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Displaying Products Alphabetically by Name (B)

Cat. No. Product Name / Activity
6764 B 973B
Positive allosteric modulator of α7 nAChRs; analgesic
6009 B I09
IRE1 endonuclease inhibitor; cell permeable
1802 2B-(SP)
Selective GSK-3 phosphopeptide substrate
2759 B-HT 920
D2 agonist; also α2-adrenoceptor agonist and 5-HT3 antagonist
2758 B-HT 933 dihydrochloride
Selective α2 agonist
6392 B02
RAD51 recombinase inhibitor
2855 B2
Promotes inclusion formation in Huntington's and Parkinson's diseases
5600 BA 1
Potent bombesin agonist
1326 BADGE
PPARγ antagonist
3606 BAG 956
Dual PI 3-kinase and PDPK1 (PDK1) inhibitor
1763 BAM (8-22)
Potent MRGPRX1 agonist
5737 BAM 15
Mitochondrial protonophore uncoupler
1650 BAM 22P
MRGPRX1 agonist; also opioid receptor agonist
4810 BAM 7
Selective Bax activator; induces Bax-mediated apoptosis
3661 BAN ORL 24
Potent and selective NOP antagonist
2786 BAPTA
Selective calcium chelator
2787 BAPTA AM
Cell-permeable Ca2+ chelator
6857 BAY 293
Potent KRas/SOS1 interaction inhibitor
6906 BAY 293 Negative Control
Negative control for BAY 293 (Cat. No. 6857)
5970 BAY 299
Potent and selective BRD1 and TAF1 inhibitor
4430 BAY 41-2272
Soluble guanylyl cyclase (sGC) activator
5708 BAY 41-8543
Guanylyl cyclase (sGC) stimulator
6052 BAY 58-2667 hydrochloride
Potent soluble guanylyl cyclase (sGC) activator
5991 BAY 598
Potent and selective SMYD2 inhibitor
4472 BAY 60-6583
Potent A2B agonist; cardioprotective
6561 BAY 6035
Potent and selective SMYD3 inhibitor
6389 BAY 677
Inactive control for BAY 678 (Cat.No.5706)
5706 BAY 678
Potent and selective cell-permeable human neutrophil elastase (HNE) inhibitor
6817 BAY 8002
Potent dual MCT1/2 inhibitor; orally bioavailable
6579 BAY 826
Potent Tie2 inhibitor
6980 BAY 87-2243
Mitochondrial complex I inhibitor
6199 BAY 876
Potent and selective GLUT1 inhibitor
3541 BAY-X 1005
Orally active 5-lipoxygenase activating protein (FLAP) inhibitor
2732 BAY-u 3405
Dual TP/DP2 (CRTH2) receptor antagonist
5266 BAZ2-ICR
Selective BAZ2 inhibitor
4372 BC 11 hydrobromide
Selective urokinase (uPA) inhibitor
4496 BC 11-38
Selective PDE11 inhibitor
6791 BC-LI-0186
Leucyl-tRNA synthase (TRS)/Ras-related GTP-binding protein D (RagD) interaction inhibitor
5027 BCH
LAT1 inhibitor
1048 1-BCP
Modulates AMPA-mediated responses
3875 BCTC
TRPV1 antagonist
0511 BD 1008 dihydrobromide
Potent, selective σ ligand
0956 BD 1047 dihydrobromide
σ1 selective antagonist
0883 BD 1063 dihydrochloride
Selective σ1 ligand, putative antagonist
3579 5-BDBD
Potent and selective P2X4 antagonist
2837 BDNF (human)
Activates TrkB and p75 receptors
5184 BDS I
Potent and reversible Kv3.4 potassium channel blocker; neuroprotective
5468 BDY 630-X, SE
Red BDY (BODIPY® or boron-dipyrromethene) fluorescent dye for the labeling of amines; supplied as NHS ester
5469 BDY 650-X, SE
Far-red BDY (BODIPY® or boron-dipyrromethene) fluorescent dye for the labeling of amines; supplied as NHS ester
5465 BDY FL, SE
Green BDY (BODIPY® or boron-dipyrromethene) fluorescent dye for the labeling of amines; supplied as NHS ester
5620 BDY FL-X, SE
Green BDY (BODIPY® or boron-dipyrromethene) fluorescent dye for the labeling of amines; supplied as NHS ester
5466 BDY TMR-X, SE
Yellow BDY (BODIPY® or boron-dipyrromethene) fluorescent dye for the labeling of amines; supplied as NHS ester
5467 BDY TR-X, SE
Orange/red BDY (BODIPY® or boron-dipyrromethene) fluorescent dye for the labeling of amines; supplied as NHS ester
