All Products

Displaying Products by Catalog Number (5300 - 5399)

Cat. No. Product Name / Activity
5300 BI 605906
Selective IKKβ inhibitor
5301 BPTES
Selective allosteric glutaminase (GLS1) inhibitor
5303 GSK 2194069
Potent human fatty acid synthase (hFASN) inhibitor
5304 FICZ
High affinity aryl hydrocarbon receptor (AhR) agonist
5305 Verteporfin
YAP inhibitor
5306 KJ Pyr 9
High affinity Myc inhibitor
5307 MM 102
Potent WDR5/MLL interaction inhibitor
5308 ASP 2535
Potent and selective GlyT1 inhibitor
5309 SP 100030
NF-κB and AP-1 dual inhibitor
5310 ASP 3026
Potent anaplastic lymphoma kinase (ALK) inhibitor; also potent ACK inhibitor
5311 RHPS 4 methosulfate
Telomerase inhibitor
5312 BRACO 19 trihydrochloride
Telomerase inhibitor
5314 SMBA 1
High affinity and selective activator of Bax
5315 Rostafuroxin
Na+/K+ ATPase modulator; antihypertensive agent
5316 Elinogrel
P2Y12 antagonist
5317 WWL 123
α/β-hydrolase domain 6 (ABHD6) inhibitor; antiepileptic
5318 AEE 788
Potent EGFR and VEGFR inhibitor
5319 ACT 462206
Potent, dual orexin receptor antagonist
5320 CORM 3
Water-soluble carbon monoxide-releasing molecule
5321 PSNCBAM-1
Negative allosteric modulator of CB1 receptors
5322 VU 0409106
Potent and selective negative allosteric modulator of mGlu5 receptors
5323 WDR5 0103
WDR5 antagonist
5324 M8 B hydrochloride
Potent and selective TRPM8 channel blocker
5325 Rosiglitazone
Potent and selective PPARγ agonist; antidiabetic agent
5326 CHR 6494 trifluoroacetate
Potent and selective haspin inhibitor
5327 BGC 20-1531 hydrochloride
High affinity and selective EP4 antagonist
5328 TY 52156
S1P3 receptor antagonist
5329 CKI 7 dihydrochloride
CK1 inhibitor
5330 AEG 40730 dihydrochloride
IAP antagonist; induces apoptosis
5331 CPI 203
BET bromodomain inhibitor; arrests cell cycle at G1 phase
5332 SP 141
High affinity MDM2 inhibitor
5334 TH 588
Potent MTH1 inhibitor
5335 Angiotensin A
Potent endogenous vasoconstrictor peptide - derivative of angiotensin II (Cat. No. 1158)
5337 ML 365
Potent and selective K2P3.1 (TASK-1) channel blocker
5338 PK-THPP
Potent K2P9.1 (TASK-3) channel blocker
5339 PFK 15
Selective PFKFB3 inhibitor
5340 NSC 617145
Werner syndrome helicase (WRN) inhibitor
5342 SCR7 pyrazine
Enhances HDR efficiency
5343 TPPB
High affinity PKC activator; also APP modulator
5344 ML 349
Selective and reversible lysophospholipase 2 (LYPLA2) inhibitor
5345 ML 348
Selective and reversible lysophospholipase 1 (LYPLA1) inhibitor
5347 Kisspeptin 10 (dog)
Endogenous ligand for canine kisspeptin receptor
5348 6,8-Bis(benzylthio)octanoic acid
PDH and KGDH inhibitor
5349 Treprostinil
Potent prostacyclin (PGI2) analog
5351 PQ 69
Potent and selective A1 inverse agonist
5353 Gap19
Cx43 hemichannel blocker
5355 TC-G 1008
Potent and selective GPR39 agonist
5356 SGX 523
Selective and potent c-MET kinase inhibitor
5357 DC 260126
FFA1 (GPR40) antagonist
5358 Cariporide
Selective NHE1 inhibitor; cardioprotective and antitumor
5359 Rifaximin
Pregnane X receptor agonist; antibiotic
5361 GSK LSD 1 dihydrochloride
Potent and selective LSD1 inhibitor
5362 TASP 0433864
Selective positive allosteric modulator of mGlu2 receptors
5363 NHI 2
LDHA inhibitor
5364 Hydroxy Dynasore
Dynamin inhibitor; analog of dynasore (Cat. No. 2897)
5365 LLY 507
Potent SMYD2 inhibitor
5367 SGC 707
Potent and selective allosteric inhibitor of PRMT3
5369 Norleual
Highly potent HGF/c-MET inhibitor; also AT4 antagonist
5371 Clemizole hydrochloride
TRPC5 blocker; also H1 antagonist
5372 Bioymifi
DR5 (TRAIL receptor) agonist; induces apoptosis
5373 C34
TLR4 inhibitor
5374 GLP-1 (7-37)
Endogenous bioactive GLP-1 receptor ligand
5375 BIX
BiP (Hsp70-5) ER chaperone inducer
5376 Pregnenolone sulfate sodium salt
NMDA potentiator; also GABAA inhibitor and TRPM3 activator
5377 VU 0483605
Positive allosteric modulator of mGlu1 receptors
5378 VU 0422288
Selective positive allosteric modulator of group III mGlu receptors
5379 VU 0469650 hydrochloride
Potent and selective negative allosteric modulator of mGlu1 receptors
5380 ML 297
Selective Kir3.1/3.2 (GIRK1/2) channel activator
5382 C16
PKR inhibitor
5385 GSK 5959
Potent and selective BRPF1 inhibitor
5387 ML 354
Selective PAR4 antagonist
5388 RQ 00203078
Potent and selective TRPM8 antagonist; orally active
5389 Ro 48-8071 fumarate
2,3-Oxidosqualene cyclase (OSC) inhibitor; blocks cholesterol synthesis
5390 Tobramycin
Aminoglycoside antibiotic
5391 SPP 86
Potent RET inhibitor
5393 ERK5-IN-1
Potent and selective ERK5 inhibitor
5395 Virodhamine trifluoroacetate
TFA salt of virodhamine, an endogenous cannabinoid receptor mixed agonist/antagonist
5397 A01
High affinity Smurf1 inhibitor; enhances BMP signaling
5398 NQTrp
Potent inhibitor of Aβ oligomer and fibril formation
5399 BTB1
Selective and ATP-competitive Kif18A inhibitor

Tocris Products Alphabetically by Name