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Displaying Products by Catalog Number (6900 - 6999)

Cat. No. Product Name / Activity
6900 NNMTi
Nicotinamide N-methyltransferase (NNMT) inhibitor; promotes myoblast differentiation
6902 Dapansutrile
NLRP3 inflammasome inhibitor; disrupts inflammasome formation
6903 DPTIP
Potent and selective N-SMase2 inhibitor; brain penetrant
6904 Idasanutlin
Potent MDM2 inhibitor; inhibits MDM2-p53 interaction
6905 Ceritinib
Highly potent ALK inhibitor; also potently inhibits IR, IGF1R, STK22D and FLT3
6907 VH 032 amide-PEG2-amine
VHL ligand with PEG linker and terminal amine for onward chemistry
6908 TR 14035
Potent integrin α4β7 and α4β1 (VLA-4) antagonist; orally bioavailable
6909 VH 032 phenol-alkylC4-amine
VHL ligand with alkyl linker and terminal amine for onward chemistry
6910 VH 032 phenol-alkylC6-amine
VHL ligand with alkyl linker and terminal amine for onward chemistry
6911 VH 032, phenol
Hydroxyl functionalized VHL ligand
6912 dTAG-7
First generation Degrader for mutant FKBP12F36V fusion proteins; useful alternative to genetic methods for target validation
6913 Thalidomide 4'-oxyacetamide-alkylC1-PEG3-alkylC3-amine
Cereblon ligand with alkyl-PEG-alkyl linker and terminal amine for onward chemistry
6914 dTAGV-1
Potent and selective degrader of mutant FKBP12F36V fusion proteins
6915 dTAGV-1-NEG
Negative control for dTAGV-1 (Cat. No. 6914)
6916 dTAG-13-NEG
Negative control for dTAG-13 (Cat. No. 6605)
6917 Thalidomide 4'-ether-alkylC4-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
6921 BSJ-03-123
Selective Cdk6 Degrader (PROTAC®)
6923 AMZ 30
Potent, selective and irreversible protein phosphatase methylesterase-1 (PME-1) inhibitor
6927 Glucagon (Human, Porcine)
Endogenous glucagon receptor agonist
6928 VU 6001966
Potent and selective negative allosteric modulator of mGlu2 receptors
6930 Amphotericin B
Forms monovalent ion channels in lipid bilyers; antifungal
6931 AF 64394
Potent and selective GPR3 inverse agonist
6935 GSK J5 HCl
Inactive isomer of GSK J4 (Cat. No. 4594); cell permeable
6936 VZ 185
Potent and selective BRD7/9 Degrader (PROTAC®)
6937 BSJ-04-132
Selective Cdk4 Degrader (PROTAC®)
6938 BSJ-03-204
Selective Cdk4/6 Degrader (PROTAC®
6939 cis-VZ 185
Negative control for VZ 185 (Cat. No. 6936)
6940 BTD
Selective TRPC5 activator
6941 Pyr 10
Selective TRPC3 inhibitor
6943 dBRD9-A
Potent BRD9 Degrader (PROTAC®)
6944 Pomalidomide 4'-alkylC8-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
6945 dBET6
Potent and selective (+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo
6946 Thalidomide 4'-oxyacetamide-alkylC8-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
6948 CRBN-6-5-5-VHL
Potent and selective cereblon Degrader (PROTAC®); cell-permeable
6949 Thalidomide 4'-oxyacetamide-alkylC2-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
6950 Thalidomide 4'-ether-PEG3-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6951 Thalidomide 4'-ether-PEG5-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6952 VH 101, phenol
Hydroxyl functionalized VHL ligand
6954 L-Buthionine sulfoximine
Irreversible γ-glutamylcysteine synthetase (γ-GCS) inhibitor; induces ferroptosis
6955 Ceapin A7
Selective inhibitor of ATF6α; sensitizes cells to ER stress
6956 Galunisertib
ALK4 and ALK5 (TGFβRI) inhibitor
6960 ABT 199
Selective, high affinity Bcl-2 inhibitor; orally bioavailable
6961 FzM1.8
Frizzled 4 allosteric agonist; exhibits biased signaling; preserves stemness
6962 JBJ-03-142-02
Highly potent EGFR and ErbB2 inhibitor; inhibts wild type and mutated receptors
6963 Pomalidomide 4'-PEG4-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6964 LY 2119620
Positive allosteric modulator of M2 and M4 receptors
6965 CGI 1746
Potent, reversible BTK inhibitor
6966 Thalidomide 4'-oxyacetamide-PEG1-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6967 Thalidomide 4'-oxyacetamide-PEG2-amine
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6968 Thalidomide 4'-oxyacetamide-alkylC6-amine
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
6969 cis VH 032, amine dihydrochloride
Negative control for VH 032, amine (Cat. No. 6462)
6970 aTAG 2139
Degrader of MTH1 fusion proteins for use within the aTAG system
6971 aTAG 4531
Degrader of MTH1 fusion proteins for use within the aTAG system
6972 A 1899
Potent K2P3.1 (TASK-1) and K2P9.1 (TASK-3) blocker
6973 NS 3728
VRAC blocker
6975 Teniposide
DNA topoisomerase II inhibitor; viral transduction enhancer
6977 Bobcat339
Ten-eleven translocation methylcytosine dioxygenase (TET) inhibitor
6978 AZD 5363
Potent pan-AKT inhibitor
6979 SEN 177
Potent glutaminyl cyclase inhibitor; disrupts binding of SIRP-α to CD47
6981 TL 0259
Selective and highly potent Fgr and Lyn kinase inhibitor; orally bioavailable
6982 Cyclosporin H
Enhances lentiviral transduction
6984 KIN001-266
Potent and selective Tpl2 (MAP3K8) inhibitor
6985 VH 032 amide-alkylC5-amine
VHL ligand with alkyl linker and terminal amine for onward chemistry
6986 EG 00229 trifluoroacetate
Neuropilin 1 (NRP1) receptor antagonist; inhibits VEGFA binding to NRP1
6990 SET 2
Selective TRPV2 antagonist
6998 SHIN 1
Potent SHMT inhibitor

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