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Displaying Products by Catalog Number (0400 - 0499)

Cat. No. Product Name / Activity
0405 β-CCB
Benzodiazepine inverse agonist; putative endogenous ligand
0414 AG 490
EGFR-kinase inhibitor. Also JAK2, JAK3 inhibitor
0415 Ro 20-1724
PDE4 inhibitor
0416 YS-035 hydrochloride
Inhibits K+ outward/pacemaker current
0417 (RS)-Baclofen
Selective GABAB agonist
0421 GBR 12909 dihydrochloride
Selective DA uptake inhibitor; also σ ligand
0424 Benzoquinonium dibromide
nAChR antagonist
0425 UK 14,304
α2 agonist
0427 Bromocriptine mesylate
D2-like agonist (D2>D3>D4)
0431 ML 9 hydrochloride
Myosin light chain kinase inhibitor
0433 SC-9
Protein kinase C activator
0435 Cimaterol
β agonist
0439 DPCPX
Selective A1 antagonist
0440 m-Chlorophenylbiguanide hydrochloride
Potent and selective 5-HT3 agonist
0442 4-Chlorophenylguanidine hydrochloride
Urokinase inhibitor
0443 6-Chloromelatonin
Melatonin agonist
0444 Clozapine
Dopamine antagonist with some D4 selectivity; also 5-HT2A/2C antagonist
0448 Calpeptin
Calpain and cathepsin L inhibitor
0452 CCCP
Oxidative phosphorylation uncoupler
0453 FCCP
Oxidative phosphorylation uncoupler
0455 (S)-(-)-Carbidopa
Aromatic L-amino acid decarboxylase inhibitor
0456 Chlormezanone
Positive allosteric modulator of benzodiazepine site
0458 5-Carboxamidotryptamine maleate
5-HT1 agonist; also has high affinity for 5-ht5a and 5-HT7
0460 Cinanserin hydrochloride
Selective 5-HT2 antagonist; also 3C-like proteinase inhibitor
0462 (E)-Capsaicin
TRPV agonist
0464 Capsazepine
TRPV antagonist; also activator of ENaCδ
0468 N1,N11-Diethylnorspermine tetrahydrochloride
Spermine and spermidine acetyltransferase potentiator
0471 (+)-U-50488 hydrochloride
Selective κ agonist; less active enantiomer of (±)-U-50488 (Cat. No. 0495)
0475 Dihydroergotamine mesylate
α partial agonist; also D2-like partial agonist and 5-HT antagonist
0477 (±)-Decanoylcarnitine chloride
Intermediate in lipid metabolism
0478 Flurofamide
Urease inhibitor
0481 Dilazep dihydrochloride
Adenosine uptake inhibitor
0482 4-DAMP
Muscarinic M3 antagonist
0483 OR-486
COMT inhibitor
0484 Dioctanoylglycol
Diacylglycerol kinase inhibitor
0495 (±)-U-50488 hydrochloride
Selective κ agonist
0496 (-)-U-50488 hydrochloride
Selective κ agonist; more active enantiomer of (±)-U-50488 (Cat. No. 0495)

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