4778 BETP
Positive allosteric modulator of GLP-1 receptors
3743 BF 2649 hydrochloride
Potent and selective H3 inverse agonist
6246 BF 738735
Potent and selective PI 4-kinase IIIβ inhibitor; broad spectrum enterovirus replication inhibitor
0348 2-BFI hydrochloride
Potent, selective I2 ligand. Putative agonist
5327 BGC 20-1531 hydrochloride
High affinity and selective EP4 antagonist
3326 BGC 20-761
High affinity 5-HT6 antagonist
6703 BGP 15
PARP inhibitor; cytoprotectant
3313 rac BHFF
Potent and selective postitive allosteric modulator of GABAB receptors
6116 BHPI
ERα antagonist; also activates unfolded protein response; active in vivo
1236 BHQ
Inhibitor of SERCA ATPase
6518 BI 01383298
Potent and selective SLC13A5 (Na+/citrate cotransporter) inhibitor
4641 BI 6015
Hepatocyte nuclear factor 4α (HNF4α) antagonist
5300 BI 605906
Selective IKKβ inhibitor
3314 BI 78D3
Selective, competitive JNK inhibitor
6665 BI 9321
Nuclear receptor-binding SET domain (NSD) 3 antagonist; selectively binds PWWP1 domain
5590 BI 9564
Potent and selective BRD9 and BRD7 inhibitor; orally active
4561 BIBN 4096
Potent and selective CGRP antagonist
2412 BIBO 3304 trifluoroacetate
Highly selective NPY Y1 receptor antagonist
2707 BIBP 3226 trifluoroacetate
Mixed NPY Y1 and NPFF receptor antagonist
2981 BIBR 1532
Selective telomerase inhibitor
2417 BIBU 1361 dihydrochloride
Selective inhibitor of EGFR-kinase
2416 BIBX 1382 dihydrochloride
Highly selective EGFR-kinase inhibitor
4608 BIIB 021
Selective Hsp90 inhibitor
1700 BIIE 0246
Potent, selective non-peptide NPY Y2 receptor antagonist
2716 BIM 187
Bombesin/GRP receptor agonist
2717 BIM 189
Bombesin antagonist
3237 BIM 23042
Selective neuromedin B receptor antagonist (NMB-R, BB1)
1844 BIM 23056
sst ligand
4374 BIMU 8
Potent 5-HT4 agonist
4048 BINA
Selective positive allosteric modulator of mGlu2 receptors
3194 BIO
Potent GSK-3 inhibitor; also inhibits cdks
3910 BIO 1211
Selective α4β1 (VLA-4) inhibitor
5051 BIO 5192
Highly potent and selective inhibitor of integrin α4β1 (VLA-4)
3874 BIO-acetoxime
Selective GSK-3α/β inhibitor
5989 BIRB 796
High affinity and selective p38 kinase inhibitor
4776 BIRT 377
Potent negative allosteric modulator of LFA-1
5216 BIS-TRIS
Commonly used buffering agent
5375 BIX
BiP (Hsp70-5) ER chaperone inducer
3364 BIX 01294
GLP and G9a inhibitor
4842 BIX 02189
Selective MEK5 and ERK5 inhibitor
5512 BIX NHE1 inhibitor
Potent and selective NHE1 inhibitor
3797 BL 1249
K2P2.1 (TREK-1) and K2P10.1 (TREK-2) activator
2538 L-BMAA hydrochloride
Neurotoxic amino acid
5417 BMH 21
RNA polymerase 1 inhibitor; also p53 pathway activator
5488 BML 111
FPR2 (lipoxin A4 receptor) agonist
1441 BMS 182874 hydrochloride
Highly selective, orally active non-peptide ETA antagonist
2665 BMS 191011
Potent BKCa (KCa1.1) channel opener
3242 BMS 193885
Potent, competitive NPY Y1 receptor antagonist
3660 BMS 195614
Selective RARα antagonist
5654 BMS 265246
Cdk inhibitor; potently inhibits cdk1 and cdk2
2870 BMS 299897
Potent γ-secretase inhibitor
4609 BMS 303141
ATP citrate lyase inhibitor; orally bioavailable
5258 BMS 309403
Potent and selective FABP4 inhibitor
4806 BMS 345541
Selective allosteric inhibitor of IKK; anti-inflammatory
3409 BMS 453
Synthetic retinoid and RARβ agonist; also RARα and RARγ antagonist
4053 BMS 470539 dihydrochloride
Potent, selective MC1 receptor agonist
3509 BMS 493
Pan-RAR inverse agonist
5009 BMS 509744
Potent and selective ITK inhibitor
