All Products

Displaying Products by Catalog Number (5800 - 5899)

Cat. No. Product Name / Activity
5802 A37
ALDH1A1 inhibitor
5803 MP A08
Selective ATP competitive SphK1 and 2 inhibitor; cell permeable
5804 Chaetoglobosin A
Antibiotic; selectively induces apoptosis of CLL cells
5807 M 084 hydrochloride
TRPC4 and TRPC5 inhibitor; antidepressant and anxiolytic
5813 NSC 668036
Wnt signaling inhibitor; binds the PDZ domain of the Dishevelled (Dvl) protein
5814 GoSlo SR 5-69
KCa1.1 (BK) channel activator
5815 SCH 336
Highly potent and selective CB2 inverse agonist
5818 NVP BSK 805
Potent JAK2 inhibitor; orally bioavailable
5819 Bexarotene
Potent and selective RXR agonist
5821 C-DIM 12
Nurr1 activator; inhibits NF-κB-dependent gene expression
5826 LEI 101 hydrochloride
Potent and selective CB2 partial agonist; orally biovailable
5828 Ambrisentan
Selective ETA antagonist
5831 SAR 7334
Potent TRPC6 inhibitor
5832 TGX 221
Potent and selective PI 3-kinase β inhibitor
5833 Ex 26
Potent and selective S1P1 receptor antagonist
5834 LTURM 34
Potent DNA-PK inhibitor
5835 LTURM 36
PI 3-kinase δ inhibitor
5836 CBR 5884
Phosphoglycerate dehydrogenase (PHGDH) inhibitor
5837 [Pro3]-GIP (Rat)
High affinity rat GIP partial agonist
5838 [Pro3]-GIP (Mouse)
GIP receptor antagonist
5842 MK 386
Potent, selective human type 1 5α-reductase inhibitor
5843 AX 15836
Potent and selective ERK5 inhibitor
5844 JZP 430
Potent and irreversible α/β-hydrolase domain 6 (ABHD6) inhibitor
5845 JX 06
Potent and selective pyruvate dehydrogenase kinase (PDK) 1/2/3 inhibitor
5846 IT 901
NF-κB c-Rel subunit inhibitor
5847 ZLD 1039
Potent and selective EZH2 inhibitor; orally bioavailable
5850 HM 50316
High affinity FABP4 inhibitor
5851 JZP 361
Potent and selective reversible MAGL inhibitor
5853 JNJ DGAT2-A
DGAT2 inhibitor
5854 SR 9238
Potent and selective LXR inverse agonist
5855 SR 9009
Rev-Erbα/β agonist
5856 Ritonavir
HIV-1 and HIV-2 protease inhibitor
5857 Neuropeptide S (Mouse)
Endogenous Neuropeptide S receptor agonist
5860 7rh
Potent and selective DDR1 inhibitor; orally bioavailable
5861 ARN 726
Potent N-acylethanolamine acid amidase (NAAA) inhibitor; NAAA activity-based protein profiling (ABPP) probe
5862 ARN 14686
Potent N-acylethanolamine acid amidase inhibitor; NAAA activity-based protein profiling (ABPP) probe
5863 PF 04620110
Potent and selective DGAT-1 inhibitor; orally bioavailable
5864 Tolcapone
COMT inhibitor; also inhibits transthyretin aggregation
5865 KLH 45
Potent DDHD2 inhibitor
5866 PH 797804
Potent and selective p38α/β inhibitor
5867 Ceefourin 1
Selective MRP4 inhibitor
5868 SR 0987
T cell-specific RORγ (RORγt) agonist
5869 CDN 1163
SERCA2 allosteric activator
5870 Cilengitide
Potent and selective inhibitor of integrins αvβ3 and αvβ5
5871 pCPA methyl ester hydrochloride
Tryptophan hydroxylase inhibitor
5872 AZ 10397767
Potent CXCR2 antagonist
5875 MES sodium salt
Buffering agent
5885 HEPPS
Used as a buffering agent
5887 MES, free acid
Commonly used buffer
5891 TES, free acid
Buffering agent; pKa at physiolgical pH (7.4) at 25°C

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