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Displaying Products by Catalog Number (3900 - 3999)

Cat. No. Product Name / Activity
3900 TCS 2314
α4β1 (VLA-4) antagonist
3904 WAY 208466 dihydrochloride
Selective 5-HT6 agonist
3905 NAADP tetrasodium salt
Ca2+ mobilizing agent
3906 Betulinic acid
Antitumor and anti-HIV agent; activates NF-κB. Also TGR5 agonist
3907 27-Hydroxycholesterol
LXR agonist; also ER partial agonist
3908 Ibutilide hemifumarate
Blocks IKr, hERG and L-type Ca2+ channels; class III antiarrhythmic
3910 BIO 1211
Selective α4β1 (VLA-4) inhibitor
3912 HX 531
Potent RXR antagonist
3913 HX 630
RXR synergist
3914 A 419259 trihydrochloride
Inhibitor of Src family kinases
3915 VX 745
Potent and selective p38α inhibitor
3917 Daptomycin
Antibiotic; inhibits protein, DNA and RNA synthesis in gram-positive bacteria
3918 Pyrimethamine
Potent inhibitor of multidrug and toxin extrusion (MATE) transporters; also DHFR and STAT3 inhibitor
3919 SC 236
Selective cyclooxygenase-2 (COX-2) inhibitor
3920 AMG 548
Potent and selective p38α inhibitor
3922 Eeyarestatin I
Potent inhibitor of ER-associated protein degradation and translocation
3924 OPC 21268
Orally active vasopressin V1 antagonist
3928 XCT 790
Selective ERRα inverse agonist
3930 NFAT Inhibitor
Inhibitor of calcineurin-mediated NFAT activation
3933 WAY 267464 dihydrochloride
Potent non-peptide oxytocin receptor agonist
3937 ANR 94
Adenosine A2A antagonist
3938 TCS 5861528
TRPA1 blocker
3939 YM 58483
Inhibitor of SOCE in non-excitable cells
3945 Colivelin
STAT3 activator; also protects against β-amyloid neurotoxicity
3946 TNP
Inhibitor of IP6K; also inhibits IP3K
3948 Terfenadine
H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker
3950 CK 666
Arp2/3 inhibitor; inhibits actin polymerization
3953 cis-Ned 19
Fluorescently labels NAADP receptors in intact cells; inhibits Ca2+ release
3954 trans-Ned 19
Fluorescently labels NAADP receptors in intact cells; inhibits Ca2+ release
3959 YIL 781 hydrochloride
Ghrelin receptor (GHS-R1a) antagonist
3960 NVP 231
Potent, selective and reversible CerK inhibitor
3961 GSK 3787
Potent and selective PPARδ antagonist
3962 kb NB 142-70
Selective PKD inhibitor; analog of CID 755673 (Cat. No. 3327)
3963 AZM 475271
Src tyrosine kinase inhibitor
3965 Tesaglitazar
PPARα/γ agonist
3966 AR-A 014418
Selective GSK-3 inhibitor
3968 AZD 5438
Cdk inhibitor; potently inhibits cdk1, 2, 5 and 9
3973 Latrunculin A
Inhibitor of actin assembly and polymerization
3974 Latrunculin B
Inhibitor of actin polymerization
3975 Zearalenone
Estrogen receptor ligand; mycotoxin
3976 Deoxynivalenol
Mycotoxin; potent protein synthesis inhibitor
3977 3-Methyladenine
Class III PI 3-kinase inhibitor; also inhibits autophagy
3979 Alexidine dihydrochloride
Selective inhibitor of PTPMT1
3982 Mdivi 1
Selective dynamin inhibitor; attenuates mitochondrial division and apoptosis
3983 PSB 0739
Highly potent P2Y12 antagonist
3984 Nutlin-3
MDM2 antagonist; inhibits MDM2-p53 interaction
3986 SR 58611A hydrochloride
β3 agonist; displays anxiolytic and antidepressant effects
3988 Hesperadin hydrochloride
Potent Aurora kinase B inhibitor
3989 AMTB hydrochloride
TRPM8 blocker
3993 EB 1089
Vitamin D receptor (VDR) agonist
3994 AZ 3146
Potent and selective Mps1 kinase inhibitor
3995 GI 254023X
Selective ADAM10 metalloprotease inhibitor

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