All ProductsDisplaying Products Alphabetically by Name (R)
| Cat. No. | Product Name / Activity |
|---|---|
| 6530 | R 121919 hydrochloride |
| High affinity CRF1 antagonist; orally bioavailable | |
| 4885 | R 1530 |
| Multi-RTK inhibitor; inhibits angiogenesis | |
| 5288 | R 268712 |
| Potent and selective inhibitor of TGF-βRI | |
| 5494 | R 547 |
| Potent and selective cdk inhibitor; orally bioavailable | |
| 3815 | R 568 hydrochloride |
| Positive allosteric modulator of human calcium-sensing receptor (CaSR) | |
| 2194 | R 59-022 |
| Diacylglycerol kinase inhibitor; increases PKC activity | |
| 5432 | R 7050 |
| Inhibitor of TNF-α receptor 1 signaling | |
| 3407 | R 715 |
| Potent and selective B1 antagonist | |
| 3226 | R 892 |
| Potent and selective B1 antagonist | |
| 1742 | R-96544 hydrochloride |
| Potent, selective 5-HT2A antagonist | |
| 6048 | R-BC154 |
| High affinity fluorescent α4β1/α9β1 inhibitor; mobilizes HSCs | |
| 2144 | R18 |
| Inhibitor of 14.3.3 proteins | |
| 1577 | L-R4W2 |
| TRPV1 antagonist peptide | |
| 7129 | RA 2 New |
| Potent negative modulator of KCa2.3 and KCa3.1 channels | |
| 5707 | RA 839 |
| Nrf2 activator; inhibits Nrf2/Keap1 interaction | |
| 6649 | RADA |
| Orange-red TAMRA-based fluorescent D-amino acid for labeling peptidoglycans in live bacteria | |
| 6015 | RAF 265 |
| Raf kinase and VEGFR-2 inhibitor | |
| 6259 | RAGE antagonist peptide |
| RAGE antagonist | |
| 5411 | RBC8 |
| RalA and RalB inhibitor | |
| 3139 | RC 160 |
| sst analog | |
| 7066 | RCGD 423 |
| gp130 modulator; activates JAK/STAT signaling | |
| 6845 | RCM 1 |
| FOXM1 inhibitor | |
| 3214 | RETRA hydrochloride |
| Antitumor agent; suppresses mutant p53-bearing cancer cells | |
| 3672 | RF 9 |
| Selective NPFF1 and NPFF2 antagonist | |
| 4683 | RFRP 3 (human) |
| NPFF1 agonist; GnIH homolog | |
| 5761 | RG 102240 |
| Gene switch ligand for use in inducible gene expression systems | |
| 3295 | RG 108 |
| Non-nucleoside DNA methyltransferase inhibitor | |
| 3498 | RGDS peptide |
| Integrin binding sequence; inhibits integrin receptor function | |
| 6728 | RGFP 966 |
| Potent and selective HDAC3 inhibitor | |
| 1842 | RHC 80267 |
| Diacylglycerol lipase inhibitor | |
| 5311 | RHPS 4 methosulfate |
| Telomerase inhibitor | |
| 6168 | RI 1 |
| RAD51 recombinase inhibitor | |
| 6567 | RI-STAD 2 |
| AKAP disruptor; selectively binds PKA-RI with high affinity and blocks its interaction with AKAP; cell permeable | |
| 6892 | RIPGBM |
| RIPK2 modulator; pro-drug of cRIPGM; orally bioavailable and brain penetrant | |
| 2443 | RITA |
| MDM2-p53 interaction inhibitor | |
| 1053 | RJR 2403 oxalate |
| Selective α4β2 nAChR agonist | |
| 1271 | RJR 2429 dihydrochloride |
| nAChR agonist; displays selectivity for α4β2, α1βγδ and α3β4 subtypes | |
| 5061 | RKI 1447 dihydrochloride |
| Potent and selective ROCK inhibitor; antitumor | |
| 3393 | RLLFT-NH2 |
| Control peptide for TFLLR-NH2 (Cat. No. 1464) | |
| 5909 | RMM 46 |
| MSK/RSK family kinase inhibitor | |
| 4977 | RN 1 dihydrochloride |
| LSD1 inhibitor | |
