All Products

Displaying Products by Catalog Number (4300 - 4399)

Cat. No. Product Name / Activity
4300 TC 14012
CXCR4 antagonist; ACKR3 (CXCR7) agonist
4301 TC-DAPK 6
Potent and selective inhibitor of DAPK1
4302 Perindopril erbumine
Angiotensin-converting enzyme (ACE) inhibitor
4303 PPQ 102
Potent, voltage-independent CFTR chloride channel inhibitor
4305 ICA 069673
KV7.2/KV7.3 channel opener
4306 INCB 3284 dimesylate
Selective CCR2 antagonist
4307 YC 1
Soluble guanylyl cyclase (sGC) activator; induces G1 cell cycle arrest
4308 Rasagiline mesylate
Selective and irreversible MAO-B inhibitor
4309 TPEN
Cell-permeable Zn2+ chelator; also inhibits RNA binding protein Lin28
4310 ML 7 hydrochloride
Selective inhibitor of myosin light chain kinase
4311 GW 542573X
Selective KCa2.1 (SK) channel activator
4312 Nigericin sodium salt
Selective K+ ionophore
4314 SB 268262
Selective non-peptide CGRP antagonist
4315 NGD 98-2 hydrochloride
High affinity CRF1 antagonist
4316 Bropirimine
Immunomodulatory and antitumor compound
4317 JNJ 10397049
Selective OX2 antagonist
4318 BX 795
PDPK1 (PDK1) inhibitor
4319 A 784168
Potent and selective TRPV1 antagonist
4322 JH 295
Irreversible Nek2 inhibitor
4323 VU 0360172 hydrochloride
Positive allosteric modulator of mGlu5 receptors
4324 KC7F2
HIF-1α inhibitor; down-regulates HIF-1α protein synthesis
4325 Phosphocreatine disodium salt
Phosphate reservoir
4326 PhiKan 083
p53 stabilizing agent
4327 JW 480
Potent and selective inhibitor of serine hydrolase KIAA1363 (AADACL1)
4330 AMG 21629
Potent and selective TRPV1 antagonist
4333 PSB 1114
Potent, selective P2Y2 agonist
4334 PSB 0777 ammonium salt
Potent adenosine A2A agonist
4335 AR-M 1000390 hydrochloride
Low-internalizing δ agonist
4336 TG 003
Potent inhibitor of Clk-family kinases; also inhibits DYRK1A/B
4337 ST 1936 oxalate
Selective, high affinity 5-HT6 agonist
4338 NSC 33994
JAK2 inhibitor
4339 Tertiapin LQ
Selective Kir1.1 blocker; derivative of tertiapin-Q (Cat. No. 1316)
4341 A 582941
α7 nAChR partial agonist
4342 UNC 0646
Potent and selective G9a and GLP inhibitor
4343 UNC 0638
Selective G9a and GLP inhibitor
4344 FH 535
Inhibitor of Wnt/β-catenin signaling
4345 TC-C 14G
High affinity and potent CB1 inverse agonist
4346 Ro 67-7476
Positive allosteric modulator of mGlu1 receptors
4347 Ro 67-4853
Positive allosteric modulator of group I mGlu receptors
4348 Ro 01-6128
Positive allosteric modulator of mGlu1 receptors
4349 Olanzapine
5-HT2A antagonist; also D2 antagonist; atypical antipsychotic
4350 Axitinib
Potent VEGFR-1, -2 and -3 inhibitor
4351 JHW 007 hydrochloride
High affinity dopamine uptake inhibitor
4352 Talsupram hydrochloride
Selective inhibitor of noradrenalin transporters
4353 TC-G 24
Potent and selective GSK-3β inhibitor
4354 ML 130
Inhibits NOD1-induced NF-κB activation
4355 TC-F 2
Potent, reversible and selective FAAH inhibitor
4357 Bicifadine hydrochloride
Noradrenalin, 5-HT and dopamine re-uptake inhibitor
4358 Dapoxetine hydrochloride
Selective serotonin reuptake inhibitor (SSRI)
4359 Lomeguatrib
MGMT inhibitor
4361 Bosutinib
Dual Src-Abl inhibitor; antiproliferative
4363 TC-SP 14
Potent S1P1 receptor agonist
4365 TC-MCH 7c
Selective melanin-concentrating hormone receptor 1 (MCH1R) antagonist
4366 SAG
Potent Smoothened receptor agonist; activates the Hedgehog signaling pathway
4367 Psora 4
Potent KV1.3 channel blocker
4368 Crizotinib
Potent c-MET/ALK inhibitor
4370 TC-N 22A
Potent and selective positive allosteric modulator of mGlu4 receptors
4371 VU 0364439
Positive allosteric modulator of mGlu4 receptors
4372 BC 11 hydrobromide
Selective urokinase (uPA) inhibitor
4373 CMPDA
Positive allosteric modulator of GluA2 receptors
4374 BIMU 8
Potent 5-HT4 agonist
4375 SMER 3
Selective inhibitor of E3 ubiquitin ligase
4376 5-OMe-UDP trisodium salt
Potent P2Y6 agonist
4379 (S)-(+)-Ketamine hydrochloride
NMDA receptor antagonist; enantiomer of ketamine hydrochloride (Cat. No. 3131); neuroprotective
4380 WAY 100635 maleate
Potent 5-HT1A antagonist; also D4 agonist
4381 VU 0285683
Negative allosteric modulator of mGlu5 receptors
4382 Letrozole
Potent, reversible non-steroidal aromatase inhibitor
4385 Donepezil hydrochloride
Potent AChE inhibitor
4386 TC-P 262
Selective P2X3 and P2X2/3 antagonist
4387 Calhex 231 hydrochloride
Negative allosteric modulator of calcium-sensing receptor (CaSR)
4388 MNI 137
Selective negative allosteric modulator of group II mGlu receptors
4390 Thiamet G
Potent O-GlcNAcase inhibitor
4391 Ro 51
Potent P2X3 and P2X2/3 antagonist
4392 680C91
Potent and selective tryptophan 2,3-dioxygenase (TDO) inhibitor
4393 L-Kynurenine
Tryptophan catabolite; endogenous aryl hydrocarbon receptor ligand
4395 Moclobemide
Reversible MAO-A inhibitor
4396 Piperlongumine
Induces apoptosis; increases p53 and ROS levels in cancer cells
4398 SC 66
Allosteric Akt inhibitor
4399 GNF 2
Selective allosteric inhibitor of Bcr-Abl tyrosine kinase activity

Tocris Products Alphabetically by Name