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Displaying Products by Catalog Number (4100 - 4199)

Cat. No. Product Name / Activity
4100 HC 067047
Potent and selective TRPV4 antagonist
4102 Mycophenolate mofetil
Inosine monophosphate dehydrogenase inhibitor
4103 6-Mercaptopurine
Purine analog; inhibits DNA and RNA synthesis
4105 CIQ
Potentiator of NMDA receptors containing GluN2C/GluN2D
4106 Nicotinamide
PARP-1 inhibitor
4107 Probenecid
MRP inhibitor
4108 Quinidine
Blocks sodium and potassium channels
4109 Chloroquine diphosphate
Antimalarial; inhibits apoptosis and autophagy
4110 Oligomycin A
Inhibitor of mitochondrial ATPase
4111 Hexamethonium bromide
Non-competitive nAChR antagonist
4112 Niflumic acid
Cyclooxygenase-2 (COX-2) inhibitor; GPR35 agonist
4113 Fenofibrate
PPARα agonist
4114 Quinine hydrochloride
Antimalarial
4115 Mometasone furoate
Synthetic corticosteroid; anti-inflammatory agent
4116 GSK 9027
Glucocorticoid receptor agonist
4117 Bepridil hydrochloride
Non-selective Ca2+ channel blocker; also NCX inhibitor
4118 SB 772077B dihydrochloride
Potent Rho-kinase inhibitor; vasodilator
4119 Cinnabarinic acid
Selective mGlu4 agonist
4120 Xanthurenic acid
Selectively activates group II mGlu receptors
4121 Rifampicin
Pregnane X receptor agonist; antibiotic
4123 C3bot (154-182)
Neurotrophic fragment of clostridial C3 protein
4124 Pioglitazone hydrochloride
Selective PPARγ agonist; antidiabetic agent
4126 DMH-1
Selective ALK2 inhibitor
4127 Salermide
SIRT1 and SIRT2 inhibitor
4128 Bisindolylmaleimide II
Potent PKC inhibitor; also potent nAChR antagonist
4130 KN 92
Inactive analog of KN 93. K+ channel (Kv) blocker
4131 G418 disulfate salt
Aminoglycoside antibiotic; used in cell culture
4132 XMD 8-92
ERK5/BMK1 inhibitor; also BRD4 inhibitor
4133 U 73343
Analog of U 73122 (Cat. No. 1268)
4134 NPS 2390
Group I mGlu antagonist
4136 Conantokin G
GluN2B-selective NMDA antagonist
4137 Hygromycin B
Aminoglycoside antibiotic; active against prokaryotic and eukaryotic cells
4138 ABT 751
Inhibitor of microtubule polymerization; antimitotic and antitumor
4139 Aprotinin
Competitive serine protease inhibitor
4140 EB 47
Potent PARP-1 inhibitor
4141 LY 2087101
Allosteric potentiator of α7, α4β2 and α4β4 nAChRs
4143 GSK 2334470
Highly potent, selective PDPK1 (PDK1) inhibitor
4144 GSK 690693
Akt kinase inhibitor. Antitumor
4145 PK 44 phosphate
Potent and selective dipeptidyl peptidase IV (DPP-IV) inhibitor
4146 Ercalcidiol
Metabolite of vitamin D2
4148 Abacavir hemisulfate
Reverse transcriptase inhibitor; antiretroviral
4149 Delavirdine mesylate
Non-nucleoside reverse transcriptase inhibitor
4150 Azidothymidine
Selective reverse transcriptase inhibitor; antiretroviral
4152 TMN 355
Cyclophilin A inhibitor
4153 Phorbol 12,13-dibutyrate
Protein kinase C activator
4154 TCN 201
GluN1/GluN2A-selective NMDA antagonist
4156 Vitamin D3
Precursor of calcifediol (Cat. No. 4036). Naturally occurring form of vitamin D
4157 Tacalcitol
Synthetic vitamin D3 (Cat. No. 4156) analog
4159 Alfacalcidol
Prodrug of vitamin D3 (Cat. No. 4156)
4160 22-Oxacalcitriol
Non-calcemic vitamin D3 (Cat. No. 4156) analog
4161 Paricalcitol
Analog of the active form of vitamin D2
4163 TCN 213
NMDA antagonist; selective for GluN2A over GluN2B containing receptors
4165 Gisadenafil besylate
Potent PDE5 inhibitor; orally bioavailable
4166 NS 5806
KV4.3 channel activator
4167 KW 3902
Selective A1 antagonist
4168 PIT 1
PIP3 antagonist. Blocks PIP3-PH interaction; inhibits Akt signaling
4169 KS 176
Selective BCRP inhibitor
4171 VU 0364739 hydrochloride
Potent and selective PLD2 inhibitor
4172 ML 145
GPR35 antagonist
4173 MDL 100907
Potent and selective 5-HT2A antagonist
4174 Pramipexole dihydrochloride
Selective D3 agonist
4175 PF 3845
Selective FAAH inhibitor
4177 AS 1269574
GPR119 receptor agonist
4179 AMD 3465 hexahydrobromide
Potent and selective CXCR4 antagonist
4180 Beraprost sodium
Potent prostacyclin IP receptor agonist
4181 Ro 3306
Cdk1 inhibitor
4184 Torcetrapib
Inhibitor of cholesteryl ester transfer protein (CETP)
4185 Sonepiprazole
Selective D4 antagonist
4186 UK 5099
MCT inhibitor; also inhibits of pyruvate transport
4187 UK 356618
Potent and selective MMP-3 inhibitor
4188 UK 383367
Potent and selective BMP-1 (PCP) inhibitor
4189 SC 26196
Selective fatty acid desaturase 2 inhibitor
4190 CP 775146
Selective, high affinity PPARα agonist
4191 PF 3716556
Selective H+,K+-ATPase inhibitor
4192 PD 0325901
Potent inhibitor of MEK1/2
4193 CP 100356 hydrochloride
P-gp inhibitor
4194 WY 45233 succinate
5-HT and NA reuptake inhibitor (SNRI)
4195 VPC 23019
S1P1 and S1P3 antagonist
4196 HA 130
Potent and selective autotaxin inhibitor
4197 VU 591 hydrochloride
Selective Kir1.1 (ROMK) inhibitor
4198 IEM 1925 dihydrobromide
Voltage- and use-dependent open-channel AMPA blocker
4199 IEM 1754 dihydrobromide
Voltage-dependent, open-channel AMPA blocker

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