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Displaying Products by Catalog Number (3500 - 3599)

Cat. No. Product Name / Activity
3501 Decanoyl-RVKR-CMK
Subtilisin/Kex2p-like proprotein convertase inhibitor
3502 Epothilone B
Microtubule stabilization agent; promotes tubulin polymerization
3503 HLI 373
Hdm2 inhibitor; activates p53-dependent transcription
3504 Risedronate
Farnesyl diphosphate (FPP) synthase inhibitor
3505 BMS 753
RARα-selective agonist
3506 NVP DPP 728 dihydrochloride
Potent, orally active dipeptidyl peptidase IV (DPP-IV) inhibitor
3507 AM 80
RARα agonist; anticancer agent
3508 LG 101506
Selective RXR modulator
3509 BMS 493
Pan-RAR inverse agonist
3512 NPE-caged-proton
Caged proton
3513 N2-Methyl-L-arginine
Lysosomal system c L-arginine uptake inhibitor
3515 FK 228
Potent and selective class I histone deacetylase inhibitor; antitumor
3516 Tunicamycin
Antibiotic; GlcNAc phosphotransferase inhibitor
3517 Nebivolol hydrochloride
Highly selective β1-adrenoceptor antagonist
3518 S 24795
α7 nAChR partial agonist
3520 C-type natriuretic peptide (1-22) (human, rat, swine)
Endogenous peptide agonist at NPR2
3521 Sirtinol
Selective sirtuin family deacetylase inhibitor
3522 Brain natriuretic peptide (1-32) (human)
Endogenous peptide agonist at ANP receptor A (NPR1)
3523 FERb 033
Potent and selective ERβ agonist
3525 ACSF
Artificial cerebrospinal fluid
3526 BIM, Biotinylated
Bim peptide fragment
3527 SB 243213 dihydrochloride
Selective 5-HT2C inverse agonist
3528 SCIO 469 hydrochloride
Selective p38 MAPK inhibitor
3529 PD 168568 dihydrochloride
Potent and selective D4 antagonist
3530 HQL 79
Human hematopoietic prostaglandin D synthase (H-PGDS) inhibitor
3531 AT 56
L-PGDS inhibitor
3532 endo-IWR 1
Wnt/β-catenin signaling inhibitor; axin stabilizer
3533 IWP 2
PORCN inhibitor; inhibits Wnt processing and secretion
3534 PNU 74654
β-catenin binder; inhibits Wnt signaling
3535 Sivelestat sodium salt
Selective leukocyte elastase inhibitor
3536 Cetrorelix Acetate
Potent GnRH receptor antagonist
3537 MMK 1
Potent and selective FPR2 agonist
3540 Orlistat
Pancreatic, gastric and carboxylester lipase inhibitor; antiobesity and antihypercholesterolemic activity
3541 BAY-X 1005
Orally active 5-lipoxygenase activating protein (FLAP) inhibitor
3542 CP 316819
Selective glycogen phosphorylase inhibitor
3543 Suplatast tosylate
Th2 cytokine synthesis inhibitor; antiasthmatic
3544 KU 55933
Potent and selective ATM kinase inhibitor
3545 Histamine dihydrochloride
Endogenous histamine receptor agonist
3546 (-)-Nicotine ditartrate
Prototypical nAChR agonist
3547 Serotonin hydrochloride
Endogenous 5-HT receptor agonist
3548 Dopamine hydrochloride
Endogenous agonist at dopamine D1-5 receptors
3549 3-Bromocytisine
Potent α4β4, α4β2 and α7 nAChR agonist
3550 Melatonin
Endogenous hormone; agonist at MT1 and MT2
3551 INH1
Hec1 inhibitor; causes arrest of mitosis
3552 PD 173212
Potent CaV2.2 blocker
3553 Parstatin (human)
Peptide cleaved from PAR1 upon receptor activation
3554 Parstatin (mouse)
Peptide cleaved from PAR1 upon receptor activation
3555 CRSP-1
Endogenous central calcitonin agonist
3556 SER 601
Potent, selective CB2 agonist
3561 L189
DNA ligase I, III and IV inhibitor
3562 LU AA33810
Potent NPY Y5 receptor antagonist
3563 Margatoxin
Potent KV1.3 channel blocker
3565 ONO AE3 208
High affinity and selective EP4 antagonist
3567 TC-S 7003
Potent Lck inhibitor
3568 Bretazenil
Benzodiazepine partial agonist
3569 Xanomeline oxalate
Functionally selective M1 agonist
3570 Z-Guggulsterone
Broad spectrum steroid receptor ligand. More active isomer of guggulsterone (Cat. No. 2013)
3571 SB 657510
Selective urotensin-II (UT) receptor antagonist
3572 GSK 650394
Serum- and glucocorticoid-regulated kinase (SGK) inhibitor
3573 SB 612111 hydrochloride
Selective NOP antagonist
3574 RuBi-Glutamate
Caged glutamate; excited by visible wavelengths
3575 VU 0155069
Potent and selective PLD1 inhibitor
3576 (±)-5'-Chloro-5'-deoxy-ENBA
Highly selective A1 agonist
3577 G-1
Potent and selective GPER agonist
3578 AS 605240
Potent and selective PI 3-kinase γ (PI 3-Kγ) inhibitor
3579 5-BDBD
Potent and selective P2X4 antagonist
3580 HKI 357
Dual irreversible inhibitor of ErbB2 and EGFR
3581 C 021 dihydrochloride
Potent CCR4 antagonist
3584 Golgicide A
Potent, selective and reversible inhibitor of GBF1 ArfGEF
3585 Org 12962 hydrochloride
Selective 5-HT2C agonist
3586 Sumatriptan succinate
5-HT1A, 5-HT1B and 5-HT1D agonist
3587 A 922500
Potent DGAT-1 inhibitor
3588 Estropipate
Estrogen receptor agonist and OATP1B1 inhibitor
3589 PIM-1 Inhibitor 2
Pim-1 kinase inhibitor
3590 Gambogic acid
Apoptosis inducer. Activates caspases and inhibits Bcl-2 family proteins
3591 VO-OHpic
Potent PTEN inhibitor
3592 Goserelin acetate
GnRH receptor agonist
3594 GRK2i
GRK2 inhibitory polypeptide. Gβγ antagonist
3595 CHR 2797
Aminopeptidase inhibitor
3596 Voglibose
Orally active α-glucosidase inhibitor
3597 Indiplon
Positive allosteric modulator of GABAA; acts at benzodiazepine site
3599 TAK 165
Potent and selective ErbB2 inhibitor

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