4774 BMS 536924
Dual IR/IGF1R inhibitor
5274 BMS 564929
Highly potent and muscle-selective androgen receptor (AR) agonist
5492 BMS 566419
Inosine monophosphatase dehydrogenase (IMPDH) inhibitor
5022 BMS 599626 dihydrochloride
Potent, selective EGFR and ErbB2 inhibitor
6069 BMS 605541
Potent VEGFR-2 inhibitor
4970 BMS 688521
Potent inhibitor of the LFA-1/ICAM interaction
3505 BMS 753
RARα-selective agonist
5762 BMS 795311
Potent cholesteryl ester transfer protein (CETP) inhibitor
3410 BMS 961
Selective RARγ agonist
6974 BMS 986094
Inhibitor of HCV RNA-dependent RNA polymerase NS5b; potent hepatitis C virus (HCV) replication inhibitor
5983 BMS 986187
Potent positive allosteric modulator of δ receptors
3129 BMS CCR2 22
High affinity, potent CCR2 antagonist
5123 BMX-IN-1
Potent and irreversible BMX inhibitor
1440 BMY 14802 hydrochloride
Sigma antagonist. Antipsychotic agent
1442 BMY 45778
Non-prostanoid prostacyclin IP receptor partial agonist
1006 BMY 7378 dihydrochloride
Selective α1D antagonist
0899 BNTX maleate
Standard δ1 selective antagonist
6047 BOP
Dual α9β1/α4β1 integrin inhibitor; preferentially mobilizes HSCs
0556 BP 554 maleate
Selective 5-HT1A agonist
5301 BPTES
Selective allosteric glutaminase (GLS1) inhibitor
6078 BPTU
P2Y1 allosteric antagonist
1500 BQ 788 sodium salt
Selective ETB antagonist
1188 BQ-123
Selective ETA antagonist
1189 BQ-3020
Selective ETB agonist
6872 BQCA
Positive allosteric modulator of M1 receptors
5312 BRACO 19 trihydrochloride
Telomerase inhibitor
6010 BRD 4354
HDAC5 and HDAC9 inhibitor
6282 BRD 4770
G9a inhibitor and S-adenosyl methionine mimetic; cell permeable
6438 BRD 6989
Cdk8 inhibitor; enhances IL-10 production
5336 BRD 7116
Inhibitor of leukemia stem cell activity
4037 BRD 7389
Ribosomal S6 kinase inhibitor
6284 BRD 73954
Dual histone deacetylase (HDAC) 6/8 inhibitor
5230 BRD 7552
PDX1 transcription factor inducer; increases insulin expression
6040 BRD 9757
Potent and selective HDAC6 inhibitor
1207 BRL 15572 hydrochloride
Selective h5-HT1D antagonist
0948 BRL 37344, sodium salt
β3 agonist
1133 BRL 44408 maleate
Selective α2A antagonist
2237 BRL 50481
Selective PDE7 inhibitor
0699 BRL 52537 hydrochloride
Potent and selective κ agonist
1129 BRL 54443
Potent 5-ht1E and 5-HT1F agonist
5608 BS 181 dihydrochloride
Selective cdk7 inhibitor
5817 BSI 201
PARP-1 inhibitor
6921 BSJ-03-123
Selective Cdk6 degrader
6938 BSJ-03-204
Selective Cdk4/6 degrader
6937 BSJ-04-132
Selective Cdk4 degrader
6922 BSJ-Bump
Negative control for BSJ-03-123 (Cat. No. 6921)
5399 BTB1
Selective and ATP-competitive Kif18A inhibitor
6940 BTD
Selective TRPC5 activator
1870 BTS
Selective inhibitor of skeletal muscle myosin II ATPase activity
2322 BTS 54-505 hydrochloride
Potent 5-HT and NA reuptake inhibitor (SNRI); active metabolite of sibutramine (Cat. No. 2290)
4724 BTT 3033
Selective inhibitor of integrin α2β1
4204 BTZO 1
MIF binder
0725 BU 224 hydrochloride
Potent, selective I2 ligand. Putative antagonist
1091 BU 226 hydrochloride
Potent, highly selective I2 ligand
0726 BU 239 hydrochloride
Potent, highly selective I2 ligand
2176 BVT 948
Non-competitive protein tyrosine phosphatase inhibitor
1663 BW 373U86
Potent, selective non-peptide δ agonist
1059 BW 723C86 hydrochloride
5-HT2B agonist
1304 BW-B 70C
5-Lipoxygenase inhibitor
5545 BX 430
Selective P2X4 allosteric antagonist
3496 BX 471
Potent, selective CCR1 antagonist
2769 BX 513 hydrochloride
Selective CCR1 antagonist
4318 BX 795
PDPK1 (PDK1) inhibitor
