Cat. No. | Product Name / Activity |
---|---|
6201 | J 2156 |
Selective high affinity human sst4 agonist | |
6202 | Vilazodone hydrochloride |
Potent 5-HT1A partial agonist and SSRI; antidepressant | |
6203 | GSK 9311 hydrochloride |
Negative control for GSK 6853 | |
6204 | 7-Ethoxyresorufin |
Fluorometric CYP450 substrate | |
6208 | MS 275 |
HDAC (Class I) inhibitor | |
6210 | ci-IP3/PM |
Caged inositol triphosphate | |
6218 | Galiellalactone |
STAT3 inhibitor; active in vivo | |
6219 | Arformoterol tartrate |
Long-acting β2 agonist (LABA) | |
6221 | PKI (5-24) |
High affinity PKA inhibitor | |
6222 | PFM 01 |
MRE11 endonuclease inhibitor | |
6223 | XY 018 |
RORγ antagonist; inhibits AR expression | |
6227 | TAT-Gap19 |
Cx43 hemichannel blocker | |
6228 | H10 |
PARP14 inhibitor; cell-permeable | |
6229 | LP 922761 |
Potent AAK1 inhibitor; peripherally restricted | |
6230 | Rucaparib camsylate |
PARP inhibitor | |
6231 | Dacomitinib |
Potent irreversible pan ErbB inhibitor | |
6232 | Bosentan |
High affinity dual ETA and ETB receptor antagonist;orally bioavailable | |
6233 | Retigabine |
KV7 channel activator | |
6234 | Entecavir |
Potent and selective hepatitis B virus inhibitor | |
6236 | O8 OGG1 Inhibitor |
Potent and selective 8-oxoguanine DNA glycosylase 1 (OGG1) inhibitor | |
6237 | FPS ZM1 |
High affinity antagonist of RAGE | |
6238 | PKRA 7 |
Potent prokineticin (PK) 1 and 2 receptor antagonist; antitumor; BBB penetrant | |
6239 | SAK 3 |
Potent CaV3.1 and 3.3 activator; orally bioavailable | |
6240 | DG 041 |
Potent and selective EP3 antagonist; antiplatelet and antithrombotic | |
6241 | Biotinyl Tyramide |
Reagent widely used for signal amplification in IHC and FISH | |
6242 | AG 205 |
Progesterone receptor membrane component 1 (Pgrmc1) ligand | |
6243 | ML 385 |
Nrf2 inhibitor; phenotypically lethal | |
6244 | OG-L002 |
Potent LSD1 inhibitor | |
6245 | SM 16 |
Potent TGF-βRI inhibitor; orally bioavailable | |
6246 | BF 738735 |
Potent and selective PI 4-kinase IIIβ inhibitor; broad spectrum enterovirus replication inhibitor | |
6248 | EHop 016 |
Rac inhibitor | |
6249 | Givinostat hydrochloride |
Histone deacetylase inhibitor | |
6250 | Filipin III |
Fluorescent cholesterol stain; also polyene antibiotic | |
6251 | L Moses dihydrochloride |
High affinity and selective PCAF bromodomain inhibitor | |
6253 | F 127 (20% solution in DMSO) |
Nonionic detergent | |
6254 | Flutax 2 |
Green fluorescent taxol derivative; binds microtubules | |
6255 | Fluo-4 AM |
Cell-permeable, fluorescent Ca2+ indicator | |
6256 | OG 488 BAPTA-1 AM |
Cell-permeable, fluorescent Ca2+ indicator | |
6258 | CC 401 dihydrochloride |
High affinity JNK inhibitor; also inhibits HCMV replication | |
6259 | RAGE antagonist peptide |
RAGE antagonist | |
6261 | VCP 171 |
Positive allosteric modulator (PAM) of A1 receptors; also allosteric partial agonist in absence of orthosteric agonist | |
6264 | Caerulein |
CCK agonist | |
6265 | Lonafarnib |
Potent farnesyltransferase inhibitor | |
6266 | Taxol Janelia Fluor® 646 |
Red fluorescent taxol derivative; probe for microtubule staining; protocol available | |
6267 | Taxol Janelia Fluor ® 549 |
Yellow fluorescent taxol derivative; probe for microtubule staining | |
6269 | JT010 |
Potent and selective TRPA1 channel activator | |
6270 | Tubastatin A hydrochloride |
Potent HDAC6 inhibitor | |
6271 | ST 034307 |
Adenylyl cyclase 1 (AC1) inhibitor; analgesic and active in vivo | |
6272 | KYP 2047 |
High affinity prolyl oligopeptidase inhibitor; anti-angiogenic, neuroprotective and brain penetrant | |
6273 | CRT 0105950 |
Potent LIMK1/2 inhibitor | |
6278 | JNJ 55511118 |
High affinity and selective negative modulator of AMPA receptors containing TARP-γ8 | |
6279 | JNJ 39758979 dihydrochloride |
High affinity and selective histamine H4 antagonist; orally bioavailable | |
6280 | FIN 56 |
Ferroptosis activator | |
6281 | SLM 6031434 hydrochloride |
Selective sphingosine kinase 2 (Sphk2) inhibitor | |
6284 | BRD 73954 |
Dual histone deacetylase (HDAC) 6/8 inhibitor | |
6285 | Megestrol Acetate |
Synthetic progesterone analog | |
6286 | st-Ht31 |
Inhibits PKA/AKAP interactions; cell permeable | |
6289 | JH-II-127 |
Potent and selective LRRK2 inhibitor | |
6290 | WZ 4002 |
Potent mutant-selective EGFR inhibitor | |
6296 | Janelia Fluor® 525, SE |
Yellow dye (Reactive group: NHS ester). Applications: super resolution microscopy, confocal and live cell imaging | |
6297 | AP 20187 |
Chemical inducer of protein dimerization; active in vivo | |
6298 | MS 21570 |
GPR171 antagonist | |
6299 | MS 15203 |
Potent and selective GPR171 partial agonist |