All Products

Displaying Products by Catalog Number (1100 - 1199)

Cat. No. Product Name / Activity
1100 Camptothecin
DNA topoisomerase inhibitor
1101 Cyclosporin A
Calcineurin inhibitor
1102 Procaterol hydrochloride
Potent β2 agonist
1103 Ketoconazole
Cytochrome P450c17 inhibitor
1104 2-Cl-IB-MECA
Highly selective A3 agonist
1105 AF-DX 116
Selective M2 antagonist
1107 ATPA
Potent and selective GluK1 kainate agonist
1110 Genistein
EGFR kinase inhibitor. Also estrogen and PPARγ ligand
1111 ACPT-I
Group III mGlu agonist
1112 ACPT-II
Competitive mGlu receptor antagonist
1114 CGP 37157
Antagonist of mitochondrial Na+/Ca2+ exchange
1115 AM 281
Potent and selective CB1 inverse agonist
1116 AM 404
Anandamide transport inhibitor
1117 AM 251
Potent CB1 antagonist; also GPR55 agonist
1119 NocII
Orphan neuropeptide
1120 AM 630
Selective CB2 inverse agonist
1122 Telenzepine dihydrochloride
Potent, selective M1 antagonist
1123 (S)-(+)-Niguldipine hydrochloride
α1 antagonist, L-type Ca2+ channel blocker
1124 (R)-(-)-Niguldipine hydrochloride
α1 antagonist, L-type Ca2+ channel blocker. Less active enantiomer of Niguldipine hydrochloride (Cat. No. 1123)
1125 Quercetin
Non-selective PI 3-kinase inhibitor
1126 Dexamethasone
Anti-inflammatory glucocorticoid
1127 Yohimbine hydrochloride
Selective α2 antagonist
1128 Picrotoxin
GABAA antagonist
1129 BRL 54443
Potent 5-ht1E and 5-HT1F agonist
1130 LY 294002 hydrochloride
Prototypical PI 3-kinase inhibitor; also inhibits other kinases
1133 BRL 44408 maleate
Selective α2A antagonist
1134 CGP 12177 hydrochloride
β3 partial agonist. β12 antagonist
1136 Okadaic acid
Protein phosphatase 1 and 2A inhibitor
1138 Thapsigargin
Potent inhibitor of SERCA ATPase
1139 L-NIL hydrochloride
Selective iNOS inhibitor
1140 8-Bromo-cAMP, sodium salt
Cell-permeable cAMP analog
1141 Dibutyryl-cAMP, sodium salt
Cell-permeable cAMP analog
1144 U0126
Potent, selective inhibitor of MEK1 and 2
1145 L-733,060 hydrochloride
Potent NK1 antagonist
1147 SKF 96365 hydrochloride
TRPC channel inhibitor; also inhibits store-operated Ca2+ entry
1148 Siguazodan
PDE3 inhibitor
1149 Bombesin
Involved in gastrointestinal tract function
1151 CRF (human, rat)
Stimulates ACTH release
1153 Neuropeptide Y (human, rat)
Influences feeding and sexual behavior
1154 Pancreatic Polypeptide (human)
NPY Y4 agonist; involved in gastrointestinal tract function
1156 Substance P
Sensory neuropeptide; inflammatory mediator
1157 Somatostatin
Influences growth hormone release
1158 Angiotensin II
Potent vasoconstrictor peptide
1159 Calcitonin (salmon)
Affects bone formation and resorption
1160 Endothelin 1 (human, porcine)
Potent vasoconstrictor peptide
1161 CGRP (rat)
Potent vasodilator
1162 Endothelin 3 (human, rat)
Potent vasoconstrictor
1164 Endothelin 2 (human)
ETA/ETB agonist
1165 Somatostatin 1-28
sst agonist
1166 CCK Octapeptide, sulfated
C-terminal octapeptide of CCK
1167 Leupeptin hemisulfate
Inhibits trypsin-like/cysteine proteases
1169 CGRP 8-37 (rat)
CGRP antagonist
1171 DAMGO
Selective μ agonist
1173 Neuropeptide Y (porcine)
Influences feeding and sexual behavior
1175 Sarafotoxin S6c
Selective ETB agonist
1176 [Leu31,Pro34]-Neuropeptide Y (human, rat)
NPY Y1 receptor agonist
1178 [Sar9,Met(O2)11]-Substance P
Potent and selective NK1 agonist
1179 Galanin (1-30) (human)
Endogenous galanin receptor agonist
1180 [D-Ala2]-Deltorphin II
Selective δ agonist peptide
1181 CGRP 8-37 (human)
CGRP antagonist
1182 VIP (guinea pig)
Involved in neurotransmission and smooth muscle relaxation
1183 PACAP 1-27
Potent stimulator of adenylyl cyclase
1184 α-helical CRF 9-41
CRF antagonist
1185 Thrombin Receptor Agonist Peptide
Causes platelet aggregation and secretion
1186 PACAP 1-38
Potent stimulator of adenylyl cyclase
1188 BQ-123
Selective ETA antagonist
1189 BQ-3020
Selective ETB agonist
1190 Pepstatin A
Selective and high affinity cathepsin D inhibitor
1191 Amyloid β-Peptide (1-40) (human)
Amyloid β-protein fragment
1192 Mastoparan
Activates Gi and Go
1193 Melittin
Inhibits Gs and stimulates Gi activity
1194 MDL 29,913
Selective NK2 antagonist
1196 IRL-1620
Highly selective ETB agonist
1198 Nocistatin (human)
Human putative counterpart of nocistatin
1199 NF 279
Potent and selective P2X1 antagonist

Tocris Products Alphabetically by Name