All Products

Displaying Products by Catalog Number (4500 - 4599)

Cat. No. Product Name / Activity
4500 Cercosporamide
Potent Mnk2 inhibitor
4501 Ribavirin
Blocks eIF4E activity; antiviral guanosine analog
4504 Chaetocin
SUV39H1 inhibitor
4505 ICG 001
Inhibits TCF/β-catenin-mediated transcription
4507 ML 218 hydrochloride
CaV3.x blocker
4509 STF 083010
Inhibits IRE1α endonuclease activity
4510 SHA 68
Selective Neuropeptide S receptor antagonist
4513 Kartogenin
Potently induces chondrogenesis in MSCs
4515 2-Deoxy-D-glucose
Non-metabolizable glucose analog; inhibits glucose metabolism
4517 NS 2028
Potent soluble guanylyl cyclase (sGC) inhibitor
4518 EPPTB
Trace amine 1 (TA1) receptor antagonist; also displays inverse agonism
4519 ML 213
KV7.2 and KV7.4 channel opener
4520 Cytarabine
Nucleoside analog; inhibits DNA replication
4522 Flufenamic acid
Calcium-activated chloride channel blocker; NSAID. Also activates TRPC6
4523 DIDS
Chloride channel blocker; TRPV1 modulator; RAD51 recombinase inhibitor
4524 EGCG
β-secretase (BACE) inhibitor; inhibits amyloid assembly
4525 Piclamilast
Potent and selective PDE4 inhibitor
4527 TC-I 15
Potent α2β1 inhibitor; displays antithrombotic activity in vivo
4528 (±)-NBI 74330
Potent and selective CXCR3 antagonist
4529 Ciliobrevin A
Hedgehog (Hh) pathway antagonist, inhibits ciliogenesis; also inhibits dynein
4530 ONO 2506
Inhibits S-100β synthesis; neuroprotective
4535 Phalloidin
Promotes actin polymerization
4536 Resiquimod
Toll-like receptor 7 (TLR7) agonist
4539 (R)-(+)-Etomoxir sodium salt
Carnitine palmitoyltransferase I (CPT1) inhibitor
4541 SGC 0946
Highly potent and selective DOT1L inhibitor; cell permeable
4543 CS 2100
Selective S1P1 agonist
4544 YM 244769
Na+/Ca2+ exchange inhibitor (reverse mode); neuroprotective
4545 E 64d
Cathepsin inhibitor; interferes with autolysosomal digestion
4546 rac-CCT 250863
Potent Nek2 inhibitor
4547 ACHP
Selective IKKα and IKKβ inhibitor
4549 ML 133 hydrochloride
Kir2 channel blocker
4551 Purmorphamine
Smo receptor agonist
4552 A 412997 dihydrochloride
Selective D4 agonist
4554 GC 1
High affinity thyroid receptor α (TRα) and TRβ agonist; thyromimetic
4556 CP 690550 citrate
Potent JAK inhibitor
4558 EMPA
Highly potent and selective OX2 antagonist; brain penetrant
4559 GNF 5837
Potent Trk inhibitor; inhibits TrkA, TrkB and TrkC
4561 BIBN 4096
Potent and selective CGRP antagonist
4562 Topotecan hydrochloride
DNA topoisomerase I inhibitor; Camptothecin (Cat. No. 1100) analog
4564 JTV 519 fumarate
Ryanodine receptor (RyR) inhibitor
4568 CPYPP
DOCK2-Rac1 interaction inhibitor
4571 A 867744
Positive allosteric modulator of α7 nAChRs
Fluorescent ligand for α4β1 (VLA-4)
4581 Grifolic acid
Selective partial FFA4 (GPR120) agonist
4582 MLR 1023
Selective allosteric activator of Lyn kinase
4583 Digoxin
Na+/K+ ATPase inhibitor
4588 8MDP
Potent equilibrative nucleoside transporter (ENT) inhibitor
4590 Honokiol
Blocks NF-κB activation; also anti-inflammatory and antioxidant
4593 GSK J1
Potent JMJD3/UTX inhibitor
4594 GSK J4
Histone KDM inhibitor; cell permeable
4596 IT1t dihydrochloride
Potent CXCR4 antagonist
4597 NS 8593 hydrochloride
Selective negative modulator of KCa2 (SK) channels; inhibits SK currents
4599 3,5-DHBA
Selective HCA1 agonist

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