All Products

Displaying Products by Catalog Number (7000 - 7099)

Cat. No. Product Name / Activity
7001 AT 7867
Potent pan-Akt and PKA inhibitor
7002 KYA 1797K
Wnt/β-catenin signaling inhibitor
7004 NAI
Reagent for RNA SHAPE-MaP experiments in vivo; cell permeable
7005 4-Thiouridine
Photoreactive uridine analog for RNA sequencing
7006 PDD 00017272
Potent PARG inhibitor
7007 PDD 00017238
High affinity and potent PARG inhibitor
7009 PDD 00031705
Negative control for PDD 00017238 (Cat. No. 7007)
7010 EM 163
TIR-TIR interaction inhibitor
7013 OptoBI-1
Photoswitchable TRPC3/6/7 agonist
7015 IA-Alkyne
Broad spectrum cysteine reactive probe
7018 CBR-470-1
PGK1 inhibitor; activates Nrf2
7020 LDV
α4β1 (VLA-4) ligand
7026 Veliparib dihydrochloride
High affinity PARP-1 and -2 inhibitor; orally bioavailable
7027 LY 2033298
Selective positive allosteric modulator of M4 receptors; active in vivo; antipsychotic
7029 GX 201
Potent and selective Nav1.7 blocker; analgesic
7030 GW 280264X
Potent ADAM10 and ADAM17 inhibitor
7033 AY 77
Potent PAR2 biased agonist; exhibits bias for Ca2+ signaling
7034 AY 254
Potent PAR2 biased agonist; exhibits bias for ERK1/2 signaling
7038 Palonosetron hydrochloride
Highly potent and high affinity 5-HT3 antagonist
7039 SK 609
Dopamine D3 receptor biased agonist
7040 C 176
mSTING antagonist
7044 (±)-α-Lipoic acid
Liquid-liquid phase separated condensate modifier; reduces stress granule formation
7045 (±)-α-Lipoamide
Phase-separated condensate modifier; orally bioavailable
7046 1,6-Hexanediol
Tool for probing liquid-liquid phase separation
7048 Ruxolitinib phosphate
Phosphate salt of Ruxolitinib (Cat. No. 7064); potent and selective JAK1/JAK2 inhibitor
7049 Nintedanib
Potent VEGFR, PDGFR and FGFR inhibitor
7050 Ribociclib
Dual cdk4/cdk6 inhibitor; orally bioavailable
7051 Tasquinimod
High affinity HDAC4 negative allosteric modulator; also binds S100A9; antiangiogenic
7052 Lopinavir
Highly potent and selective HIV-1 protease inhibitor
7054 T4
Modulator of alternative polyadenylation; inhibits rod photoreceptor gene expression via Nr2e3
7055 WS 383
Potent, selective and reversible DCN1-UBC12 interaction inhibitor
7056 Conduritol B epoxide
Irreversible glucocerebrosidase (β-glucosidase) inhibitor; used to generate Gaucher disease models
7057 VU 0071063
Selective activator of SUR1 Kir6.2 channels
7059 GLPG 0187
Potent αv integrin inhibitor
7064 Ruxolitinib
Potent and selective JAK1/JAK2 inhibitor; orally bioavailable
7065 Kainic acid (synthetic)
Kainate agonist; excitant and neurotoxin
7066 RCGD 423
gp130 modulator; activates JAK/STAT signaling
7070 Mirabegron
Potent and selective β3 agonist
7071 GSK 2239633A
Potent CCR4 antagonist
7073 VH 032 amide-alkylC3-amine
VHL ligand with alkyl linker and terminal amine for onward chemistry
7074 VH 032 amide-alkylC7-amine
VHL ligand with alkyl linker and terminal amine for onward chemistry
7075 Lenalidomide 4'-PEG1-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
7076 Lenalidomide 4'-PEG3-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
7081 LY 2886721 Hydrochloride
Potent and selective β-secretase (BACE) inhibitor
7082 DL 175
Potent and selective GPR84 agonist
7086 StemRegenin 1
Aryl hydrocarbon receptor (AhR) antagonist; promotes HSC expansion and engraftment
7087 AGI 5198
Potent and selective inhibitor of mutant isocitrate dehydrogenase 1 (mIDH1)
7088 Janelia Fluor® 646, Azide
Red dye (Reactive group: azide). Applications: super resolution microscopy e.g. dSTORM & STED, confocal, and live cell imaging
7089 CSN5i-3
Potent and selective CSN5 (COP9 signalosome) inhibitor
7091 Miro1 Reducer
Promotes mitochondrial Rho GTPase 1 (Miro1) degradation
7093 Lenalidomide 4'-PEG2-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
7094 Pomalidomide 4'-PEG1-acid
Cereblon ligand with PEG linker and terminal acid for onward chemistry
7095 Pomalidomide 4'-PEG5-acid
Cereblon ligand with PEG linker and terminal acid for onward chemistry
7096 Pomalidomide 4'-alkylC3-acid
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7097 Pomalidomide 4'-alkylC7-acid
Cereblon ligand with alkyl linker and terminal acid for onward chemistry

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