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Displaying Products Alphabetically by Name (R)

Cat. No. Product Name / Activity
6530 R 121919 hydrochloride
High affinity CRF1 antagonist; orally bioavailable
5288 R 268712
Potent and selective inhibitor of TGF-βRI
5494 R 547
Potent and selective cdk inhibitor; orally bioavailable
3815 R 568 hydrochloride
Positive allosteric modulator of human calcium-sensing receptor (CaSR)
5432 R 7050
Inhibitor of TNF-α receptor 1 signaling
3407 R 715
Potent and selective B1 antagonist
1742 R-96544 hydrochloride
Potent, selective 5-HT2A antagonist
2144 R18
Inhibitor of 14.3.3 proteins
7129 RA 2
Potent negative modulator of KCa2.3 and KCa3.1 channels
5707 RA 839
Nrf2 activator; inhibits Nrf2/Keap1 interaction
6649 RADA
Orange-red TAMRA-based fluorescent D-amino acid for labeling peptidoglycans in live bacteria
7701 RAGE 229
ctRAGE-DIAPH1 interaction antagonist; reduces inflammatory signaling in diabetic mice
6259 RAGE antagonist peptide
RAGE antagonist
5411 RBC8
RalA and RalB inhibitor
7066 RCGD 423
gp130 modulator; activates JAK/STAT signaling
6845 RCM 1
FOXM1 inhibitor
IKBKAP pre-mRNA splicing modulator
3672 RF 9
Selective NPFF1 and NPFF2 antagonist
4683 RFRP 3 (human)
NPFF1 agonist; GnIH homolog
3295 RG 108
Non-nucleoside DNA methyltransferase inhibitor
7723 RGD peptide
Minimal recognition sequence for integrin binding; potent integrin inhibitor
3498 RGDS peptide
Integrin binding sequence; inhibits integrin receptor function
6728 RGFP 966
Potent and selective HDAC3 inhibitor
1842 RHC 80267
Diacylglycerol lipase inhibitor
5311 RHPS 4 methosulfate
Telomerase inhibitor
7339 RIPA 56
Potent and metabolically stable RIP1 kinase inhibitor
RIPK2 modulator; pro-drug of cRIPGM; orally bioavailable and brain penetrant
6603 RIPK2 inhibitor 1
Potent RIPK2 inhibitor
2443 RITA
MDM2-p53 interaction inhibitor
1053 RJR 2403 oxalate
Selective α4β2 nAChR agonist
5061 RKI 1447 dihydrochloride
Potent and selective ROCK inhibitor; antitumor
3393 RLLFT-NH2
Control peptide for TFLLR-NH2 (Cat. No. 1464)
8013 RMR-Tre
Far-red fluorogenic trehalose probe for live mycobacteria imaging
4977 RN 1 dihydrochloride
LSD1 inhibitor
3746 RN 1734
Selective TRPV4 antagonist
3745 RN 1747
Selective TRPV4 agonist
5678 RN 9893 hydrochloride
Potent and selective TRPV4 antagonist
6833 RO 5263397 hydrochloride
Potent TA1 receptor agonist
7375 RO 8191
IFNα receptor 2 agonist
3052 RO-3
Selective P2X3 and P2X2/3 antagonist
4289 RP 001 hydrochloride
Potent S1P1 agonist
8031 RP 6306
Potent and selective PKMYT1 inhibitor
1635 RP 67580
Potent and selective NK1 antagonist
5388 RQ 00203078
Potent and selective TRPM8 antagonist; orally active
1325 RS 100329 hydrochloride
Potent, subtype-selective α1A antagonist
1050 RS 102221 hydrochloride
Selective 5-HT2C antagonist
2089 RS 102895 hydrochloride
CCR2b chemokine receptor antagonist
2993 RS 127445 hydrochloride
High affinity and selective 5-HT2B antagonist
0985 RS 17053 hydrochloride
α1A antagonist
0728 RS 23597-190 hydrochloride
5-HT4 antagonist
0991 RS 39604 hydrochloride
5-HT4 antagonist
2517 RS 504393
Highly selective CCR2 chemokine receptor antagonist
0987 RS 79948 hydrochloride
Potent and selective α2 antagonist
6687 1R,3R-RSL3
Negative control for 1S,3R-RSL3 (Cat. No. 6118)
6118 1S,3R-RSL3
Inhibits glutathione peroxidase (GPX4); induces ferroptosis
0912 RU 24969 hemisuccinate
5-HT1A and 5-HT1B agonist
1672 RU 28318, potassium salt
Potent, selective mineralocorticoid receptor antagonist
7904 RU.521
Potent and selective inhibitor of cyclic GMP-AMP synthase (cGAS)
2614 RWJ 56110
Selective PAR1 antagonist
2999 RWJ 67657
Potent, selective p38α and p38β inhibitor
1324 RX 821002 hydrochloride
Potent, selective α2D antagonist
1810 Raclopride
Potent and selective D2 and D3 antagonist
1589 Radicicol
Hsp90 inhibitor. Antifungal antibiotic
2280 Raloxifene hydrochloride
Selective estrogen receptor modulator (SERM)
5250 Ramipril
Non-peptide, competitive angiotensin-converting enzyme (ACE) inhibitor
3118 Ranolazine dihydrochloride
Antianginal, activates pyruvate dehydrogenase
1292 Rapamycin
mTOR inhibitor; immunosuppressant
6760 Raphin 1
Inhibitor of the regulatory subunit PPP1R15B of protein phosphatase 1; orally bioavailable and brain penetrant
