation) media component
1255 SDZ SER 082 fumarate
Selective 5-HT2B/2C antagonist
1256 Vinblastine sulfate
Disrupts microtubules
1257 Vincristine sulfate
Disrupts microtubules
1258 1-Deoxynojirimycin
Glucosidase I and II inhibitor
1259 1-Deoxymannojirimycin hydrochloride
α-Mannosidase I inhibitor
1260 Ivermectin
Positive allosteric modulator of α7 nAChRs; also positive allosteric modulator of P2X4 receptors
1261 EHNA hydrochloride
Adenosine deaminase inhibitor
1262 SR 95531 hydrobromide
Competitive and selective GABAA antagonist
1263 GR 144053 trihydrochloride
Glycoprotein IIb/IIIa (integrin αIIbβ3) receptor antagonist. Antithrombotic
1264 SB 202190
Potent, selective inhibitor of p38 MAPK
1265 D-CPP-ene
Potent competitive NMDA antagonist
1266 Nociceptin (1-7)
Bioactive metabolite of nociceptin
1267 Pifithrin-α hydrobromide
p53 inhibitor. Also aryl hydrocarbon receptor agonist
1268 U 73122
Phospholipase C inhibitor
1269 PD 150606
Cell permeable calpain inhibitor
1271 RJR 2429 dihydrochloride
nAChR agonist; displays selectivity for α4β2, α1βγδ and α3β4 subtypes
1274 GR 159897
Non-peptide, potent NK2 antagonist
1276 AG 1478 hydrochloride
Highly potent EGFR-kinase inhibitor
1277 KN-62
Non-competitive P2X7 antagonist
1278 KN 93
CaM kinase II inhibitor; also K+ channel blocker (KV)
1280 (-)-Xestospongin C
Reported inhibitor of IP3-dependent Ca2+ release
1282 GNTI dihydrochloride
Potent, selective κ antagonist
1283 ARL 67156 trisodium salt
NTPDase inhibitor
1284 Olomoucine
Cdk inhibitor
1285 Staurosporine
Non-selective protein kinase inhibitor
1286 LY 231617
Antioxidant; neuroprotective in vitro and in vivo
1288 KT 5720
Selective protein kinase A inhibitor
1289 KT 5823
Selective protein kinase G inhibitor
1290 Anisomycin
JNK, SAPK and p38 activator
1291 Ochratoxin A
Stimulates SERCA-ATP-dependent Ca2+ pump activity
1292 Rapamycin
mTOR inhibitor; immunosuppressant
1293 β-Lapachone
DNA topoisomerase I inhibitor
1295 Loreclezole hydrochloride
Subtype-selective GABAA modulator
1296 CI 966 hydrochloride
Selective inhibitor of GAT-1
1297 Abn-CBD
Selective GPR55 agonist; neurobehaviorally inactive
1298 2-Arachidonylglycerol
Endogenous and non-selective CB agonist; potent GPR55 agonist

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