All ProductsDisplaying Products Alphabetically by Name (E)
| Cat. No. | Product Name / Activity |
|---|---|
| 5550 | E 2012 |
| γ-secretase modulator; Notch-sparing | |
| 5208 | E 64 |
| Potent and irreversible cysteine protease inhibitor | |
| 4545 | E 64d |
| Cathepsin inhibitor; interferes with autolysosomal digestion | |
| 6785 | E 7820 |
| α2 integrin inhibitor; anti-angiogenic | |
| 1808 | E-4031 dihydrochloride |
| KV11.1 (hERG) channel blocker; inhibits rapid delayed rectifier K+ current (IKr) | |
| 3993 | EB 1089 |
| Vitamin D receptor (VDR) agonist | |
| 4140 | EB 47 |
| Potent PARP-1 inhibitor | |
| 1041 | 1-EBIO |
| Epithelial KCa channel activator | |
| 4701 | EC 144 |
| High affinity, potent and selective Hsp90 inhibitor | |
| 4011 | EC 23 |
| Synthetic retinoid; induces differentiation of stem cells | |
| 7714 | EDA-DA New |
| Unnatural dipeptide building block with alkyne group for functionalizing peptidoglycan | |
| 2811 | EDTA |
| Chelating agent | |
| 6986 | EG 00229 trifluoroacetate |
| Neuropilin 1 (NRP1) receptor antagonist; inhibits VEGFA binding to NRP1 | |
| 4524 | EGCG |
| β-secretase (BACE) inhibitor; inhibits amyloid assembly | |
| 2807 | EGTA |
| Calcium chelating agent | |
| 1261 | EHNA hydrochloride |
| Adenosine deaminase inhibitor | |
| 3872 | EHT 1864 |
| Potent Rac family inhibitor | |
| 6248 | EHop 016 |
| Rac inhibitor | |
| 7231 | EIDD 1931 |
| Viral RNA-dependent RNA polymerase (RdRP) inhibitor; broad spectrum antiviral nucleoside | |
| 3378 | EIPA |
| Inhibits TRPP3-mediated currents; also inhibits the Na+/H+ exchanger (NHE) | |
| 6293 | ELA-14 (human) |
| Potent apelin agonist; bioactive fragment of ELA-32 (Cat. No. 6291) | |
| 6291 | ELA-32 (human) |
| Potent and high affinity apelin agonist; stimulates angiogenesis | |
| 7010 | EM 163 New |
| TIR-TIR interaction inhibitor | |
| 4470 | EMD 281014 hydrochloride |
| Selective 5-HT2A antagonist | |
| 2382 | EMD 386088 hydrochloride |
| Potent 5-HT6 agonist | |
| 7508 | EMD 527040 hydrochloride |
| ανβ6 integrin inhibitor | |
| 1849 | EMD 66684 |
| Potent and selective non-peptide AT1 antagonist | |
| 7424 | EMI 48 |
| Inhibitor of EGFR mutants | |
| 5646 | EML 425 |
| Reversible and non-competitive CBP/p300 inhibitor | |
| 4558 | EMPA |
| Highly potent and selective OX2 antagonist; brain penetrant | |
| 7474 | EN6 |
| H+ ATPase activator; activates autophagy; inactivates mTORC1 signaling | |
| 3576 | (±)-5'-Chloro-5'-deoxy-ENBA |
| Highly selective A1 agonist | |
| 2908 | EO 1428 |
| Selective inhibitor of p38α and p38β2 | |
| 4518 | EPPTB |
| Trace amine 1 (TA1) receptor antagonist; also displays inverse agonism | |
| 5567 | EPZ 004777 |
| Highly potent DOT1L inhibitor | |
| 6516 | EPZ 015666 |
| Potent and selective PRMT5 inhibitor | |
| 2471 | ER 27319 maleate |
| Selective Syk kinase inhibitor | |
| 3823 | ER 50891 |
| Selective RARα antagonist | |
| 5924 | ER 819762 |
| Potent EP4 receptor antagonist; orally bioavailable | |
| 4276 | ERB 041 |
| Potent ERβ agonist | |
| 6632 | ERGi-USU |
| Rio2 kinase (RIOK2) inhibitor; inhibits ERG protein | |
| 5393 | ERK5-IN-1 |
| Potent and selective ERK5 inhibitor | |
| 6320 | ESI 05 |
| Epac2 inhibitor | |
| 4773 | ESI 09 |
| Epac inhibitor | |
| 7462 | ET 18-OCH3 |
| Selective PI-PLC inhibitor, also PAF receptor agonist | |
| 4702 | ETP 45658 |
| Potent PI 3-kinase inhibitor; also inhibits DNA-PK and mTOR | |
| 5183 | ETP 45835 dihydrochloride |
| Mnk1 and Mnk2 inhibitor | |
| 2780 | EX 527 |
| Selective SIRT1 inhibitor | |
| 5728 | EXP 3174 |
| Potent and selective AT1 antagonist | |
| 4876 | Eact |
| Activator of Ca2+-activated Cl- channel transmembrane protein 16A (TMEM16A) | |
| 5245 | Ebselen |
| Glutathione peroxidase mimic; peroxynitrite scavenger | |
| 6832 | Ec2la |
| Positive allosteric modulator of CB2 receptors; active in vivo | |
| 5520 | Echinomycin |
| Highly potent and selective HIF-1α inhibitor | |
| 3202 | Echistatin, α1 isoform |
| αVβ3 and glycoprotein IIb/IIIa (integrin αIIbβ3) inhibitor | |
