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Displaying Products by Catalog Number (4500 - 4599)

Cat. No. Product Name / Activity
4500 Cercosporamide
Potent Mnk2 inhibitor
4501 Ribavirin
Blocks eIF4E activity; antiviral guanosine analog
4502 DIM
Inhibits EGFR activation; also induces apoptosis
4503 CC 0651
Allosteric inhibitor of hCdc34
4504 Chaetocin
SUV39H1 inhibitor
4505 ICG 001
Inhibits TCF/β-catenin-mediated transcription
4506 TAME hydrochloride
Ubiquitin ligase APC/C inhibitor; promotes Cdc20 autoubiquitination
4507 ML 218 hydrochloride
CaV3.x blocker
4508 S 32212 hydrochloride
5-HT2C inverse agonist; α2-adrenoceptor antagonist
4509 STF 083010
Inhibits IRE1α endonuclease activity
4510 SHA 68
Selective Neuropeptide S receptor antagonist
4511 MMF
Activator of Nrf2 pathway; primary metabolite of DMF (Cat. No. 4512)
4512 DMF
Nrf2 pathway activator; neuroprotective
4513 Kartogenin
Potently induces chondrogenesis in MSCs
4514 JW 55
Tankyrase inhibitor
4515 2-Deoxy-D-glucose
Non-metabolizable glucose analog; hexokinase substrate
4516 UNC 926 hydrochloride
L3MBTL1 domain inhibitor
4517 NS 2028
Potent soluble guanylyl cyclase (sGC) inhibitor
4518 EPPTB
Trace amine 1 (TA1) receptor antagonist; also displays inverse agonism
4519 ML 213
KV7.2 and KV7.4 channel opener
4520 Cytarabine
Nucleoside analog; inhibits DNA replication
4521 TAS 301
Inhibitor of smooth muscle cell migration and proliferation
4522 Flufenamic acid
Calcium-activated chloride channel blocker; NSAID. Also activates TRPC6
4523 DIDS
Chloride channel blocker; TRPV1 modulator; RAD51 recombinase inhibitor
4524 EGCG
β-secretase (BACE) inhibitor; inhibits amyloid assembly
4525 Piclamilast
Potent and selective PDE4 inhibitor
4527 TC-I 15
Potent α2β1 inhibitor; displays antithrombotic activity in vivo
4528 (±)-NBI 74330
Potent and selective CXCR3 antagonist
4529 Ciliobrevin A
Hedgehog (Hh) pathway antagonist, inhibits ciliogenesis; also inhibits dynein
4530 ONO 2506
Inhibits S-100β synthesis; neuroprotective
4531 NCX 4040
NO-donating aspirin; anti-inflammatory and antitumor
4532 VUF 10166
High affinity 5-HT3 antagonist
4533 PTAC oxalate
Muscarinic receptor ligand; exhibits partial agonist and antagonist activity at different subtypes
4534 CZC 54252 hydrochloride
Potent LRRK2 inhibitor; neuroprotective
4535 Phalloidin
Promotes actin polymerization
4536 Resiquimod
Toll-like receptor 7 (TLR7) agonist
4537 NCX 466
Cyclooxygenase-inhibiting nitric oxide donor
4538 T16Ainh - A01
Ca2+-activated Cl- channel transmembrane protein 16A (TMEM16A) inhibitor
4539 (R)-(+)-Etomoxir sodium salt
Carnitine palmitoyltransferase I (CPT1) inhibitor
4540 U 104
Potent carbonic anhydrase (CA) IX and XII inhibitor
4541 SGC 0946
Highly potent and selective DOT1L inhibitor; cell permeable
4542 (+)-Fluprostenol
High affinity FP prostaglandin receptor agonist
4543 CS 2100
Selective S1P1 agonist
4544 YM 244769
Na+/Ca2+ exchange inhibitor (reverse mode); neuroprotective
4545 E 64d
Cathepsin inhibitor; interferes with autolysosomal digestion
4546 rac-CCT 250863
Potent Nek2 inhibitor
4547 ACHP
Selective IKKα and IKKβ inhibitor
4549 ML 133 hydrochloride
Kir2 channel blocker
4550 IQ 3
Selective JNK3 inhibitor
4551 Purmorphamine
Smo receptor agonist
4552 A 412997 dihydrochloride
Selective D4 agonist
4553 Azilsartan
Potent AT1 inverse agonist; antihypertensive
4554 GC 1
High affinity thyroid receptor α (TRα) and TRβ agonist; thyromimetic
4555 HI TOPK 032
Selective T-LAK-cell-originated protein kinase (TOPK) inhibitor
4556 CP 690550 citrate
Potent JAK inhibitor
4557 GTS 21 dihydrochloride
α7 nAChR partial agonist
4558 EMPA
Highly potent and selective OX2 antagonist; brain penetrant
4559 GNF 5837
Potent Trk inhibitor; inhibits TrkA, TrkB and TrkC
4561 BIBN 4096
Potent and selective CGRP antagonist
4562 Topotecan hydrochloride
DNA topoisomerase I inhibitor; Camptothecin (Cat. No. 1100) analog
4564 JTV 519 fumarate
Ryanodine receptor (RyR) inhibitor
4565 ML 228
HIF pathway activator
4566 NSC 687852
Inhibitor of UCHL5 and USP14
4567 CCG 50014
Potent and selective inhibitor of regulator of G-protein signaling 4 (RGS4) protein
4568 CPYPP
DOCK2-Rac1 interaction inhibitor
4569 PS 1145 dihydrochloride
Selective IKK inhibitor; orally active
4570 ML 161
Inhibits PAR1-mediated platelet activation
4571 A 867744
Positive allosteric modulator of α7 nAChRs
4572 TC-E 5005
Potent and selective PDE10A inhibitor
4575 TC HSD 21
Potent and selective 17β-hydroxysteroid dehydrogenase type 3 inhibitor
Fluorescent ligand for α4β1 (VLA-4)
4579 Pentobarbital sodium salt
Enhances GABAergic activity
4580 Atiprimod dihydrochloride
JAK2 inhibitor
4581 Grifolic acid
Selective partial FFA4 (GPR120) agonist
4582 MLR 1023
Selective allosteric activator of Lyn kinase
4583 Digoxin
Na+/K+ ATPase inhibitor
4584 SNS 314 mesylate
Potent pan-Aurora kinase inhibitor
4585 MRT 10
Smoothened (Smo) antagonist
4586 ML 3403
p38 inhibitor
4588 8MDP
Potent equilibrative nucleoside transporter (ENT) inhibitor
4590 Honokiol
Blocks NF-κB activation; also anti-inflammatory and antioxidant
4591 Deltorphin I
Potent δ agonist
4592 R8-T198wt
Pim-1 kinase inhibitor
4593 GSK J1
Potent JMJD3/UTX inhibitor
4594 GSK J4
Histone KDM inhibitor; cell permeable
4596 IT1t dihydrochloride
Potent CXCR4 antagonist
4597 NS 8593 hydrochloride
Selective negative modulator of KCa2 (SK) channels; inhibits SK currents
4598 PHT 427
Dual Akt and PDK1 inhibitor; antitumor
4599 3,5-DHBA
Selective HCA1 agonist

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