All Products

Displaying Products by Catalog Number (6500 - 6599)

Cat. No. Product Name / Activity
6500 Janelia Fluor® 549, Maleimide
Yellow dye (Reactive group: maleimide). Applications: super resolution microscopy e.g. dSTORM & STED, confocal, flow and live cell imaging
6502 Janelia Fluor® 549, Tetrazine
Yellow dye (Reactive group: tetrazine). Applications: super resolution microscopy e.g. dSTORM & STED, confocal and live cell imaging
6503 Janelia Fluor® 549, free acid
Yellow dye (Reactive group: free acid). Applications: super resolution microscopy e.g. dSTORM & STED, confocal, flow and live cell imaging
6505 Avasimibe
ACAT inhibitor
6506 PF 06551600 malonate
Potent and selective JAK3 inhibitor
6507 Saxagliptin hydrochloride
High affinity DPP-IV inhibitor; active in vivo
6508 GSK 1702934A
Potent and selective TRPC3/6 activator
6510 LNT 1
Potent flap endonuclease 1 (FEN1) inhibitor; induces DNA damage response
6515 (D)-PPA 1
PD-1/PD-L1 interaction inhibitor
6516 EPZ 015666
Potent and selective PRMT5 inhibitor
6517 Liraglutide
Highly potent, long-acting GLP-1 receptor agonist
6518 BI 01383298
Potent and selective SLC13A5 (Na+/citrate cotransporter) inhibitor
6520 Abiraterone acetate
Potent CYP17A1 inhibitor
6521 I-BET 762
Potent and high affinity BET bromodomain inhibitor; anti-inflammatory; orally bioavailable.
6524 TL 12-186
Multikinase Degrader (PROTAC®)
6525 TL 13-27
Negative control for TL 12-186 (Cat. No. 6524)
6526 Dynarrestin
Inhibitor of Hedgehog (Hh) signaling; inhibits cytoplasmic dynein
6528 SGC AAK1 1
AAK1 and BMP2K inhibitor; activates Wnt signaling
6529 SGC AAK1 1N
Negative control for SGC AAK1 1 (Cat.No. 6528)
6530 R 121919 hydrochloride
High affinity CRF1 antagonist; orally bioavailable
6531 NLS-StAx-h
Wnt signaling inhibitor; inhibits β-catenin-transcription factor interactions
6532 THAL SNS 032
Potent and selective Cdk9 Degrader (PROTAC®)
6534 TH 5427 hydrochloride
Potent NUDT5 inhibitor
6535 NVP 2
Potent and selective ATP-competitive CDK9 inhibitor
6537 UNC 2881
Potent Mer kinase inhibitor
6538 PF 04449913 maleate
Potent Smo antagonist
6539 Obatoclax mesylate
Inhibitor of Bcl-2 family members; antiapoptotic
6541 AZD 2098
Potent and selective CCR4 antagonist
6542 Ivabradine hydrochloride
HCN channel blocker; inhibits If pacemaker current
6544 CID 1375606
GPR27 agonist
6545 OB-1
Stomatin-like protein-3 (STOML3) oligomerization inhibitor
6551 PAMP-12 (human, porcine)
Potent MRGPRX2 agonist
6552 PAMP-20 (human)
MRGPRX2 agonist; also non-competitive nAChR antagonist
6553 JF-NP-26
Caged Raseglurant (Cat. No. 4416)
6555 TokeOni
NIR-emission luciferin analog; ideal for deep tissue applications; orally bioavailable and brain penetrant
6558 CP 43
Potent TAOK inhibitor
6559 LY 450139
γ-secretase pseudo-inhibitor
6561 BAY 6035
Potent and selective SMYD3 inhibitor
6562 BAY 707
Potent and selective MTH1 inhibitor
6564 SGC GAK 1
High affinity cyclin G associated kinase (GAK) inhibitor
6568 Dooku 1
Reversibly blocks Yoda1 activity; does not affect constitutive Piezo1 activity
6571 Biotin-11-dUTP
Biotin-labeled dUTP
6572 Biotin-LC-NAD+
Biotinylated analog of β-NAD+; commonly used reagent in LSD1 and PARP1 assays
6573 Biotin-NAD+
Biotinylated-NAD+; substrate for ADP-ribosylation
6574 Fluorescein-NAD+
Fluorescent NAD+; substrate for ADP-ribosylation for use in PARP assays
6576 ABT 594 hydrochloride
Selective α4β2 nAChR agonist
6577 Pyridone 6
Potent pan-JAK inhibitor; induces intermediate mesoderm; cell-permeable
6578 GT 949
Potent and selective positive allosteric modulator of EAAT2
6579 BAY 826
Potent Tie2 inhibitor
6580 PKUMDL WQ 2101
Negative allosteric modulator of 3-phosphoglycerate dehydrogenase (PHGDH)
6581 PKUMDL WQ 2201
Negative allosteric modulator of 3-Phosphoglycerate dehydrogenase (PHGDH)
6583 UCLA GP130 2
gp130 agonist; brain penetrant and neuroprotectant
6584 L-Azidohomoalanine hydrochloride
Unnatural amino acid for bio-orthogonal labeling of newly synthesized proteins
6585 L-Azidonorleucine hydrochloride
Unnatural amino acid for bio-orthogonal or fluorescent labeling of newly synthesized proteins
6586 Targapremir 210
Inhibits formation of miR-210
6587 TAK 242
TLR4 signaling inhibitor
6590 Janelia Fluor® 646, Maleimide
Red dye (Reactive group: maleimide). Applications: super resolution microscopy e.g. dSTORM & STED, confocal, flow and live cell imaging
6597 SPRi 3
Potent sepiapterin reductase (SPR) inhibitor; attenuates proliferation of CD4+ T cells
6598 OD 36 hydrochloride
Potent RIP2 kinase inhibitor
6599 Yhhu 3792
Notch signaling pathway activator; enhances the self-renewal capability of NSCs; active in vivo

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