All Products

Displaying Products by Catalog Number (6000 - 6099)

Cat. No. Product Name / Activity
6000 TP 472
Potent BRD9/7 inhibitor
6001 ZQ 16
Selective GPR84 agonist
6002 Trolox
Antifade reagent; antioxidant vitamin E derivative; cell permeable and water soluble
6004 PF 06281355
Selective myeloperoxidase (MPO) inhibitor
6005 PF 3758309 dihydrochloride
Potent PAK4 inhibitor; orally available
6007 INCB 024360-analog
Potent indoleamine 2,3-dioxygenase (IDO) inhibitor
6008 TP 064
Potent and selective PRMT 4 inhibitor
6009 B I09
IRE1 endonuclease inhibitor; cell permeable
6010 BRD 4354
HDAC5 and HDAC9 inhibitor
6011 FSL 1
TLR2/6 agonist (also a putative TLR10 ligand)
6012 OXSI 2
Potent Syk kinase inhibitor; also inhibits assembly of NLRP3 inflammasomes
6013 TAPI 2
ADAM-17 (TACE) and MMP inhibitor
6014 Org 48762-0
Selective p38α/β inhibitor; orally bioavailable
6015 RAF 265
Raf kinase and VEGFR-2 inhibitor
6016 IN 1130
Potent and selective inhibitor of TGF-βRI
6017 THPN
Nur77 agonist; induces autophagy in melanoma cell lines
6018 Nicotinamide Riboside
NAD+ precursor; substrate for nicotinamide riboside kinases
6019 Diprotin A
Dipeptidyl peptidase IV (DPP-IV) inhibitor
6020 URB 602
Non-competitive MAGL inhibitor
6024 PF 04671536 hydrochloride
Potent and selective PDE8B/8A inhibitor
6025 (S)-Crizotinib
MTH1 inhibitor
6029 FRAX 597
Potent group I PAK inhibitor
6030 Amylin (rat)
Potent endogenous peptide agonist for amylin, calcitonin, CGRP and adrenomedullin receptors
6031 Calcitonin (human)
Endogenous calcitonin agonist; inhibits bone resorption
6033 (R)-MG 132
Potent 20S proteasome inhibitor
6034 AM 2394
Potent glucokinase activator; orally bioavailable
6035 (S)-C33
Potent PDE9 inhibitor
6036 STK16-IN-1
Serine/threonine protein kinase 16 (STK16) inhibitor; also inhibits PI 3Kδ, PI 3Kγ and mTOR kinases
6037 LM22B 10
TrkB and TrkC agonist; brain penetrant
6038 SR 10067
Selective Rev-Erbα/β agonist; anxiolytic
6040 BRD 9757
Potent and selective HDAC6 inhibitor
6043 AMBMP hydrochloride
Wnt canonical signaling activator; also tubulin polymerization inhibitor
6045 NITD 008
Antiflaviviral; active against Zika, Dengue and Hepatitis C viruses
6046 Naloxone fluorescein acetate
Fluorescent opioid antagonist; fluorescent-derivative of naloxone (Cat. No. 0599)
6047 BOP
Dual α9β1/α4β1 integrin inhibitor; preferentially mobilizes HSCs
6048 R-BC154
High affinity fluorescent α4β1/α9β1 inhibitor; mobilizes HSCs
6049 PF 04937319
Glucokinase partial activator
6051 G 5555
High affinity group I PAK inhibitor
6052 BAY 58-2667 hydrochloride
Potent soluble guanylyl cyclase (sGC) activator
6053 LDN 193189 dihydrochloride
Potent and selective ALK2 and ALK3 inhibitor; inhibits BMP4 signaling; promotes neural induction of hPSCs
6055 SPT Imidazopyridine 1
Potent serine palmitoyl transferase inhibitor
6056 GSK 1363089
Potent inhibitor of MET, VEGFR2, Ron and AXL
6058 ATN 161
α5β1 integrin receptor antagonist
6060 AZD 2461
Potent PARP inhibitor; orally bioavailable
6061 XMD 8-87
Potent Ack1/TNK2 inhibitor
6063 CCF 642
Protein disulfide isomerase (PDI) inhibitor
6065 2-NBDG
Fluorescent glucose uptake indicator
6066 OAC-2
Oct4 activator; enhances iPSC reprogramming efficiency
6067 M 30 dihydrochloride
Potent and non-selective MAO inhibitor; also an iron chelator and antioxidant
6068 Lin28 1632
RNA binding protein Lin28 inhibitor; promotes mESC differentiation; also bromodomain inhibitor
6069 BMS 605541
Potent VEGFR-2 inhibitor
6070 Pladienolide B
mRNA splicing inhibitor; antitumor
6071 CZC 25146
Potent LRRK2 inhibitor
6073 P21d hydrochloride
Potent and selective Brk inhibitor
6075 Nutlin 3a
MDM2 antagonist; active enantiomer of Nutlin-3 (Cat. No. 3984)
6076 Ani 9
Potent and selective TMEM16A (Anoctamin-1; ANO1) blocker
6078 BPTU
P2Y1 allosteric antagonist
6079 TC KHNS 11
Potent and selective PI 3-kinase δ inhibitor; orally bioavailable
6082 AMG 837 hemicalcium salt
Potent FFA1 (GPR40) partial agonist
6083 PSB 12379
Ecto-5'-nucleotidase (CD73) inhibitor
6084 ASP 9521
Potent 17β-hydroxysteroid dehydrogenase type 5 inhibitor;orally bioavailable
6085 AZD 1283
High affinity P2Y12 antagonist
6086 AMP PNP
Kir6 blocker; non-hydrolyzable AMP analog
6087 Perifosine
PKB/Akt inhibitor; also modulates Kv2.1 current
6088 SB 3CT
High affinity and selective MMP2 inhibitor
6089 Nexinhib20
Rab27 inhibitor; inhibits neutrophil exocytosis; active in vivo
6090 Spexin
Potent GAL2/3 agonist; exhibits anxiolytic effects in vivo
6092 TDZD 8
Selective non-ATP competitive inhibitor of GSK 3β
6094 2R,6R-Hydroxynorketamine hydrochloride
Enhances AMPA currents; decreases D-serine (a NMDA co-agonist); lacks ketamine-related side effects
6095 2S,6S-Hydroxynorketamine hydrochloride
Decreases D-serine (a NMDA co-agonist); antidepressant
6098 Lalistat 1
Potent and selective LAL inhibitor
6099 Lalistat 2
Selective LAL inhibitor

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