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Displaying Products by Catalog Number (2400 - 2499)

Cat. No. Product Name / Activity
2400 FK 888
High affinity NK1 antagonist
2402 MRS 2211
Competitive P2Y13 antagonist
2404 Ambroxol hydrochloride
Na+ channel blocker
2407 FTI 277
Prodrug form of FTI 276 (Cat. No. 2406)
2408 Ro 90-7501
Inhibitor of Aβ42 fibril formation
2410 L-371,257
Potent and selective oxytocin receptor antagonist
2411 A-71623
Potent and selective CCK1 agonist; suppresses feeding
2412 BIBO 3304 trifluoroacetate
Highly selective NPY Y1 receptor antagonist
2414 H 1152 dihydrochloride
Selective Rho-kinase (ROCK) inhibitor
2415 HA 1100 hydrochloride
Cell-permeable, selective Rho-kinase inhibitor
2416 BIBX 1382 dihydrochloride
Highly selective EGFR-kinase inhibitor
2417 BIBU 1361 dihydrochloride
Selective inhibitor of EGFR-kinase
2418 LY 303511
Negative control of LY 294002 (Cat. No. 1130)
2419 GT 2016
Selective H3 antagonist
2420 [Pyr1]-Apelin-13
Potent peptide apelin agonist
2421 Scriptaid
Histone deacetylase inhibitor
2422 AKTide-2T
Akt/PKB substrate (synthetic)
2423 DAPTA
Chemokine receptor 5 (CCR5) antagonist
2424 Amyloid β-peptide (1-40) (rat)
Amyloid β-protein fragment
2425 Amyloid β-peptide (1-42) (rat)
Predominant amyloid β-protein fragment
2426 Apelin-36 (human)
Endogenous apelin agonist
2427 Apelin-36 (rat, mouse)
Endogenous apelin agonist
2429 Fexofenadine hydrochloride
H1 receptor antagonist; non-sedating antiallergic agent
2430 GGTI 298
Geranylgeranyltransferase I (GGTase I) inhibitor
2432 Anagrelide hydrochloride
Potent PDE3 inhibitor
2435 CCT 018159
Hsp90 inhibitor
2436 AC 55649
Selective RARβ2 agonist
2438 TMPH hydrochloride
Neuronal nAChR antagonist
2440 NNC 26-9100
Selective sst4 agonist
2441 JNJ 10191584 maleate
Selective H4 antagonist; orally active
2442 CGP 53353
Selective inhibitor of PKCβII
2443 RITA
MDM2-p53 interaction inhibitor
2444 (1R,1'S,3'R/1R,1'R,3'S)-L-054,264
Potent and selective sst2 agonist
2445 Obestatin (rat)
Endogenous reported anorexigenic peptide
2446 AS 101
Immunomodulator; inhibits IL-10 synthesis and potentiates IL-1α, IL-2 and TNF-α release
2447 Desmethyl-YM 298198
Derivative of mGlu1 antagonist YM 298198 (Cat. No. 2448)
2448 YM 298198 hydrochloride
Highly potent, selective non-competitive mGlu1 antagonist
2450 NF 157
Selective P2Y11/P2X1 antagonist
2451 LY 344864 hydrochloride
Potent and selective 5-HT1F agonist
2452 LY 2183240
Highly potent anandamide uptake inhibitor; also inhibits FAAH
2453 LY 379268
Highly selective group II mGlu agonist
2454 CH 275
Potent and selective sst1 agonist
2456 Co 101244 hydrochloride
GluN2B-selective NMDA antagonist
2457 Arcyriaflavin A
Potent cdk4 inhibitor; also potently inhibits CaM kinase II; antiviral
2458 ZM 447439
Inhibits Aurora kinase B
2459 Tropisetron hydrochloride
Potent 5-HT3 antagonist; also α7 nAChR partial agonist
2460 Lazabemide hydrochloride
Selective MAO-B inhibitor
2463 SCH 442416
Very selective, high affinity A2A antagonist
2464 TNP-ATP triethylammonium salt
Potent, selective P2X antagonist
2465 SDZ WAG 994
Potent, selective A1 agonist
2466 UK 14,304 tartrate
α2 agonist. Water-soluble form of UK 14,304 (Cat. No. 0425)
2467 CGS 20625
Selective benzodiazepine partial agonist
2469 IBC 293
Selective agonist for the GPR109B (HM74) receptor. Antilipolytic
2470 Nimesulide
Cyclooxygenase-2 (COX-2) inhibitor
2471 ER 27319 maleate
Selective Syk kinase inhibitor
2472 Triacsin C
Inhibitor of acyl-CoA synthetase
2473 GW 4064
Selective farnesoid X receptor (FXR) agonist
2474 GW 3965 hydrochloride
Orally active liver X receptor (LXR) agonist
2475 ZM 323881 hydrochloride
Potent, selective inhibitor of VEGFR-2
2476 SR 11302
AP-1 inhibitor; antitumor agent
2477 Proxyfan oxalate
High affinity H3 ligand
2478 2-Pyridylethylamine dihydrochloride
H1 agonist
2479 JTE 907
Selective CB2 receptor inverse agonist
2481 JTC 801
Selective NOP antagonist
2483 Costunolide
Inhibitor of human telomerase activity
2484 (±)-AC 7954 hydrochloride
Non-peptide UT receptor agonist
2485 Glycyl-H 1152 dihydrochloride
Selective Rho-kinase (ROCK) inhibitor. More selective analog of H 1152 dihydrochloride (Cat. No. 2414)
2489 C 75
Potent fatty acid synthase inhibitor; proapoptotic
2490 (±)-Clopidogrel hydrochloride
Selective P2Y12 antagonist
2491 Xaliproden hydrochloride
High affinity 5-HT1A agonist; orally active
2492 MNITMT
Novel, non-toxic immunosuppressive agent
2493 VUF 5681 dihydrobromide
Potent H3 receptor silent antagonist
2494 VUF 8430 dihydrobromide
Potent and high affinity H4 agonist
2495 Melperone hydrochloride
5-HT2A antagonist; also D2 antagonist; neuroleptic
2496 DR 2313
PARP-1 and PARP-2 inhibitor
2498 PNU 120596
Positive allosteric modulator of α7 nAChRs; active in vivo
2499 ZM 306416 hydrochloride
Inhibitor of VEGF receptor tyrosine kinase

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