2866 BYK 191023 dihydrochloride
Potent and selective inhibitor of iNOS
3734 BYK 204165
Selective PARP-1 inhibitor
3735 BYK 49187
PARP-1 and PARP-2 inhibitor
0796 (R)-Baclofen
Selective GABAB agonist; active enantiomer of (RS)-Baclofen (Cat. No. 0417)
0417 (RS)-Baclofen
Selective GABAB agonist
1334 Bafilomycin A1
H+-ATPase (vacuolar) inhibitor
1761 Baicalein
5- and 12-Lipoxygenase inhibitor
5585 Balicatib
Potent and selective cathepsin K inhibitor
4219 Banoxantrone dihydrochloride
Prodrug topoisomerase II inhibitor
2961 Batimastat
Potent, broad spectrum MMP inhibitor
2160 Bax channel blocker
Allosteric inhibitor of Bax channel activation
1785 Bax inhibitor peptide V5
Inhibitor of Bax-mediated apoptosis
1743 Bay 11-7085
Irreversible inhibitor of TNF-α-induced IκBα phosphorylation
1744 Bay 11-7821
E2 ubiquitin (Ub) conjugating enzymes inhibitor
2501 Bay 36-7620
mGlu1 inverse agonist
2711 Bay 55-9837
Potent and selective VPAC2 agonist
2500 Bay 59-3074
CB1/CB2 receptor partial agonist
1544 (±)-Bay K 8644
CaV1.x activator
1545 (R)-(+)-Bay K 8644
CaV1.x blocker; (R)-(+)-enantiomer of (±)-Bay K 8644; also TMEM176B inhibitor
1546 (S)-(-)-Bay K 8644
CaV1.x activator; (S)-(-)-enantiomer of (±)-Bay K 8644
5263 Bazedoxifene acetate
Potent and selective estrogen receptor modulator (SERM)
5929 BeKm 1
Potent and selective KV11.1 (hERG) channel blocker
4283 Begacestat
γ-secretase inhibitor; lowers Aβ40 and Aβ42 levels
2578 Benazepril hydrochloride
Angiotensin-converting enzyme (ACE) inhibitor
3681 Bendamustine hydrochloride
Cytostatic agent; exhibits DNA alkylating and purine analog properties
5273 Bengamide B
Potent inhibitor of NF-κB activation
3934 Benidipine hydrochloride
Non-selective Cav blocker; also mineralocorticoid receptor antagonist
3380 Benzamil
NCX inhibitor, Deg/ENaC channel blocker; amiloride (Cat. No. 0890) derivative
5420 Benzbromarone
TMEM16A/B calcium-activated chloride channel (CaCC) blocker
0424 Benzoquinonium dibromide
nAChR antagonist
0754 N-Benzylnaltrindole hydrochloride
Selective non-peptide δ2 antagonist
4117 Bepridil hydrochloride
Non-selective Ca2+ channel blocker; also NCX inhibitor
4180 Beraprost sodium
Potent prostacyclin IP receptor agonist
1956 Bestatin
Aminopeptidase inhibitor
0906 Betaxolol hydrochloride
Selective β1 antagonist
3906 Betulinic acid
Antitumor and anti-HIV agent; activates NF-κB. Also TGR5 agonist
5819 Bexarotene
Potent and selective RXR agonist
3389 Bicalutamide
Non-steroidal androgen receptor antagonist
4357 Bicifadine hydrochloride
Noradrenalin, 5-HT and dopamine re-uptake inhibitor
5881 Bicine
General purpose buffer
2503 (-)-Bicuculline methiodide
GABAA antagonist; more water soluble version of (+)-bicuculline (Cat. No. 0130)
0109 (-)-Bicuculline methobromide
GABAA antagonist; more water soluble version of (+)-bicuculline (Cat. No. 0130)
0131 (-)-Bicuculline methochloride
GABAA antagonist; more water soluble version of (+)-bicuculline (Cat. No. 0130)
0130 (+)-Bicuculline
Potent GABAA antagonist
0767 Bifemelane hydrochloride
Non-selective MAO inhibitor
6304 BigLEN (mouse)
GPR171 agonist
6306 BigLEN (rat)
Potent GPR171 agonist
0347 nor-Binaltorphimine dihydrochloride
Selective κ antagonist
3349 Biocytin
Versatile marker for neuroanatomical investigations
3526 BIM, Biotinylated
Bim peptide fragment
6571 Biotin-11-dUTP
Biotin-labeled dUTP
6572 Biotin-LC-NAD+
Biotinylated analog of β-NAD+; commonly used reagent in LSD1 and PARP1 assays
6573 Biotin-NAD+