| 4784 | Edaglitazone |
| Potent and selective PPARγ agonist; antidiabetic | |
| 0786 | Edaravone |
| Anti-ischemic and antioxidant | |
| 3922 | Eeyarestatin I |
| Potent inhibitor of ER-associated protein degradation and translocation | |
| 4646 | Elacridar hydrochloride |
| P-gp and BCRP inhibitor | |
| 5316 | Elinogrel |
| P2Y12 antagonist | |
| 2195 | Eliprodil |
| Non-competitive and GluN2B-selective NMDA antagonist | |
| 3357 | Ellipticine |
| Antitumor and intercalating agent; inhibits DNA topoisomerase II | |
| 2156 | Embelin |
| Inhibitor of X-linked inhibitor of apoptosis (XIAP); cell-permeable and antitumor | |
| 7342 | Emetine dihydrochloride |
| RNA polymerase inhibitor; inhibits replication of a broad range of RNA and DNA viruses, including SARS-CoV-2 and Zika | |
| 7310 | Emricasan |
| Potent pan-caspase inhibitor | |
| 1055 | Endomorphin-1 |
| Potent and selective μ agonist | |
| 1160 | Endothelin 1 (human, porcine) |
| Potent vasoconstrictor peptide | |
| 1164 | Endothelin 2 (human) |
| ETA/ETB agonist | |
| 1162 | Endothelin 3 (human, rat) |
| Potent vasoconstrictor | |
| 3705 | Endoxifen |
| Potent antiestrogen; ERα ligand | |
| 1889 | [Leu5]-Enkephalin |
| Endogenous opioid agonist peptide | |
| 1693 | Enoximone |
| PDE3 inhibitor | |
| 4720 | Entacapone |
| Potent COMT inhibitor; blocks α-synuclein aggregation | |
| 6234 | Entecavir |
| Potent and selective hepatitis B virus inhibitor | |
| 0684 | (±)-Epibatidine |
| High affinity nAChR agonist | |
| 6340 | Epiblastin A |
| CK1 inhibitor; converts epiblast stem cells to ESCs and promotes ESC self-renewal | |
| 3260 | Epirubicin hydrochloride |
| Inhibits DNA synthesis and function. Inhibits DNA topoisomerase II | |
| 2397 | Eplerenone |
| Selective mineralocorticoid receptor antagonist | |
| 4958 | Eplivanserin hemifumarate |
| Potent and selective 5-HT2A antagonist | |
| 2989 | Epoprostenol |
| Endogenous IP receptor agonist | |
| 4725 | Eptifibatide |
| Glycoprotein IIb/IIIa inhibitor; inhibits platelet aggregation | |
| 5449 | Erastin |
| Mitochondrial VDAC modulator; also Ferroptosis activator | |
| 7199 | (±)-Eriodictyol |
| Potent TRPV1 antagonist; also antioxidant; activates Nrf2/ARE signaling | |
| 7194 | Erlotinib Hydrochloride |
| Potent, reversible EGFR tyrosine kinase inhibitor | |
| 4796 | Escitalopram oxalate |
| Selective serotonin reuptake inhibitor (SSRI) | |
| 2823 | α-Estradiol |
| Endogenous estrogen receptor agonist | |
| 2824 | β-Estradiol |
| Endogenous ER agonist | |
| 6204 | 7-Ethoxyresorufin |
| Fluorometric CYP450 substrate | |
| 5950 | Ethyl LipotF |
| Selective FTO inhibitor | |
| 5712 | 4-Ethynyl-N-ethyl-1,8-naphthalimide |
| Fluorescent probe for imaging of cell surface, intracellular fucosylated glycoproteins and glycolipids | |
| 7206 | 5-Ethynyluridine New |
| Uridine analog, used for labeling RNA synthesis | |
| 1847 | Eticlopride hydrochloride |
| D2 and D3 antagonist (D3 > D2) | |
| 3113 | Etifoxine hydrochloride |
| Ligand of the translocator protein (TSPO); also GABAA receptor potentiator | |
| 1471 | Etomidate |
| GABA-mimetic; selectively interacts with β2- and β3-subunit containing GABAA receptors | |
| 4539 | (R)-(+)-Etomoxir sodium salt |
| Carnitine palmitoyltransferase I (CPT1) inhibitor | |
| 1226 | Etoposide |
| Topoisomerase II inhibitor | |
| 0845 | Evans Blue tetrasodium salt |
| Dye for assessing cell viability and blood brain barrier permeability; also EAAT inhibitor and iGluR antagonist | |
| 6188 | Everolimus |
| mTOR inhibitor; Immunosuppressant | |
| 7507 | Evofosfamide New |
| Hypoxia-activated DNA alkylating agent prodrug | |
| 5833 | Ex 26 |
| Potent and selective S1P1 receptor antagonist | |
| 3759 | Exemestane |
| Steroidal aromatase (CYP19) inhibitor | |
| 2081 | Exendin-3 (9-39) amide |
| Potent GLP-1 receptor antagonist | |
| 1933 | Exendin-4 |
| Potent GLP-1 receptor agonist | |
| 1850 | Exo1 |
| Inhibits Golgi-ER traffic; blocks exocytosis |
Tocris Products by Catalog Number
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