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Displaying Products Alphabetically by Name (B)

Cat. No. Product Name / Activity
6764 B 973B
Positive allosteric modulator of α7 nAChRs; analgesic
6009 B I09
IRE1 endonuclease inhibitor; cell permeable
2758 B-HT 933 dihydrochloride
Selective α2 agonist
6392 B02
RAD51 recombinase inhibitor
3606 BAG 956
Dual PI 3-kinase and PDPK1 (PDK1) inhibitor
1763 BAM (8-22)
Potent MRGPRX1 agonist
5737 BAM 15
Mitochondrial protonophore uncoupler
2786 BAPTA
Selective calcium chelator
Cell-permeable Ca2+ chelator
7673 BAY 091
Potent and selective PIP4K2A inhibitor
7573 BAY 1797
Selective P2X4 antagonist
7549 BAY 1816032
Potent and selective BUB1 kinase inhibitor
6857 BAY 293
Potent KRas/SOS1 interaction inhibitor
6906 BAY 293 Negative Control
Negative control for BAY 293 (Cat. No. 6857)
5970 BAY 299
Potent and selective BRD1 and TAF1 inhibitor
4430 BAY 41-2272
Soluble guanylyl cyclase (sGC) activator
5708 BAY 41-8543
Guanylyl cyclase (sGC) stimulator
6052 BAY 58-2667 hydrochloride
Potent soluble guanylyl cyclase (sGC) activator
5991 BAY 598
Potent and selective SMYD2 inhibitor
4472 BAY 60-6583
Potent partial A2B agonist; cardioprotective
6561 BAY 6035
Potent and selective SMYD3 inhibitor
6389 BAY 677
Inactive control for BAY 678 (Cat.No.5706)
5706 BAY 678
Potent and selective cell-permeable human neutrophil elastase (HNE) inhibitor
6562 BAY 707
Potent and selective MTH1 inhibitor
6817 BAY 8002
Potent dual MCT1/2 inhibitor; orally bioavailable
6579 BAY 826
Potent Tie2 inhibitor
6980 BAY 87-2243
Mitochondrial complex I inhibitor
6199 BAY 876
Potent and selective GLUT1 inhibitor
2732 BAY-u 3405
Dual TP/DP2 (CRTH2) receptor antagonist
5266 BAZ2-ICR
Selective BAZ2 inhibitor
4372 BC 11 hydrobromide
Selective urokinase (uPA) inhibitor
6791 BC-LI-0186
Leucyl-tRNA synthase (TRS)/Ras-related GTP-binding protein D (RagD) interaction inhibitor
5027 BCH
LAT1 inhibitor
7481 BCI
DUSP6 and DUSP1 inhibitor
3875 BCTC
TRPV1 antagonist
0956 BD 1047 dihydrobromide
σ1 selective antagonist
0883 BD 1063 dihydrochloride
Selective σ1 ligand, putative antagonist
3579 5-BDBD
Potent and selective P2X4 antagonist
2837 BDNF (human)
Activates TrkB and p75 receptors
7857 BDY FL Lenalidomide
Fluorescent cereblon ligand
7985 BDY FL Staurosporine
Fluorescent probe targeting kinases; kinase tracer for TR-FRET assays
7633 BDY FL Thalidomide
High affinity fluorescent probe for TR-FRET cereblon binding assay
7483 BDY FL VH032
High-affinity VHL fluorescent probe for TR-FRET and FP assays
5465 BDY FL, SE
Green BDY (BODIPY® or boron-dipyrromethene) fluorescent dye supplied with an NHS ester for the labeling of primary amines
4778 BETP
Positive allosteric modulator of GLP-1 receptors
3743 BF 2649 hydrochloride
Potent and selective H3 inverse agonist
6246 BF 738735
Potent and selective PI 4-kinase IIIβ inhibitor; broad spectrum enterovirus replication inhibitor
0348 2-BFI hydrochloride
Potent, selective I2 ligand. Putative agonist
5327 BGC 20-1531 hydrochloride
High affinity and selective EP4 antagonist
3326 BGC 20-761
High affinity 5-HT6 antagonist
6703 BGP 15
PARP inhibitor; cytoprotectant
3313 rac BHFF
Potent and selective postitive allosteric modulator of GABAB receptors
6116 BHPI
ERα antagonist; also activates unfolded protein response; active in vivo
6518 BI 01383298
Potent and selective SLC13A5 (Na+/citrate cotransporter) inhibitor
4641 BI 6015
Hepatocyte nuclear factor 4α (HNF4α) antagonist
3314 BI 78D3
Selective, competitive JNK inhibitor
6665 BI 9321
Nuclear receptor-binding SET domain (NSD) 3 antagonist; selectively binds PWWP1 domain
5590 BI 9564
Potent and selective BRD9 and BRD7 inhibitor; orally active
7466 BI dihydrochloride
DFHBI derivative for imaging of RNA in living cells that bind Broccoli aptamers
6141 BI-6901
