All Products

Displaying Products Alphabetically by Name (E)

Cat. No. Product Name / Activity
5550 E 2012
γ-secretase modulator; Notch-sparing
5208 E 64
Potent and irreversible cysteine protease inhibitor
4545 E 64d
Cathepsin inhibitor; interferes with autolysosomal digestion
6785 E 7820
α2 integrin inhibitor; anti-angiogenic
1808 E-4031 dihydrochloride
KV11.1 (hERG) channel blocker; inhibits rapid delayed rectifier K+ current (IKr)
3993 EB 1089
Vitamin D receptor (VDR) agonist
4140 EB 47
Potent PARP-1 inhibitor
1041 1-EBIO
Epithelial KCa channel activator
4701 EC 144
High affinity, potent and selective Hsp90 inhibitor
4011 EC 23
Synthetic retinoid; induces differentiation of stem cells
2811 EDTA
Chelating agent
6986 EG 00229 trifluoroacetate
Neuropilin 1 (NRP1) receptor antagonist; inhibits VEGFA binding to NRP1
4524 EGCG
β-secretase (BACE) inhibitor; inhibits amyloid assembly
2807 EGTA
Calcium chelating agent
1261 EHNA hydrochloride
Adenosine deaminase inhibitor
3872 EHT 1864
Potent Rac family inhibitor
6248 EHop 016
Rac inhibitor
7231 EIDD 1931
Viral RNA-dependent RNA polymerase (RdRP) inhibitor; broad spectrum antiviral nucleoside
3378 EIPA
Inhibits TRPP3-mediated currents; also inhibits the Na+/H+ exchanger (NHE)
6293 ELA-14 (human)
Potent apelin agonist; bioactive fragment of ELA-32 (Cat. No. 6291)
6291 ELA-32 (human)
Potent and high affinity apelin agonist; stimulates angiogenesis
4470 EMD 281014 hydrochloride
Selective 5-HT2A antagonist
2382 EMD 386088 hydrochloride
Potent 5-HT6 agonist
1849 EMD 66684
Potent and selective non-peptide AT1 antagonist
5646 EML 425
Reversible and non-competitive CBP/p300 inhibitor
4558 EMPA
Highly potent and selective OX2 antagonist; brain penetrant
3576 (±)-5'-Chloro-5'-deoxy-ENBA
Highly selective A1 agonist
2908 EO 1428
Selective inhibitor of p38α and p38β2
4518 EPPTB
Trace amine 1 (TA1) receptor antagonist; also displays inverse agonism
5567 EPZ 004777
Highly potent DOT1L inhibitor
6516 EPZ 015666
Potent and selective PRMT5 inhibitor
2471 ER 27319 maleate
Selective Syk kinase inhibitor
3823 ER 50891
Selective RARα antagonist
5924 ER 819762
Potent EP4 receptor antagonist; orally bioavailable
4276 ERB 041
Potent ERβ agonist
6632 ERGi-USU
Rio2 kinase (RIOK2) inhibitor; inhibits ERG protein
5393 ERK5-IN-1
Potent and selective ERK5 inhibitor
6320 ESI 05
Epac2 inhibitor
4773 ESI 09
Epac inhibitor
7462 ET 18-OCH3
Selective PI-PLC inhibitor, also PAF receptor agonist
4702 ETP 45658
Potent PI 3-kinase inhibitor; also inhibits DNA-PK and mTOR
5183 ETP 45835 dihydrochloride
Mnk1 and Mnk2 inhibitor
2780 EX 527
Selective SIRT1 inhibitor
5728 EXP 3174
Potent and selective AT1 antagonist
4876 Eact
Activator of Ca2+-activated Cl- channel transmembrane protein 16A (TMEM16A)
5245 Ebselen
Glutathione peroxidase mimic; peroxynitrite scavenger
6832 Ec2la
Positive allosteric modulator of CB2 receptors; active in vivo
5520 Echinomycin
Highly potent and selective HIF-1α inhibitor
3202 Echistatin, α1 isoform
αVβ3 and glycoprotein IIb/IIIa (integrin αIIbβ3) inhibitor
4784 Edaglitazone
Potent and selective PPARγ agonist; antidiabetic
0786 Edaravone
Anti-ischemic and antioxidant
3922 Eeyarestatin I
Potent inhibitor of ER-associated protein degradation and translocation
0792 Efaroxan hydrochloride
