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Displaying Products by Catalog Number (3900 - 3999)

Cat. No. Product Name / Activity
3900 TCS 2314
α4β1 (VLA-4) antagonist
3903 Neuropeptide Y (scrambled)
Control peptide for neuropeptide Y (Cat. No. 1173)
3904 WAY 208466 dihydrochloride
Selective 5-HT6 agonist
3905 NAADP tetrasodium salt
Ca2+ mobilizing agent
3906 Betulinic acid
Antitumor and anti-HIV agent; activates NF-κB. Also TGR5 agonist
3907 27-Hydroxycholesterol
LXR agonist; also ER partial agonist
3908 Ibutilide hemifumarate
Blocks IKr, hERG and L-type Ca2+ channels; class III antiarrhythmic
3909 Toceranib
Potent PDGFR and VEGFR inhibitor
3910 BIO 1211
Selective α4β1 (VLA-4) inhibitor
3911 S 18986
Positive allosteric modulator of AMPA receptors
3912 HX 531
Potent RXR antagonist
3913 HX 630
RXR synergist
3914 A 419259 trihydrochloride
Inhibitor of Src family kinases
3915 VX 745
Potent and selective p38α inhibitor
3917 Daptomycin
Antibiotic; inhibits protein, DNA and RNA synthesis in gram-positive bacteria
3918 Pyrimethamine
Potent inhibitor of multidrug and toxin extrusion (MATE) transporters; also DHFR and STAT3 inhibitor
3919 SC 236
Selective cyclooxygenase-2 (COX-2) inhibitor
3920 AMG 548
Potent and selective p38α inhibitor
3922 Eeyarestatin I
Potent inhibitor of ER-associated protein degradation and translocation
3923 PF 998425
Non-steroidal androgen receptor antagonist
3924 OPC 21268
Orally active vasopressin V1 antagonist
3928 XCT 790
Selective ERRα inverse agonist
3929 SJ 172550
MDMX inhibitor. Disrupts MDMX-p53 interaction
3930 NFAT Inhibitor
Inhibitor of calcineurin-mediated NFAT activation
3931 Ticlopidine hydrochloride
Selective P2Y12 antagonist
3932 Orphanin FQ (1-11)
Potent NOP agonist; displays analgesic properties
3933 WAY 267464 dihydrochloride
Potent non-peptide oxytocin receptor agonist
3934 Benidipine hydrochloride
Non-selective Cav blocker; also mineralocorticoid receptor antagonist
3935 RWJ 52353
α2D agonist
3936 CDP 840 hydrochloride
Potent and selective PDE4 inhibitor
3937 ANR 94
Adenosine A2A antagonist
3938 TCS 5861528
TRPA1 blocker
3939 YM 58483
Inhibitor of SOCE in non-excitable cells
3940 GSK 789472 hydrochloride
D3 antagonist. Also D2 partial agonist
3941 TCS 1205
GABAA agonist; displays subtype selectivity
3942 TCS 1105
GABAA α2 benzodiazepine agonist
3943 PG 01
CFTR potentiator; corrects F508del-CFTR conductance defect
3945 Colivelin
STAT3 activator; also protects against β-amyloid neurotoxicity
3946 TNP
Inhibitor of IP6K; also inhibits IP3K
3947 exo-IWR 1
Negative control for endo-IWR 1 (Cat. No. 3532)
3948 Terfenadine
H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker
3949 CBiPES hydrochloride
Positive allosteric modulator of mGlu2 receptors
3950 CK 666
Arp2/3 inhibitor; inhibits actin polymerization
3951 WZ 811
Potent CXCR4 antagonist
3953 cis-Ned 19
Fluorescently labels NAADP receptors in intact cells; inhibits Ca2+ release
3954 trans-Ned 19
Fluorescently labels NAADP receptors in intact cells; inhibits Ca2+ release
3959 YIL 781 hydrochloride
Ghrelin receptor (GHS-R1a) antagonist
3960 NVP 231
Potent, selective and reversible CerK inhibitor
3961 GSK 3787
Potent and selective PPARδ antagonist
3962 kb NB 142-70
Selective PKD inhibitor; analog of CID 755673 (Cat. No. 3327)
3963 AZM 475271
Src tyrosine kinase inhibitor
3965 Tesaglitazar
PPARα/γ agonist
3966 AR-A 014418
Selective GSK-3 inhibitor
3967 GPi 688
Allosteric glycogen phosphorylase inhibitor
3968 AZD 5438
Cdk inhibitor; potently inhibits cdk1, 2, 5 and 9
3969 AR-C 102222
Selective iNOS inhibitor
3970 Ercalcitriol
Active metabolite of vitamin D2
3972 AA 29504
Positive allosteric modulator of GABAA receptors
3973 Latrunculin A
Inhibitor of actin assembly and polymerization
3974 Latrunculin B
Inhibitor of actin polymerization
3975 Zearalenone
Estrogen receptor ligand; mycotoxin
3976 Deoxynivalenol
Mycotoxin; potent protein synthesis inhibitor
3977 3-Methyladenine
Class III PI 3-kinase inhibitor; also inhibits autophagy
3978 MEN 11270
Selective B2 antagonist; analog of HOE 140 (Cat. No. 3014)
3979 Alexidine dihydrochloride
Selective inhibitor of PTPMT1
3982 Mdivi 1
Selective dynamin inhibitor; attenuates mitochondrial division and apoptosis
3983 PSB 0739
Highly potent P2Y12 antagonist
3984 Nutlin-3
MDM2 antagonist; inhibits MDM2-p53 interaction
3986 SR 58611A hydrochloride
β3 agonist; displays anxiolytic and antidepressant effects
3988 Hesperadin hydrochloride
Potent Aurora kinase B inhibitor
3989 AMTB hydrochloride
TRPM8 blocker
3991 NPEC-caged-serotonin
Caged serotonin
3992 NPEC-caged-dopamine
Caged dopamine
3993 EB 1089
Vitamin D receptor (VDR) agonist
3994 AZ 3146
Potent and selective Mps1 kinase inhibitor
3995 GI 254023X
Selective ADAM10 metalloprotease inhibitor
3996 Zotepine
5-HT2A antagonist; also D2 and H1 antagonist; atypical antipsychotic
3997 Tazarotene
Receptor-selective retinoid; binds RAR-β and -γ
3998 LDN 57444
Ubiquitin C-terminal hydrolase-L1 (UCH-L1) inhibitor
3999 Cyclofenil
Selective estrogen receptor modulator (SERM)

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