4308 Rasagiline mesylate
Selective and irreversible MAO-B inhibitor
1982 Reboxetine mesylate
Potent and selective noradrenalin uptake inhibitor; orally active
7226 Remdesivir
Viral RNA-dependent RNA polymerase (RdRP) inhibitor; broad spectrum antiviral nucleotide prodrug
5193 Remodelin
N-acetyltransferase 10 (NAT10) inhibitor
3742 RepSox
Potent and selective inhibitor of TGF-βRI
TB3742-RMU RepSox
RepSox synthesized to Ancillary Material Grade
3805 Repaglinide
Kir6 (KATP) channel blocker
6957 Reparixin L-lysine salt
Potent CXCR1 and CXCR2 allosteric antagonist
2742 Reserpine
Inhibitor of vesicular monoamine transport
4536 Resiquimod
Toll-like receptor 7 (TLR7) agonist
1418 Resveratrol
Cyclooxygenase inhibitor
6233 Retigabine
KV7 channel activator
0695 Retinoic acid
Endogenous retinoic acid receptor agonist
3722 Reversan
Selective MRP1 and P-gp inhibitor
7406 Rf470DL
Blue rotor-fluorogenic fluorescent D-amino acid for labeling peptidoglycans in live bacteria
6867 Rhein
FTO (mRNA N6-methyladenine demethylase) inhibitor; also inhibits ALKBH2 and ALKBH3
5003 Rhosin hydrochloride
Rho inhibitor
4501 Ribavirin
Blocks eIF4E activity; antiviral guanosine analog
7050 Ribociclib
Dual cdk4/cdk6 inhibitor; orally bioavailable
0790 Rilmenidine hemifumarate
I1 ligand. Also α2 agonist
7684 Rilpivirine
Non-nucleoside reverse transcriptase inhibitor
0768 Riluzole hydrochloride
GABA uptake inhibitor; also inhibits glutamate release and blocks NaV channels
1497 Rimcazole dihydrochloride
σ2 antagonist. Also DAT inhibitor
7916 Risdiplam
Selective SMN2 gene splicing modifier
3504 Risedronate
Farnesyl diphosphate (FPP) synthase inhibitor
2865 Risperidone
5-HT2A antagonist; also D2 antagonist; atypical antipsychotic
1955 Ritanserin
Potent 5-HT2 antagonist
5856 Ritonavir
HIV-1 and HIV-2 protease inhibitor
4440 Rivastigmine tartrate
Dual AChE and BChE inhibitor
2272 Ro 08-2750
Inhibits NGF binding to p75NTR and TrkA
1997 Ro 15-4513
Benzodiazepine partial inverse agonist
0415 Ro 20-1724
PDE4 inhibitor
1594 Ro 25-6981 maleate
GluN2B-selective NMDA antagonist
2002 Ro 31-8220 mesylate
Protein kinase inhibitor
1587 Ro 32-0432 hydrochloride
Potent, orally active PKC inhibitor
4181 Ro 3306
Cdk1 inhibitor
5389 Ro 48-8071 fumarate
2,3-Oxidosqualene cyclase (OSC) inhibitor; blocks cholesterol synthesis
4694 Ro 5-3335
Core binding factor inhibitor; attenuates hematopoiesis
4391 Ro 51
Potent P2X3 and P2X2/3 antagonist
1854 Ro 60-0175 fumarate
Potent, selective 5-HT2C agonist
3254 Ro 61-8048
Potent kynurenine 3-monooxygenase (KMO) inhibitor
2913 Ro 64-5229
Selective, non-competitive mGlu2 antagonist
4347 Ro 67-4853
Positive allosteric modulator of group I mGlu receptors
4346 Ro 67-7476
Positive allosteric modulator of mGlu1 receptors
5913 Ro 6842262
Potent LPA1 antagonist
2408 Ro 90-7501
Inhibitor of Aβ42 fibril formation
0905 Rolipram
PDE4 inhibitor
1349 (R)-(-)-Rolipram
PDE4 inhibitor. More active enantiomer of rolipram (Cat. No. 0905)
3680 Ropinirole
Selective D2-like agonist
1332 Roscovitine
5325 Rosiglitazone
Potent and selective PPARγ agonist; antidiabetic agent
5315 Rostafuroxin
Na+/K+ ATPase modulator; antihypertensive agent
6343 Rosuvastatin calcium
Potent HMG-CoA reductase inhibitor
3616 Rotenone
Inhibits complex I of the mitochondrial electron transport chain
3896 Rotigotine hydrochloride
D2 and D3 agonist
1610 Rottlerin
Reported PKCδ inhibitor
7486 Roxadustat
HIF-PH inhibitor; erythropoietic
5524 Rp-8-pCPT-cGMPS sodium
PKG inhibitor
3400 RuBi-GABA
Caged GABA; excitable at visible wavelengths
3574 RuBi-Glutamate
Caged glutamate; excited by visible wavelengths
3855 RuBi-Nicotine
Caged nicotine; rapidly excitable by visible light
4709 RuBi GABA trimethylphosphine
Caged GABA; inhibits neural activity
6230 Rucaparib camsylate
PARP inhibitor
3828 Rufinamide
Prolongs inactivation of sodium channels; anticonvulsant
1439 Ruthenium Red
Non-selective CaV2.1 and 2.2 blocker; also blocks TRPV channels
7064 Ruxolitinib
Potent and selective JAK1/JAK2 inhibitor; orally bioavailable
7048 Ruxolitinib phosphate
Phosphate salt of Ruxolitinib (Cat. No. 7064); potent and selective JAK1/JAK2 inhibitor
1329 Ryanodine
Ca2+ release inhibitor
2609 Ryuvidine
SETD8 inhibitor; also CDK4 inhibitor

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