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Displaying Products by Catalog Number (1600 - 1699)

Cat. No. Product Name / Activity
1600 pep2-AVKI
Peptide inhibitor of GluA2 subunit binding to PICK1
1601 Pep1-TGL
GluA1 subunit C-terminus peptide analog
1602 Pep1-AGL
GluA1 subunit C-terminus peptide analog; also analog of Pep1-TGL (Cat. No. 1601)
1603 NKH 477
Water-soluble adenylyl cyclase activator
1604 Urocortin (human)
Endogenous CRF agonist
1605 Urocortin (rat)
Endogenous CRF agonist
1606 Astressin
Potent CRF antagonist
1607 CRF (6-33)
CRF-binding protein inhibitor
1608 Stressin I
CRF1 agonist
1609 Sauvagine
CRF agonist
1610 Rottlerin
Reported PKCδ inhibitor
1611 Lamotrigine
Inhibits glutamate release. Anticonvulsant
1612 SB 269970 hydrochloride
Potent and selective 5-HT7 antagonist; brain penetrant
1614 SB 431542
Potent, selective inhibitor of TGF-βRI, ALK4 and ALK7
1615 SB 366791
Potent, selective, competitive TRPV1 antagonist
1616 SB 216763
Potent, selective GSK-3 inhibitor
1617 SB 415286
Potent, selective GSK-3 inhibitor
1618 Peptide YY (3-36)
Selective NPY Y2 receptor agonist
1620 Alprostadil
Prostaglandin. Vasodilator and antiplatelet agent in vivo
1621 Streptozocin
DNA alkylator; antitumor and induces diabetes
1622 Remacemide hydrochloride
NMDA antagonist; blocks ion channel and allosteric modulatory site
1623 Cyclopamine
Inhibitor of Hedgehog (Hh) signaling
1624 2-Methylthioadenosine diphosphate trisodium salt
Potent agonist at P2Y1, P2Y12 and P2Y13
1625 DFB
Positive allosteric modulator of mGlu5 receptors
1626 Calphostin C
Potent, selective and photo-dependent PKC inhibitor
1629 Herbimycin A
Src family kinase inhibitor. Also Hsp90 inhibitor
1632 MEN 10376
Potent, selective NK2 antagonist
1634 Y-29794 oxalate
Prolyl endopeptidase inhibitor
1635 RP 67580
Potent and selective NK1 antagonist
1636 IEM 1460
Open-channel blocker of AMPA currents; selective for non-GluA2-containing receptors
1637 Argatroban
Potent thrombin inhibitor
1638 U 18666A
Inhibitor of Hedgehog (Hh) signaling. Also inhibits cholesterol synthesis
1639 AY 9944 dihydrochloride
Inhibitor of Hedgehog (Hh) signaling. Inhibits Δ7-dehydrocholesterol reductase
1640 [bAla8]-Neurokinin A(4-10)
NK2 agonist
1641 OLDA
Potent, selective endogenous TRPV1 agonist
1642 Urotensin II (human)
Endogenous vasoactive agonist for the UT receptor
1643 D-64131
Tubulin polymerization inhibitor. Antitumor in vivo
1644 Mesulergine hydrochloride
5-HT2A and 5-HT2C antagonist; also D2-like partial agonist
1645 8-CPT-2Me-cAMP, sodium salt
Selective Epac activator
1646 Lonidamine
Mitochondrial hexokinase inhibitor
1650 BAM 22P
MRGPRX1 agonist; also opioid receptor agonist
1652 Apamin
KCa2 channel blocker (small conductance)
1655 O-2050
Putative CB1 antagonist; displays mixed activity at CB receptors
1657 Ginkgolide B
PAF receptor antagonist
1658 GR 125487 sulfamate
Potent and selective 5-HT4 antagonist; active in vivo
1659 Fenoldopam hydrochloride
Selective D1-like partial agonist
1661 SB 206553 hydrochloride
Potent and selective 5-HT2B and 5-HT2C antagonist; orally active
1662 SKF 77434 hydrobromide
Selective D1-like partial agonist
1663 BW 373U86
Potent, selective non-peptide δ agonist
1664 GW 1929 hydrochloride
Selective PPARγ agonist. Orally active
1667 GR 94800
Potent, selective NK2 antagonist
1668 GR 64349
Potent, selective NK2 agonist
1669 GR 73632
Potent and selective NK1 agonist
1670 GR 82334
NK1 antagonist
1671 PD 102807
Selective M4 antagonist
1672 RU 28318, potassium salt
Potent, selective mineralocorticoid receptor antagonist
1673 Cl-HIBO
GluA1 and GluA2 selective AMPA agonist
1674 LE 300
Potent and selective D1 antagonist
1675 YM 90709
Interleukin-5 receptor antagonist
1676 T 0156 hydrochloride
Highly potent, selective PDE5 inhibitor
1677 GW 7647
Highly selective, potent PPARα agonist. Orally active
1682 PIT
P2Y ligand; displays mixed antagonism/potentiation
1683 K 252a
Protein kinase inhibitor
1688 Autocamtide-2-related inhibitory peptide
Selective CaM kinase II inhibitor
1690 SCH 28080
H+,K+-ATPase inhibitor
1691 NECA
High affinity adenosine agonist
1692 Cilostazol
PDE3A inhibitor. Also adenosine uptake inhibitor
1693 Enoximone
PDE3 inhibitor
1694 Ibudilast
PDE inhibitor (non-selective)
1695 Cisapride
5-HT4 agonist; stimulates intestinal ACh release
1697 Noscapine hydrochloride
Tubulin inhibitor; induces apoptosis
1699 CGS 15943
Potent adenosine receptor antagonist

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