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Displaying Products by Catalog Number (4200 - 4299)

Cat. No. Product Name / Activity
4200 C 646
Selective p300/CBP inhibitor
4202 Adenine
Adenine receptor agonist
4204 BTZO 1
MIF binder
4205 MDA 19
CB2 agonist
4206 Valdecoxib
Selective and potent COX-2 inhibitor
4207 SB 277011A dihydrochloride
Selective D3 antagonist
4208 MS 245 oxalate
High affinity 5-HT6 antagonist
4210 Ascomycin
Calcineurin phosphatase inhibitor; analog of FK 506 (Cat. No. 3631)
4212 PIR 3.5
Negative control of IPA 3 (Cat. No. 3622)
4213 SB 297006
Potent and selective CCR3 antagonist
4214 Prostaglandin F2α
Naturally-occurring prostanoid; potent vasoconstrictor
4215 4E1RCat
Inhibits eIF4F subunit interaction; inhibits protein translation
4216 Valsartan
High affinity, selective AT1 antagonist
4218 Travaprost
Potent and selective FP prostaglandin receptor agonist
4219 Banoxantrone dihydrochloride
Prodrug topoisomerase II inhibitor
4220 XCC
Adenosine receptor antagonist
4221 TCS 21311
Potent JAK3 inhibitor. Also inhibits GSK-3β and PKC
4222 Dynole 34-2
Dynamin I inhibitor
4224 MitMAB
Dynamin inhibitor
4225 OctMAB
Dynamin inhibitor
4227 RWJ 50271
Inhibitor of LFA-1/ICAM mediated cell adhesion
4228 A 286982
Potent inhibitor of the LFA-1/ICAM-1 interaction
4230 NPEC-caged-D-AP5
Caged D-AP5 (Cat.No. 0106)
4231 Nateglinide
Kir6 (KATP) blocker; displays high affinity for SUR1/Kir6.2 channels
4232 A 839977
Potent P2X7 antagonist
4233 TQS
Positive allosteric modulator of α7 nAChRs
4234 4BP-TQS
α7 nAChR agonist; acts at an allosteric site
4236 CP 945598 hydrochloride
CB1 antagonist
4237 PD 184352
Selective MEK inhibitor
4238 PF 184
Potent and selective IKKβ inhibitor
4239 PF 04217903 mesylate
Highly selective MET inhibitor
4240 SCH 529074
Restores mutant p53 activity
4241 Olopatadine hydrochloride
H1 antagonist; ocular antiallergic agent
4242 GW 803430
MCH1 antagonist
4243 Kisspeptin 10 (rat)
Endogenous ligand for kisspeptin receptor
4244 TCS 3035
GPR35 agonist
4245 Meclizine dihydrochloride
Human pregnane X receptor agonist; H1 antagonist
4246 CID 2858522
Selectively inhibits PKC-induced NF-κB activation
4247 Torin 1
Potent and selective mTOR inhibitor
4248 Torin 2
Potent and selective mTOR inhibitor
4249 A 887826
Potent voltage-dependent NaV1.8 channel blocker
4250 Mitoxantrone dihydrochloride
Topoisomerase II inhibitor; immunosuppressive and antineoplastic agent
4252 PF 4981517
Selective CYP3A4 inhibitor
4253 TMPyP4 tosylate
Inhibitor of human telomerase
4254 TAK 715
Potent p38 MAPK inhibitor; anti-inflammatory
4255 TC-O 9311
Potent and selective GPR139 agonist
4256 Tiagabine hydrochloride
Selective GAT-1 inhibitor; anticonvulsant
4257 PP 242
Dual mTORC1/mTORC2 inhibitor
4259 TCN 238
Positive allosteric modulator of mGlu4 receptors
4260 MRS 2957 triethylammonium salt
Potent and selective P2Y6 agonist
4261 MRS 4062 triethylammonium salt
Selective P2Y4 receptor agonist
4265 AS 1842856
Potent and selective Foxo1 inhibitor; orally bioavailable
4266 ML 141
Selective Cdc42 Rho family inhibitor
4268 Ro 1138452 hydrochloride
Selective prostacyclin IP receptor antagonist
4270 TC-H 106
Class I histone deacetylase inhibitor
4272 [D-Trp8]-γ-MSH
Selective MC3 receptor agonist
4273 LRRK2-IN-1
Potent and selective LRRK2 inhibitor
4274 AP 24534
Potent multi-kinase and pan-Bcr-Abl inhibitor
4276 ERB 041
Potent ERβ agonist
4277 PF 477736
Selective Chk1 inhibitor
4278 PF 431396
Dual FAK/PYK2 inhibitor
4279 PF 3644022
Potent MK2 inhibitor
4281 PF 4800567 hydrochloride
Selective casein kinase 1ε inhibitor
4282 WYE 687 dihydrochloride
Potent and selective mTOR inhibitor
4283 Begacestat
γ-secretase inhibitor; lowers Aβ40 and Aβ42 levels
4285 HBX 41108
Selective USP7 inhibitor
4286 UA 62784
Inhibits microtubule polymerization
4287 Poly(I:C)
TLR3 agonist
4288 ISO 1
Macrophage migration inhibitory factor (MIF) inhibitor
4289 RP 001 hydrochloride
Potent S1P1 agonist
4291 CCT 137690
Potent pan-Aurora kinase inhibitor
4293 CID 2745687
GPR35 antagonist
4295 VU 0357017 hydrochloride
Positive allosteric modulator of M1 receptors
4297 SMER 28
Positive regulator of autophagy
4298 Pamoic acid disodium salt
GPR35 agonist
4299 iCRT 14
Inhibits β-catenin-responsive transcription (CRT)

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