α2 antagonist and I1, I3 ligand
4646 Elacridar hydrochloride
P-gp and BCRP inhibitor
1920 Eledoisin-Related Peptide
Tachykinin receptor ligand
5316 Elinogrel
P2Y12 antagonist
2195 Eliprodil
Non-competitive and GluN2B-selective NMDA antagonist
3357 Ellipticine
Antitumor and intercalating agent; inhibits DNA topoisomerase II
2156 Embelin
Inhibitor of X-linked inhibitor of apoptosis (XIAP); cell-permeable and antitumor
7342 Emetine dihydrochloride
RNA polymerase inhibitor; inhibits replication of a broad range of RNA and DNA viruses, including SARS-CoV-2 and Zika
1055 Endomorphin-1
Potent and selective μ agonist
1056 Endomorphin-2
Potent and selective μ agonist
1160 Endothelin 1 (human, porcine)
Potent vasoconstrictor peptide
1164 Endothelin 2 (human)
ETA/ETB agonist
1162 Endothelin 3 (human, rat)
Potent vasoconstrictor
3705 Endoxifen
Potent antiestrogen; ERα ligand
1889 [Leu5]-Enkephalin
Endogenous opioid agonist peptide
1693 Enoximone
PDE3 inhibitor
4720 Entacapone
Potent COMT inhibitor; blocks α-synuclein aggregation
6234 Entecavir
Potent and selective hepatitis B virus inhibitor
6102 Ep23, 5'-DY647
High affinity fluorescently tagged aptamer for EpCam
0684 (±)-Epibatidine
High affinity nAChR agonist
6340 Epiblastin A
CK1 inhibitor; converts epiblast stem cells to ESCs and promotes ESC self-renewal
3260 Epirubicin hydrochloride
Inhibits DNA synthesis and function. Inhibits DNA topoisomerase II
2397 Eplerenone
Selective mineralocorticoid receptor antagonist
4958 Eplivanserin hemifumarate
Potent and selective 5-HT2A antagonist
2989 Epoprostenol
Endogenous IP receptor agonist
4725 Eptifibatide
Glycoprotein IIb/IIIa inhibitor; inhibits platelet aggregation
6158 (S)-Equol
Potent estrogen receptor β (ERβ) agonist; dihydrotestosterone antagonist
5449 Erastin
Mitochondrial VDAC modulator; also Ferroptosis activator
4146 Ercalcidiol
Metabolite of vitamin D2
7199 (±)-Eriodictyol
Potent TRPV1 antagonist; also antioxidant; activates Nrf2/ARE signaling
7194 Erlotinib Hydrochloride
Potent, reversible EGFR tyrosine kinase inhibitor
4796 Escitalopram oxalate
Selective serotonin reuptake inhibitor (SSRI)
2823 α-Estradiol
Endogenous estrogen receptor agonist
2824 β-Estradiol
Endogenous ER agonist
6204 7-Ethoxyresorufin
Fluorometric CYP450 substrate
5950 Ethyl LipotF
Selective FTO inhibitor
5712 4-Ethynyl-N-ethyl-1,8-naphthalimide
Click-activated fluorescent probe
1847 Eticlopride hydrochloride
D2 and D3 antagonist (D3 > D2)
3113 Etifoxine hydrochloride
Ligand of the translocator protein (TSPO); also GABAA receptor potentiator
1471 Etomidate
GABA-mimetic; selectively interacts with β2- and β3-subunit containing GABAA receptors
4539 (R)-(+)-Etomoxir sodium salt
Carnitine palmitoyltransferase I (CPT1) inhibitor
1226 Etoposide
Topoisomerase II inhibitor
0845 Evans Blue tetrasodium salt
Dye for assessing cell viability and blood brain barrier permeability; also EAAT inhibitor and iGluR antagonist
6188 Everolimus
mTOR inhibitor; Immunosuppressant
5833 Ex 26
Potent and selective S1P1 receptor antagonist
3759 Exemestane
Steroidal aromatase (CYP19) inhibitor
2081 Exendin-3 (9-39) amide
Potent GLP-1 receptor antagonist
1933 Exendin-4
Potent GLP-1 receptor agonist
1850 Exo1
Inhibits Golgi-ER traffic; blocks exocytosis

Tocris Products by Catalog Number