Potent and selective CCR10 antagonist
4561 BIBN 4096
Potent and selective CGRP antagonist
2412 BIBO 3304 trifluoroacetate
Highly selective NPY Y1 receptor antagonist
2707 BIBP 3226 trifluoroacetate
Mixed NPY Y1 and NPFF receptor antagonist
2981 BIBR 1532
Selective telomerase inhibitor
7377 BIIE 0246 hydrochloride
Potent, selective and competitive non-peptide NPY Y2 receptor antagonist; active in vivo
4374 BIMU 8
Potent 5-HT4 agonist
4048 BINA
Selective positive allosteric modulator of mGlu2 receptors
3194 BIO
Potent GSK-3 inhibitor; also inhibits cdks
3910 BIO 1211
Selective α4β1 (VLA-4) inhibitor
5051 BIO 5192
Highly potent and selective inhibitor of integrin α4β1 (VLA-4)
5989 BIRB 796
High affinity and selective p38 kinase inhibitor
4776 BIRT 377
Potent negative allosteric modulator of LFA-1
3364 BIX 01294
GLP and G9a inhibitor
4842 BIX 02189
Selective MEK5 and ERK5 inhibitor
5512 BIX NHE1 inhibitor
Potent and selective NHE1 inhibitor
3797 BL 1249
K2P2.1 (TREK-1) and K2P10.1 (TREK-2) activator
2538 L-BMAA hydrochloride
Neurotoxic amino acid
5417 BMH 21
RNA polymerase I inhibitor; also p53 pathway activator
5488 BML 111
FPR2 (lipoxin A4 receptor) agonist
2665 BMS 191011
Potent KCa1.1 (BK) channel opener
3242 BMS 193885
Potent, competitive NPY Y1 receptor antagonist
3660 BMS 195614
Selective RARα antagonist
5654 BMS 265246
Cdk inhibitor; potently inhibits cdk1 and cdk2
2870 BMS 299897
Potent γ-secretase inhibitor
4609 BMS 303141
ATP citrate lyase inhibitor; orally bioavailable
5258 BMS 309403
Potent and selective FABP4 inhibitor
4806 BMS 345541
Selective allosteric inhibitor of IKK; anti-inflammatory
6878 BMS 466442
Potent and selective inhibitor of asc-1
3509 BMS 493
Pan-RAR inverse agonist
4774 BMS 536924
Dual IR/IGF1R inhibitor
5274 BMS 564929
Highly potent and muscle-selective androgen receptor (AR) agonist
5492 BMS 566419
Inosine monophosphatase dehydrogenase (IMPDH) inhibitor
4970 BMS 688521
Potent inhibitor of the LFA-1/ICAM interaction
3505 BMS 753
RARα-selective agonist
3410 BMS 961
Selective RARγ agonist
6974 BMS 986094
Inhibitor of HCV RNA-dependent RNA polymerase (RdRP; NS5b); potent hepatitis C virus (HCV) replication inhibitor
5983 BMS 986187
Potent positive allosteric modulator of δ receptors
3129 BMS CCR2 22
High affinity, potent CCR2 antagonist
5123 BMX-IN-1
Potent and irreversible BMX inhibitor
6047 BOP
Dual α9β1/α4β1 integrin inhibitor; preferentially mobilizes HSCs
6996 BOP-JF549
Yellow fluorescent dual α9β1/α4β1 integrin inhibitor comprising BOP conjugated to Janelia Fluor® 549; fluorogenic; photostable
6997 BOP-JF646
Red fluorescent dual α9β1/α4β1 integrin inhibitor comprising BOP conjugated to Janelia Fluor® 646; fluorogenic; photostable
5301 BPTES
Selective allosteric glutaminase (GLS1) inhibitor
6078 BPTU
P2Y1 allosteric antagonist
1500 BQ 788 sodium salt
Selective ETB antagonist
1188 BQ-123
Selective ETA antagonist
1189 BQ-3020
Selective ETB agonist
6872 BQCA
Positive allosteric modulator of M1 receptors
5312 BRACO 19 trihydrochloride
Telomerase inhibitor
7153 BRD 0539
Cell permeable and reversible Cas9 inhibitor
6438 BRD 6989
Cdk8 inhibitor; enhances IL-10 production
4037 BRD 7389
Ribosomal S6 kinase inhibitor
6284 BRD 73954
Dual histone deacetylase (HDAC) 6/8 inhibitor
Photoswitchable BET bromodomain Degrader (PHOTAC)
0948 BRL 37344, sodium salt
β3 agonist
1133 BRL 44408 maleate
Selective α2A antagonist
2237 BRL 50481
Selective PDE7 inhibitor
0699 BRL 52537 hydrochloride
Potent and selective κ agonist
5608 BS 181 dihydrochloride
Selective cdk7 inhibitor
6921 BSJ-03-123
Selective Cdk6 Degrader (PROTAC®)
6938 BSJ-03-204
Selective Cdk4/6 Degrader (PROTAC®)
6937 BSJ-04-132
Selective Cdk4 Degrader (PROTAC®)
7528 BSJ-4-116
Selective CDK12 PROTAC® Degrader
7529 BSJ-4-116-NC
Negative control for BSJ-4-116 (Cat. No. 7528).