Biotinylated-NAD+; substrate for ADP-ribosylation
6241 Biotinyl Tyramide
Reagent widely used for signal amplification in IHC and ISH
5372 Bioymifi
DR5 (TRAIL receptor) agonist; induces apoptosis
2853 Biperiden hydrochloride
Muscarinic receptor antagonist; some selectivity for M1
5348 6,8-Bis(benzylthio)octanoic acid
PDH and KGDH inhibitor
0918 3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride
Potent dopamine uptake inhibitor
4128 Bisindolylmaleimide II
Potent PKC inhibitor; also potent nAChR antagonist
0914 (±)-Bisoprolol hemifumarate
β1 antagonist
5502 Blasticidin S HCl
Antibiotic; selection reagent for bis, bsr and BSD transformed cells
1853 (R)-(+)-Blebbistatin
Selective inhibitor of myosin II ATPase activity. Inactive enantiomer of (±)-blebbistatin (Cat. No. 1760)
1852 (S)-(-)-Blebbistatin
Selective inhibitor of myosin II ATPase activity. Active enantiomer of (±)-blebbistatin (Cat. No. 1760)
1760 (±)-Blebbistatin
Selective inhibitor of myosin II ATPase activity
5255 6-Bnz-cAMP sodium salt
Cell permeable cAMP analog
3730 Boc-MLF
FPR1 antagonist
1149 Bombesin
Involved in gastrointestinal tract function
3422 [D-Phe12,Leu14]-Bombesin
Bombesin receptor antagonist
2371 Bombinakinin M
Potent bradykinin agonist
2370 Bombinakinin-GAP
Bioactive, bradykinin-related peptide
4706 Borrelidin
Antiangiogenic; inhibits threonyl-tRNA synthetase
6232 Bosentan
High affinity dual ETA and ETB receptor antagonist;orally bioavailable
4361 Bosutinib
Dual Src-Abl inhibitor; antiproliferative
5217 Bovine Serum Albumin
Widely used blocking agent for ELISA and blotting
3004 Bradykinin
Endogenous agonist at bradykinin receptors (B2 > B1)
3230 Sar-[D-Phe8]-des-Arg9-Bradykinin
Potent and selective B1 agonist
3225 Lys-[Des-Arg9]Bradykinin
Selective B1 agonist
3229 [Phe8Ψ(CH-NH)-Arg9]-Bradykinin
Selective B2 agonist
3522 Brain natriuretic peptide (1-32) (human)
Endogenous peptide agonist at ANP receptor A (NPR1)
1231 Brefeldin A
Disrupts protein translocation to Golgi
6196 Brequinar sodium
Potent and selective DHODH inhibitor
3568 Bretazenil
Benzodiazepine partial agonist
1140 8-Bromo-cAMP, sodium salt
Cell-permeable cAMP analog
1089 8-Bromo-cGMP, sodium salt
cGMP analog; activates PKG
0427 Bromocriptine mesylate
D2-like agonist (D2>D3>D4)
3549 3-Bromocytisine
Potent α4β4, α4β2 and α7 nAChR agonist
5015 5-BrdU
Synthetic thymidine analog; used for cell proliferation assays
0735 3-Bromo-7-nitroindazole
Selective nNOS inhibitor
5218 Bromophenol Blue
Dye used in gel loading buffers
4758 Bromosporine
Broad spectrum bromodomain inhibitor
4316 Bropirimine
Immunomodulatory and antitumor compound
2383 Bryostatin 1
Protein kinase C activator
5238 Bryostatin 3
Potent protein kinase C activator
2671 Budesonide
Synthetic glucocorticoid; anti-inflammatory and chemopreventive
3108 Bumetanide
Na+/2Cl-/K+ (NKCC) symporter inhibitor
2133 α-Bungarotoxin
Selective α7 nAChR antagonist
2808 Buprenorphine hydrochloride
NOP agonist; also displays mixed action δ, κ and μ receptors
2831 Bupropion hydrochloride
Non-selective inhibitor of dopamine and noradrenalin transporters
0962 Buspirone hydrochloride
5-HT1A partial agonist
1323 Butabindide oxalate
High affinity CCK-inactivating serine protease inhibitor
5791 Bz 423
ATP synthase inhibitor; proapoptotic
3312 BzATP triethylammonium salt
Photoaffinity label for ATPase; also P2X7 agonist and P2X1/P2Y1 partial agonist
6786 BzF
Photoreactive unnatural amino acid; photo-crosslinker

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