| 3746 | RN 1734 |
| Selective TRPV4 antagonist | |
| 3745 | RN 1747 |
| Selective TRPV4 agonist | |
| 5678 | RN 9893 hydrochloride |
| Potent and selective TRPV4 antagonist | |
| 6833 | RO 5263397 hydrochloride |
| Potent TA1 receptor agonist | |
| 7375 | RO 8191 New |
| IFNα receptor 2 agonist | |
| 3052 | RO-3 |
| Selective P2X3 and P2X2/3 antagonist | |
| 4289 | RP 001 hydrochloride |
| Potent S1P1 agonist | |
| 1635 | RP 67580 |
| Potent and selective NK1 antagonist | |
| 5388 | RQ 00203078 |
| Potent and selective TRPM8 antagonist; orally active | |
| 5928 | RS 09 |
| TLR4 peptide agonist; acts as an adjuvant in vivo | |
| 1325 | RS 100329 hydrochloride |
| Potent, subtype-selective α1A antagonist | |
| 1050 | RS 102221 hydrochloride |
| Selective 5-HT2C antagonist | |
| 2089 | RS 102895 hydrochloride |
| CCR2b chemokine receptor antagonist | |
| 2993 | RS 127445 hydrochloride |
| High affinity and selective 5-HT2B antagonist | |
| 0985 | RS 17053 hydrochloride |
| α1A antagonist | |
| 0728 | RS 23597-190 hydrochloride |
| 5-HT4 antagonist | |
| 0991 | RS 39604 hydrochloride |
| 5-HT4 antagonist | |
| 2517 | RS 504393 |
| Highly selective CCR2 chemokine receptor antagonist | |
| 0987 | RS 79948 hydrochloride |
| Potent and selective α2 antagonist | |
| 6687 | 1R,3R-RSL3 New |
| Negative control for 1S,3R-RSL3 (Cat. No. 6118) | |
| 6118 | 1S,3R-RSL3 |
| Inhibits glutathione peroxidase (GPX4); induces ferroptosis | |
| 5138 | RSVA 405 |
| AMPK activator; also STAT3 inhibitor | |
| 0912 | RU 24969 hemisuccinate |
| 5-HT1A and 5-HT1B agonist | |
| 1672 | RU 28318, potassium salt |
| Potent, selective mineralocorticoid receptor antagonist | |
| 4886 | RU-SKI 43 hydrochloride |
| Hedgehog acyltransferase (Hhat) inhibitor; cell permeable | |
| 4227 | RWJ 50271 |
| Inhibitor of LFA-1/ICAM mediated cell adhesion | |
| 2614 | RWJ 56110 |
| Selective PAR1 antagonist | |
| 2999 | RWJ 67657 |
| Potent, selective p38α and p38β inhibitor | |
| 1324 | RX 821002 hydrochloride |
| Potent, selective α2D antagonist | |
| 1239 | Ac-RYYRIK-NH2 |
| High affinity NOP ligand | |
| 1387 | Ac-RYYRWK-NH2 |
| Potent, selective NOP partial agonist peptide | |
| 1810 | Raclopride |
| Potent and selective D2 and D3 antagonist | |
| 1589 | Radicicol |
| Hsp90 inhibitor. Antifungal antibiotic | |
| 2280 | Raloxifene hydrochloride |
| Selective estrogen receptor modulator (SERM) | |
| 5250 | Ramipril |
| Non-peptide, competitive angiotensin-converting enzyme (ACE) inhibitor | |
| 1967 | Ranitidine hydrochloride |
| Selective H2 antagonist | |
| 3118 | Ranolazine dihydrochloride |
| Antianginal, activates pyruvate dehydrogenase | |
| 1292 | Rapamycin |
| mTOR inhibitor; immunosuppressant | |
| 6760 | Raphin 1 |
| Inhibitor of the regulatory subunit PPP1R15B of protein phosphatase 1; orally bioavailable and brain penetrant | |
| 4308 | Rasagiline mesylate |
| Selective and irreversible MAO-B inhibitor | |
| 0891 | Rauwolscine hydrochloride |
| α2 antagonist | |
| 1982 | Reboxetine mesylate |
| Potent and selective noradrenalin uptake inhibitor; orally active | |
