All Products

Displaying Products by Catalog Number (4900 - 4999)

Cat. No. Product Name / Activity
4901 Optovin
Reversible photoactive TRPA1 activator
4902 NSC 405020
Histone deacetylase inhibitor
4903 NU 9056
Inhibitor of KAT5 (Tip60)
4904 UNC 1999
Potent and selective EZH2/EZH1 inhibitor
4905 UNC 2400
Negative control of UNC 1999 (Cat. No. 4904)
4906 JW 642
MAGL inhibitor
4907 SN 2
Selective TRPML3 channel activator
4908 GNF 5
Selective allosteric inhibitor of Bcr-Abl; analog of GNF 2 (Cat. No. 4399)
4911 GaTx2
High affinity, selective ClC-2 blocker; inhibits slow-gating
4912 GsMTx4
TRPC1 and TRPC6 blocker; inhibits mechanosensitive ion channels
4913 Jingzhaotoxin III
Selective NaV1.5 channel blocker
4914 Phrixotoxin 3
Potent blocker of NaV1.2, NaV1.3 and NaV1.5 channels
4916 PF 04885614
Potent and selective NaV1.8 channel blocker; active in vivo
4917 M 25
Potent Smoothened (Smo) receptor antagonist
4918 GSA 10
Smo receptor agonist
4919 PG 106
Selective MC3 receptor antagonist
4920 Methoxy-X04
Fluorescent amyloid β detector; brain penetrant
4921 Leukadherin 1
Allosteric activator of CD11b/CD18
4923 Shz 1
Activator of early cardiac genes in pluripotent stem cells; induces differentiation in M-PBMCs
4924 CEP 1347
Inhibitor of JNK signaling
4926 UPF 648
Potent kynurenine 3-monooxygenase (KMO) inhibitor
4927 AS 1892802
Potent ROCK inhibitor; orally bioavailable
4928 OXF BD 02
Selective BRD4(1) inhibitor
4930 UNC 2399
Biotinylated UNC 1999 (Cat.No. 4904)
4934 MA 2029
Potent and selective, competitive motilin receptor antagonist; orally active
4935 Sulfasalazine
Inhibitor of NF-κB activation; also inhibits SXC and folate transporter 1
4936 Clozapine N-oxide
Activator of muscarinic DREADDs
4941 PKI 166 hydrochloride
Potent EGFR-kinase inhibitor
4942 Pitavastatin calcium
HMG-CoA reductase inhibitor
4943 Sulfidefluor 7 AM
H2S fluorescent probe
4944 Peroxy Orange 1
Fluorescent hydrogen peroxide indicator
4945 ML 347
Potent and selective ALK1 and ALK2 inhibitor
4946 AIM 100
Potent and selective Ack1 (TNK2) inhibitor
4948 CYM 50769
Novel non-peptide NPBWR1 antagonist
4949 MaxiPost
Potassium channel modulator; exerts subtype-specific effects
4950 ICA 110381
KV7.2/7.3 activator; displays anticonvulsant properties
4951 SA 4503 dihydrochloride
Selective σ1 receptor agonist
4952 TRAM 39
Potent KCa3.1 blocker
4953 CHIR 99021 trihydrochloride
Hydrochloride salt of CHIR 99021 (Cat. No. 4423); selective GSK-3 inhibitor
4954 UAMC 00039 dihydrochloride
Dipeptidyl peptidase II (DPP-II) inhibitor
4957 ML 179
Selective liver receptor homolog 1 (LRH1) inverse agonist
4958 Eplivanserin hemifumarate
Potent and selective 5-HT2A antagonist
4959 CID 16020046
Selective GPR55 antagonist
4960 AR-C155858
MCT1 and MCT2 inhibitor; inhibits glycolysis in cancer cells
4961 TC-S 7001
Potent and highly selective ROCK inhibitor; orally active
4962 SB 204990
ATP citrate lyase (ACLY) inhibitor
4963 SC 144 hydrochloride
gp130 inhibitor; blocks cytokine-triggered gp130 signaling
4964 R 1485 dihydrochloride
Selective and high affinity 5-HT6 antagonist
4965 PD 180970
p210Bcr/Abl kinase inhibitor; also inhibits c-Src and KIT
4968 CCT 241533 dihydrochloride
Potent Chk2 inhibitor
4969 LY 2389575 hydrochloride
Selective negative allosteric modulator of mGlu3 receptors
4970 BMS 688521
Potent inhibitor of the LFA-1/ICAM interaction
4972 JIB 04
Pan Jumonji inhibitor; active in vivo
4975 CRT 0066101
Potent protein kinase D (PKD) inhibitor
4976 ML 289
Selective negative allosteric modulator of mGlu3 receptors
4977 RN 1 dihydrochloride
LSD1 inhibitor
4978 Pyrintegrin
Enhances survival of human ESCs following enzymatic dissociation
4979 Methylmalonate
Succinate dehydrogenase inhibitor
4981 Cystamine dihydrochloride
Transglutaminase inhibitor; neuroprotective
4982 ML 337
Selective negative allosteric modulator of mGlu3 receptors
4983 ACT 335827
Potent and selective OX1 antagonist
4984 CK 869
Arp2/3 inhibitor; inhibits actin polymerization
4985 Miglitol
α-glucosidase inhibitor
4986 K 02288
Type 1 BMP receptor inhibitor
4988 Vialinin A
Inhibitor of USP4 and USP5/IsoT
4989 Salirasib
Ras inhibitor; also induces autophagy
4990 Stavudine
Nucleoside analog; antiviral
4991 HaXS8
Chemical dimerizer
4992 IWP L6
Potent PORCN inhibitor
4993 NSC 624206
Ubiquitin-activating enzyme (E1) inhibitor
4994 PYZD 4409
Ubiquitin-activating enzyme (E1) inhibitor
4995 Phortress
Prodrug of the antitumor agent 5F 203
4996 PMX 464
Putative inhibitor of the Trx-TrxR system; antiproliferative
4997 INDY
DYRK1A/B inhibitor
4998 ProINDY
DYRK1A/B inhibitor; prodrug of INDY (Cat. No. 4997)
4999 9-Phenanthrol
Selective TRPM4 blocker

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