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Displaying Products by Catalog Number (6100 - 6199)

Cat. No. Product Name / Activity
6100 Fasentin
GLUT1/GLUT4 inhibitor; also Fas-sensitizer
6101 SHIP 2a
Cystathione γ lyase (CSE) inhibitor
6102 Ep23, 5'-DY647
High affinity fluorescently tagged aptamer for EpCam
6103 CD133-A15, 5'-DY647
High affinity fluorescently tagged aptamer for CD133 (AC133 epitope)
6104 CD133-B19, 5'-DY647
High affinity fluorescently tagged aptamer for CD133 (extracellular domain epitope)
6105 TC AC 28
High affinity BET bromodomain ligand
6106 T 3364366
Potent and reversible fatty acid desaturase 1 inhibitor; orally bioavailable
6107 CP 424174
Inhibitor of IL-1β post-translational processing; indirectly inhibits NLRP3
6108 Galeterone
CYP17 inhibitor; also androgen receptor antagonist
6109 Methylnaltrexone bromide
μ antagonist; peripherally restricted
6110 HJC 0416 hydrochloride
STAT3 inhibitor
6111 Zoledronic Acid
Potent farnesyl diphosphate (FPP) synthase inhibitor
6112 (S)-Norketamine hydrochloride
NMDA receptor modulator; analgesic
6113 Liproxstatin-1 hydrochloride
Potent ferroptosis inhibitor
6114 PF 06409577
Potent and selective allosteric activator of AMPK
6115 PF 06273340
Potent and selective pan-Trk inhibitor; peripherally restricted
6116 BHPI
ERα antagonist; also activates unfolded protein response; active in vivo
6117 CORM 2
Carbon monoxide-releasing molecule
6118 1S,3R-RSL3
Induces ferroptosis; inhibits glutathione peroxidase 4 (GPX4)
6119 OB 24 hydrochloride
Potent and selective heme oxygenase 1 (HO-1) inhibitor
6121 NB-caged Tyrosine hydrochloride
ortho-nitrobenzyl caged L- tyrosine
6124 (R)-2-Hydroxyglutaric acid disodium salt
KDM4A inhibitor; also NF-κB activator
6125 TC JL 37
Potent TYK2 inhibitor
6126 KRH 3955 hydrochloride
Highly potent CXCR4 antagonist; inhibits HIV-1 replication
6128 GSK 343
Potent and selective SAM-competitive EZH2 inhibitor
6131 (R)-Modafinil
Dopamine uptake inhibitor
6132 NVS PAK1 1
Potent and selective PAK1 inhibitor
6133 NVS PAK1 C
Negative control of NVS PAK1 1 (Cat. No. 6132)
6134 T 26c disodium salt
Highly potent and selective MMP13 inhibitor
6137 8-Cyclopentyl-1,3-dimethylxanthine
High affinity adenosine A1 receptor antagonist
6138 SR 9243
Selective LXR inverse agonist
6139 NS 6740
High affinity α7 nAChR partial agonist; anti-inflammatory
6142 CL 075
TLR8 agonist
6143 WZB 117
GLUT inhibitor
6144 CX08005
Competitive PTP1B inhibitor
6146 LAP
Photocrosslinker for hydrogels
6147 Janelia Fluor® 549, SE
Yellow dye (Reactive group: NHS ester). Applications: super resolution microscopy e.g. dSTORM & STED, confocal, flow and live cell imaging
6148 Janelia Fluor® 646, SE
Red dye (Reactive group: NHS ester). Applications: super resolution microscopy e.g. dSTORM & STED, confocal, flow and live cell imaging
6149 PA Janelia Fluor® 549, SE
Yellow photoactivatable dye (Reactive group: NHS ester). Applications: super resolution microscopy (PALM), single molecule tracking and live cell imaging
6150 PA Janelia Fluor® 646, SE
Red photoactivatable dye (Reactive group: NHS ester). Applications: super resolution microscopy (PALM), single molecule tracking and live cell imaging
6151 LDN 212854
Potent bone morphogenetic protein type I (ALK) inhibitor
6152 LDN 214117
Potent and selective ALK2 inhibitor
6153 JQEZ5
Potent and selective SAM-competitive EZH2 inhibitor
6154 MZ 1
(+)-JQ1 based PROTAC that selectively degrades BRD4 in cells
6155 cis MZ 1
Negative Control for MZ 1 (Cat. No. 6154)
6156 VH 298
High-affinity inhibitor of VHL
6157 cis VH 298
Negative control for VH 298
6158 (S)-Equol
Potent estrogen receptor β (ERβ) agonist; dihydrotestosterone antagonist
6159 4,9-Anhydrotetrodotoxin
Potent and selective Nav1.6 channel blocker
6160 VE 821
High affinity and selective ATP-competitive ATR inhibitor
6161 Ailanthone
Potent inhibitor of androgen receptor (AR)
6162 TAPI 1
ADAM-17 (TACE) and MMP inhibitor
6163 AR 420626
FFA3 agonist
6164 SEA 0400
Potent Na+/Ca2+ exchanger (NCX) inhibitor
6165 AC 265347
Biased allosteric modulator of calcium-sensing receptor (CaSR)
6166 AMG 18 hydrochloride
Potent and selective IRE1α inhibitor
6167 A 196
Potent and selective SUV420H1/H2 inhibitor
6168 RI 1
RAD51 recombinase inhibitor
6169 PF 06726304 acetate
Highly potent and SAM-competitive EZH2 inhibitor
6170 Cinacalcet hydrochloride
Allosteric Calcium-sensing receptor (CaSR) agonist; also CYP2D2 inhibitor and Ca2+ channel blocker; orally bioavailable
6171 MLS 1547
G protein-biased D2 partial agonist
6172 INF 4E
Caspase-1 and NLRP3 inflammasome inhibitor
6174 CVT 313
Cdk2 and cdk5 inhibitor
6175 DBHDA
Reagent for synthetic biology; converts cysteine to dehydroalanine
6176 FTY 720
Potent S1P receptor agonist; also immunosuppressant
6177 AZ 13705339
Highly potent PAK1 and PAK2 inhibitor
6179 UK 59811 hydrochloride
CaVAb blocker
6180 NMS 873
Potent and selective p97 ATPase (VCP) allosteric inhibitor
6181 OTX 015
BET bromodomain inhibitor; orally bioavailable
6182 Pimonidazole
Hypoxia detection reagent
6185 Pemetrexed
Thymidylate synthetase inhibitor, also inhibits dihydrofolate reductase, GARFT and AICART
6187 SK 216
Plasminogen activator inhibitor-1 (PAI-1) inhibitor
6188 Everolimus
mTOR inhibitor; Immunosuppressant
6189 Myricetin
Irreversible TrxR inhibitor
6191 TH 1020
Toll-like receptor (TLR) 5/Flagellin complex antagonist
6192 PZ-II-029
α6β3γ2-selective GABAA positive allosteric modulator
6193 AM 4113
High affinity and selective CB1 antagonist
6194 TM 5441
Plasminogen activator inhibitor-1 (PAI-1) inhibitor
6195 SSR 149415
Potent and selective vasopressin V1B antagonist
6196 Brequinar sodium
Potent and selective DHODH inhibitor
6198 GSK 6853
Potent and selective BRPF1 inhibitor
6199 BAY 876
Potent and selective GLUT1 inhibitor

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