| 3284 | Rec 15/2615 dihydrochloride |
| Selective α1B antagonist | |
| 1622 | Remacemide hydrochloride |
| NMDA antagonist; blocks ion channel and allosteric modulatory site | |
| 7226 | Remdesivir |
| Viral RNA-dependent RNA polymerase (RdRP) inhibitor; broad spectrum antiviral nucelotide prodrug | |
| 5193 | Remodelin |
| N-acetyltransferase 10 (NAT10) inhibitor | |
| 0916 | Remoxipride hydrochloride |
| Selective D2-like antagonist | |
| 3742 | RepSox |
| Potent and selective inhibitor of TGF-βRI | |
| TB3742-RMU | RepSox |
| RepSox synthesized to Ancillary Material Grade | |
| 3805 | Repaglinide |
| Kir6 (KATP) channel blocker | |
| 6957 | Reparixin L-lysine salt |
| Potent CXCR1 and CXCR2 allosteric antagonist | |
| 2742 | Reserpine |
| Inhibitor of vesicular monoamine transport | |
| 4536 | Resiquimod |
| Toll-like receptor 7 (TLR7) agonist | |
| 1418 | Resveratrol |
| Cyclooxygenase inhibitor | |
| 6233 | Retigabine |
| KV7 channel activator | |
| 0695 | Retinoic acid |
| Endogenous retinoic acid receptor agonist | |
| 3722 | Reversan |
| Selective MRP1 and P-gp inhibitor | |
| 7406 | Rf470DL New |
| Blue rotor-fluorogenic fluorescent D-amino acid for labeling peptidoglycans in live bacteria | |
| 6867 | Rhein |
| FTO (mRNA N6-methyladenine demethylase) inhibitor; also inhibits ALKBH2 and ALKBH3 | |
| 5003 | Rhosin hydrochloride |
| Rho inhibitor | |
| 4501 | Ribavirin |
| Blocks eIF4E activity; antiviral guanosine analog | |
| 7050 | Ribociclib |
| Dual cdk4/cdk6 inhibitor; orally bioavailable | |
| 4121 | Rifampicin |
| Pregnane X receptor agonist; antibiotic | |
| 5359 | Rifaximin |
| Pregnane X receptor agonist; antibiotic | |
| 0790 | Rilmenidine hemifumarate |
| α2 agonist. Also I1 ligand | |
| 0768 | Riluzole hydrochloride |
| GABA uptake inhibitor; also inhibits glutamate release and blocks NaV channels | |
| 1497 | Rimcazole dihydrochloride |
| σ2 antagonist. Also DAT inhibitor | |
| 3504 | Risedronate |
| Farnesyl diphosphate (FPP) synthase inhibitor | |
| 2865 | Risperidone |
| 5-HT2A antagonist; also D2 antagonist; atypical antipsychotic | |
| 1955 | Ritanserin |
| Potent 5-HT2 antagonist | |
| 5856 | Ritonavir |
| HIV-1 and HIV-2 protease inhibitor | |
| 4440 | Rivastigmine tartrate |
| Dual AChE and BChE inhibitor | |
| 5136 | Rizatriptan benzoate |
| Potent 5-HT1B and 5-HT1D agonist | |
| 4348 | Ro 01-6128 |
| Positive allosteric modulator of mGlu1 receptors | |
| 2005 | Ro 04-5595 hydrochloride |
| GluN2B-selective NMDA antagonist | |
| 2911 | Ro 04-6790 |
| Potent and selective 5-HT6 antagonist | |
| 2188 | Ro 0437626 |
| Selective P2X1 antagonist | |
| 2272 | Ro 08-2750 |
| Inhibits NGF binding to p75NTR and TrkA | |
| 4268 | Ro 1138452 hydrochloride |
| Selective prostacyclin IP receptor antagonist | |
| 1997 | Ro 15-4513 |
| Benzodiazepine partial inverse agonist | |
| 0415 | Ro 20-1724 |
| PDE4 inhibitor | |
| 1594 | Ro 25-6981 maleate |
| GluN2B-selective NMDA antagonist | |
| 2002 | Ro 31-8220 mesylate |
| Protein kinase inhibitor | |