6922 BSJ-Bump
Negative control for BSJ-03-123 (Cat. No. 6921)
5399 BTB1
Selective and ATP-competitive Kif18A inhibitor
6940 BTD
Selective TRPC5 activator
1870 BTS
Selective inhibitor of skeletal muscle myosin II ATPase activity
4724 BTT 3033
Selective inhibitor of integrin α2β1
4204 BTZO 1
MIF binder
0725 BU 224 hydrochloride
Potent, selective I2 ligand. Putative antagonist
2176 BVT 948
Non-competitive protein tyrosine phosphatase inhibitor
5545 BX 430
Selective P2X4 allosteric antagonist
3496 BX 471
Potent, selective CCR1 antagonist
2769 BX 513 hydrochloride
Selective CCR1 antagonist
4318 BX 795
PDPK1 (PDK1) inhibitor
0796 (R)-Baclofen
Selective GABAB agonist; active enantiomer of (RS)-Baclofen (Cat. No. 0417)
0417 (RS)-Baclofen
Selective GABAB agonist
1334 Bafilomycin A1
H+-ATPase (vacuolar) inhibitor
5585 Balicatib
Potent and selective cathepsin K inhibitor
4219 Banoxantrone dihydrochloride
Prodrug topoisomerase II inhibitor
7222 Baricitinib
Highly potent JAK1 and JAK2 inhibitor; also inhibits JAK3 and Tyk2
2961 Batimastat
Potent, broad spectrum MMP inhibitor
2160 Bax channel blocker
Allosteric inhibitor of Bax channel activation
1743 Bay 11-7085
Irreversible inhibitor of TNF-α-induced IκBα phosphorylation
1744 Bay 11-7821
E2 ubiquitin (Ub) conjugating enzymes inhibitor
2501 Bay 36-7620
mGlu1 inverse agonist
2711 Bay 55-9837
Potent and selective VPAC2 agonist
1544 (±)-Bay K 8644
CaV1.x activator
1545 (R)-(+)-Bay K 8644
CaV1.x blocker; (R)-(+)-enantiomer of (±)-Bay K 8644; also TMEM176B inhibitor
1546 (S)-(-)-Bay K 8644
CaV1.x activator; (S)-(-)-enantiomer of (±)-Bay K 8644
7981 Belinostat
Potent pan-HDAC inhibitor
3681 Bendamustine hydrochloride
Cytostatic agent; exhibits DNA alkylating and purine analog properties
3380 Benzamil
NCX inhibitor, Deg/ENaC channel blocker; amiloride (Cat. No. 0890) derivative
4117 Bepridil hydrochloride
Non-selective Ca2+ channel blocker; also NCX inhibitor
4180 Beraprost sodium
Potent prostacyclin IP receptor agonist
1956 Bestatin
Aminopeptidase inhibitor
0906 Betaxolol hydrochloride
Selective β1 antagonist
3906 Betulinic acid
Antitumor and anti-HIV agent; activates NF-κB. Also TGR5 agonist
5819 Bexarotene
Potent and selective RXR agonist
3389 Bicalutamide
Non-steroidal androgen receptor antagonist
2503 (-)-Bicuculline methiodide
GABAA antagonist; more water soluble version of (+)-bicuculline (Cat. No. 0130)
0109 (-)-Bicuculline methobromide
GABAA antagonist; more water soluble version of (+)-bicuculline (Cat. No. 0130)
0131 (-)-Bicuculline methochloride
GABAA antagonist; more water soluble version of (+)-bicuculline (Cat. No. 0130)
0130 (+)-Bicuculline
Potent GABAA antagonist
0767 Bifemelane hydrochloride
Non-selective MAO inhibitor
6304 BigLEN (mouse)
GPR171 agonist
3349 Biocytin
Versatile marker for neuroanatomical investigations
6571 Biotin-11-dUTP
Biotin-labeled dUTP
6572 Biotin-LC-NAD+
Biotinylated analog of β-NAD+; commonly used reagent in LSD1 and PARP1 assays
6573 Biotin-NAD+
Biotinylated-NAD+; substrate for ADP-ribosylation
7524 Biotin-PEG3-Azide
