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Displaying Products by Catalog Number (2900 - 2999)

Cat. No. Product Name / Activity
2900 UK 370106
Highly selective MMP-3 and MMP-12 inhibitor
2901 SB 242084
Selective 5-HT2C antagonist; brain penetrant
2902 D 4476
Selective CK1 inhibitor. Also inhibits TGF-βRI
2903 Granisetron hydrochloride
5-HT3 antagonist
2905 TB 21007
α5-selective GABAA inverse agonist
2906 TRO 19622
Binds voltage-dependent anion channel (VDAC)
2907 SU 9516
Cdk inhibitor; potently inhibits cdk1 and cdk2
2908 EO 1428
Selective inhibitor of p38α and p38β2
2910 H 89 dihydrochloride
Protein kinase A inhibitor
2911 Ro 04-6790
Potent and selective 5-HT6 antagonist
2913 Ro 64-5229
Selective, non-competitive mGlu2 antagonist
2915 MRS 2690
Potent P2Y14 agonist
2917 Venlafaxine hydrochloride
5-HT and NA reuptake inhibitor (SNRI)
2918 Veratridine
Voltage-gated Na+ channel opener
2919 NPE-caged-HPTS
Caged fluorescent pH indicator
2921 MTEP hydrochloride
Potent and selective mGlu5 antagonist
2924 NBMPR
Equilibrative nucleoside transporter 1 (ENT1) inhibitor
2926 FPA 124
Akt/PKB inhibitor
2927 WS 3
TRPM8 agonist; cooling agent
2928 CB 13
Potent dual CB1/CB2 agonist
2930 PI 103 hydrochloride
Inhibitor of PI 3-kinase, mTOR and DNA-PK
2931 Spinorphin
Enkephalin-degrading and ACE inhibitor
2932 CP 465022 hydrochloride
Selective and non-competitive AMPA antagonist
2934 [Lys8]-Vasopressin
Antidiuretic hormone
2935 [Arg8]-Vasopressin
Antidiuretic hormone
2936 NSC 66811
MDM2 antagonist. Disrupts MDM2-p53 interaction
2937 Atipamezole hydrochloride
Selective α2 antagonist
2939 A 83-01
Selective inhibitor of TGF-βRI, ALK4 and ALK7
2940 PAF (C16)
Endogenous platelet-activating factor (PAF)
2942 CI 1020
Highly selective, orally active ETA antagonist
2945 SNX 482
Potent and selective CaV2.3 blocker
2946 TRAM 34
Potent and highly selective KCa3.1 channel blocker
2950 Acetyl-Calpastatin (184-210) (human)
Selective calpain inhibitor
2951 [Des-octanoyl]-Ghrelin (rat)
Major circulating form of ghrelin; devoid of activity at GHS receptor
2952 CI 994
Class I histone deacetylase inhibitor; orally active
2953 CyPPA
Activator of KCa2.2 and KCa2.3 channels
2954 PX 12
Thioredoxin-1 inhibitor
2956 Picropodophyllotoxin
Selective IGF1R inhibitor
2957 Org 27569
Potent allosteric modulator of CB1 receptors
2958 DSP-4
Adrenergic neurotoxin
2959 Lercanidipine hydrochloride
CaV1.x blocker
2960 Felodipine
CaV1.x blocker
2961 Batimastat
Potent, broad spectrum MMP inhibitor
2962 6'-GNTI dihydrochloride
Selective κ/δ opioid heterodimer receptor agonist
2963 MMPIP hydrochloride
Potent and selective negative allosteric modulator of mGlu7 receptors
2964 Doxazosin mesylate
α1 antagonist
2965 Diprenorphine
Non-selective opioid antagonist
2966 CGP 3466B maleate
GAPDH inhibitor; neuroprotective
2967 Phenserine
Cholinesterase inhibitor
2968 Spironolactone
Mineralocorticoid receptor antagonist
2969 SR 12813
Pregnane X receptor agonist
2972 A 438079 hydrochloride
Competitive P2X7 antagonist
2973 Piracetam
Modulates Na+-flux at AMPA receptors; nootropic
2974 CCG 2046
Inhibitor of regulator of G-protein signaling 4 (RGS4)
2975 Sarcosine
GlyT1 inhibitor
2976 A 803467
Selective NaV1.8 channel blocker
2977 GW 843682X
Selective inhibitor of PLK1 and PLK3
2978 PYR 41
Ubiquitin-activating enzyme (E1) inhibitor
2979 TCS PIM-1 1
Selective, ATP-competitive Pim-1 kinase inhibitor
2980 CX 546
AMPA potentiator
2981 BIBR 1532
Selective telomerase inhibitor
2983 GM 6001
Broad spectrum MMP inhibitor
2985 LEP (116-130) (mouse)
Synthetic leptin peptide fragment
2986 YM 230888
Selective mGlu1 antagonist
2988 VULM 1457
ACAT inhibitor
2989 Epoprostenol
Endogenous IP receptor agonist
2992 PKC 412
Protein kinase C inhibitor
2993 RS 127445 hydrochloride
High affinity and selective 5-HT2B antagonist
2994 Signal Enhancer Hikari
Antibody-antigen signal enhancer
2995 NS 1738
Positive allosteric modulator of α7 nAChRs; active in vivo
2999 RWJ 67657
Potent, selective p38α and p38β inhibitor

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