| 1587 | Ro 32-0432 hydrochloride |
| Potent, orally active PKC inhibitor | |
| 5968 | Ro 3280 |
| Potent and selective PLK1 inhibitor | |
| 4181 | Ro 3306 |
| Cdk1 inhibitor | |
| 5389 | Ro 48-8071 fumarate |
| 2,3-Oxidosqualene cyclase (OSC) inhibitor; blocks cholesterol synthesis | |
| 4694 | Ro 5-3335 |
| Core binding factor inhibitor; attenuates hematopoiesis | |
| 4391 | Ro 51 |
| Potent P2X3 and P2X2/3 antagonist | |
| 1854 | Ro 60-0175 fumarate |
| Potent, selective 5-HT2C agonist | |
| 3254 | Ro 61-8048 |
| Potent kynurenine 3-monooxygenase (KMO) inhibitor | |
| 2913 | Ro 64-5229 |
| Selective, non-competitive mGlu2 antagonist | |
| 4347 | Ro 67-4853 |
| Positive allosteric modulator of group I mGlu receptors | |
| 4346 | Ro 67-7476 |
| Positive allosteric modulator of mGlu1 receptors | |
| 5913 | Ro 6842262 |
| Potent LPA1 antagonist | |
| 2408 | Ro 90-7501 |
| Inhibitor of Aβ42 fibril formation | |
| 6641 | Roflumilast |
| Potent and selective PDE4 inhibitor | |
| 0905 | Rolipram |
| PDE4 inhibitor | |
| 1349 | (R)-(-)-Rolipram |
| PDE4 inhibitor. More active enantiomer of rolipram (Cat. No. 0905) | |
| 3680 | Ropinirole |
| Selective D2-like agonist | |
| 1332 | Roscovitine |
| 5168 | Rose Bengal |
| Stains exposed epithelium in eye. Also VGlut and VMAT inhibitor | |
| 5325 | Rosiglitazone |
| Potent and selective PPARγ agonist; antidiabetic agent | |
| 5315 | Rostafuroxin |
| Na+/K+ ATPase modulator; antihypertensive agent | |
| 6343 | Rosuvastatin calcium |
| Potent HMG-CoA reductase inhibitor | |
| 3616 | Rotenone |
| Inhibits complex I of the mitochondrial electron transport chain | |
| 3896 | Rotigotine hydrochloride |
| D2 and D3 agonist | |
| 1610 | Rottlerin |
| Reported PKCδ inhibitor | |
| 7486 | Roxadustat New |
| HIF-PH inhibitor; erythropoietic | |
| 1559 | Roxindole hydrochloride |
| Dopamine D2 autoreceptor agonist. Also has affinity for D3, D4, 5-HT1A receptors and the 5-HT transporter | |
| 5524 | Rp-8-pCPT-cGMPS sodium |
| PKG inhibitor | |
| 3400 | RuBi-GABA |
| Caged GABA; excitable at visible wavelengths | |
| 3574 | RuBi-Glutamate |
| Caged glutamate; excited by visible wavelengths | |
| 3855 | RuBi-Nicotine |
| Caged nicotine; rapidly excitable by visible light | |
| 4709 | RuBi GABA trimethylphosphine |
| Caged GABA; inhibits neural activity | |
| 6230 | Rucaparib camsylate |
| PARP inhibitor | |
| 3828 | Rufinamide |
| Prolongs inactivation of sodium channels; anticonvulsant | |
| 6414 | Rupintrivir |
| Potent and selective irreversible human rhinovirus 3Cpro inhibitor | |
| 1439 | Ruthenium Red |
| Non-selective CaV2.1 and 2.2 blocker; also blocks TRPV channels | |
| 7064 | Ruxolitinib |
| Potent and selective JAK1/JAK2 inhibitor; orally bioavailable | |
| 7048 | Ruxolitinib phosphate |
| Phosphate salt of Ruxolitinib (Cat. No. 7064); potent and selective JAK1/JAK2 inhibitor | |
| 1329 | Ryanodine |
| Ca2+ release inhibitor | |
| 2609 | Ryuvidine |
| SETD8 inhibitor; also CDK4 inhibitor |
Tocris Products by Catalog Number
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