Biotin with PEG linker and reactive click handle
6241 Biotinyl Tyramide
Reagent widely used for signal amplification in IHC and FISH
2853 Biperiden hydrochloride
Muscarinic receptor antagonist; some selectivity for M1
5348 6,8-Bis(benzylthio)octanoic acid
PDH and KGDH inhibitor
4128 Bisindolylmaleimide II
Potent PKC inhibitor; also potent nAChR antagonist
5502 Blasticidin S HCl
Antibiotic; selection reagent for bis, bsr and BSD transformed cells
1853 (R)-(+)-Blebbistatin
Selective inhibitor of myosin II ATPase activity. Inactive enantiomer of (±)-blebbistatin (Cat. No. 1760)
1852 (S)-(-)-Blebbistatin
Selective inhibitor of myosin II ATPase activity. Active enantiomer of (±)-blebbistatin (Cat. No. 1760)
1760 (±)-Blebbistatin
Selective inhibitor of myosin II ATPase activity
5255 6-Bnz-cAMP sodium salt
Cell permeable cAMP analog
6977 Bobcat339
Ten-eleven translocation methylcytosine dioxygenase (TET) inhibitor
3730 Boc-MLF
FPR1 antagonist
7282 Bortezomib
High affinity proteasome inhibitor
6232 Bosentan
High affinity dual ETA and ETB receptor antagonist;orally bioavailable
4361 Bosutinib
Dual Src-Abl inhibitor; antiproliferative
5217 Bovine Serum Albumin
BSA (bovine serum albumin) is a blocking buffer for IHC, ICC, ELISA and Western blotting; used to block non-specific antibody binding. Commonly used in cell culture
3004 Bradykinin
Endogenous agonist at bradykinin receptors (B2 > B1)
3225 Lys-[Des-Arg9]Bradykinin
Selective B1 agonist
3522 Brain natriuretic peptide (1-32) (human)
Endogenous peptide agonist at ANP receptor A (NPR1)
1231 Brefeldin A
Disrupts protein translocation to Golgi
6196 Brequinar sodium
Potent and selective DHODH inhibitor
3568 Bretazenil
Benzodiazepine partial agonist
7271 Brivaracetam
SV2A ligand; antiepileptic
1140 8-Bromo-cAMP, sodium salt
Cell-permeable cAMP analog
1089 8-Bromo-cGMP, sodium salt
cGMP analog; activates PKG
7686 BromoTag® AGB1
Potent and selective Degrader of Brd4BD2 L387A fusion proteins (BromoTag®)
7688 BromoTag® AGB3
Selective Degrader of Brd4BD2 L387A fusion proteins (BromoTag®)
7687 BromoTag® cis-AGB1
Negative control for BromoTag® AGB1 (Cat. No. 7686)
0427 Bromocriptine mesylate
D2-like agonist (D2>D3>D4)
3549 3-Bromocytisine
Potent α4β4, α4β2 and α7 nAChR agonist
5015 5-BrdU
Synthetic thymidine analog; used for cell proliferation assays
0735 3-Bromo-7-nitroindazole
Selective nNOS inhibitor
7512 3-Bromopyruvate
MCT1 inhibitor; also inhibits hexokinase II
4758 Bromosporine
Broad spectrum bromodomain inhibitor
4316 Bropirimine
Immunomodulatory and antitumor compound
2383 Bryostatin 1
Protein kinase C activator
2671 Budesonide
Synthetic glucocorticoid; anti-inflammatory and chemopreventive
3108 Bumetanide
Na+/2Cl-/K+ (NKCC) symporter inhibitor
2133 α-Bungarotoxin
Selective α7 nAChR antagonist
2831 Bupropion hydrochloride
Non-selective inhibitor of dopamine and noradrenalin transporters
5791 Bz 423
ATP synthase inhibitor; proapoptotic
3312 BzATP triethylammonium salt
Photoaffinity label for ATPase; also P2X7 agonist and P2X1/P2Y1 partial agonist

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