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Displaying Products by Catalog Number (2100 - 2199)

Cat. No. Product Name / Activity
2132 Amisulpride
Selective D2 and D3 antagonist; atypical antipsychotic
2133 α-Bungarotoxin
Selective α7 nAChR antagonist
2134 Salvinorin A
Highly potent and selective κ agonist
2137 2,3-DCPE hydrochloride
Selectively induces cancer cell apoptosis
2138 Xenin 8
Neurotensin-like peptide; potentiates insulin and glucagon secretion
2139 Leelamine hydrochloride
CB1 agonist
2141 Paroxetine maleate
Highly potent and selective 5-HT uptake inhibitor
2142 [Ala11,D-Leu15]-Orexin B
Potent and selective OX2 agonist
2143 SCS
Potent GABAA antagonist; β1-subunit selective
2144 R18
Inhibitor of 14.3.3 proteins
2146 MRS 2578
Selective P2Y6 antagonist
2147 Nicorandil
Kir6 (KATP) channel opener and NO donor
2148 (±)-McN 5652
Potent, orally active 5-HT uptake inhibitor; also inhibits noradrenalin and dopamine uptake in vitro
2150 nTZDpa
Potent, selective PPARγ partial agonist
2151 API-2
Selective inhibitor of Akt/PKB signaling. Antitumor and antiviral
2152 NSC 625987
Cdk4 inhibitor
2154 ZD 2079
β3-adrenoceptor agonist
2155 NTNCB hydrochloride
Potent and selective non-peptidic NPY Y5 antagonist
2156 Embelin
Inhibitor of X-linked inhibitor of apoptosis (XIAP); cell-permeable and antitumor
2157 MRS 2365
Highly potent and selective P2Y1 agonist
2158 MRS 2279
Selective, high affinity P2Y1 antagonist
2159 MRS 2500 tetraammonium salt
Highly potent and selective P2Y1 antagonist
2160 Bax channel blocker
Allosteric inhibitor of Bax channel activation
2161 NSC 23766
Selective inhibitor of Rac1-GEF interaction; antioncogenic
2162 INCA-6
Inhibitor of calcineurin-substrate association
2163 Z-VAD-FMK
Cell-permeable, irreversible caspase inhibitor
2166 Z-DEVD-FMK
Cell-permeable, irreversible caspase-3 inhibitor
2168 Z-DQMD-FMK
Caspase-3 inhibitor
2173 WAY 629 hydrochloride
Selective 5-HT2C agonist
2174 Hispidulin
Partial positive allosteric modulator at the benzodiazepine site
2175 Tetrabenazine
Potent inhibitor of vesicular monoamine transport
2176 BVT 948
Non-competitive protein tyrosine phosphatase inhibitor
2181 Vanilloid TRPV1 Receptor Tocriset™
Selection of 5 vanilloid TRPV1 receptor ligands (Cat. Nos. 0462, 0934, 1137, 0464 and 1615)
2183 ZK 164015
Potent estrogen receptor antagonist
2184 SN-6
Selective Na+/Ca2+ exchange inhibitor (reverse mode)
2185 NSC 146109 hydrochloride
Cell-permeable, genotype-selective antitumor agent; activates p53-dependent transcription
2186 CMPD-1
Selective inhibitor of p38α-mediated MK2a phosphorylation; also tubulin polymerization inhibitor
2187 NS 3763
GluK1 selective and non-competitive kainate antagonist
2188 Ro 0437626
Selective P2X1 antagonist
2190 SR 27897
Potent and selective CCK1 antagonist
2191 S-Trityl-L-cysteine
Potent, selective inhibitor of mitotic kinesin Eg5
2192 4-HQN
PARP inhibitor
2193 Carmoxirole hydrochloride
Selective, peripherally acting D2-like agonist
2194 R 59-022
Diacylglycerol kinase inhibitor; increases PKC activity
2195 Eliprodil
Non-competitive and GluN2B-selective NMDA antagonist
2196 3-MATIDA
Potent and selective mGlu1 antagonist
2197 L-755,507
Very potent and selective β3 partial agonist
2198 Mibefradil dihydrochloride
CaV3.x blocker
2199 CGP 71683 hydrochloride
Highly selective and potent non-peptide NPY Y5 receptor antagonist

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