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Displaying Products by Catalog Number (3300 - 3399)

Cat. No. Product Name / Activity
3300 SU 5402
Potent FGFR and VEGFR inhibitor
3301 NU 6140
Cdk2 inhibitor; also potent inhibitor of aurora kinase A and B
3302 CD 3254
Potent and selective RXRα agonist
3303 UVI 3003
RXR antagonist
3304 SU 16f
Potent and selective PDGFRβ inhibitor
3305 Alfuzosin hydrochloride
Uroselective α1 antagonist
3306 8-(3-Chlorostyryl)caffeine
Selective A2A antagonist. Also MAO-B inhibitor
3307 PF 750
Selective FAAH inhibitor
3308 Zileuton
5-LOX inhibitor; orally bioavailable
3309 Fluvastatin sodium
Potent HMG-CoA reductase inhibitor
3311 VU 0155041 sodium salt
Potent positive allosteric modulator of mGlu4 receptors; sodium salt of VU 0155041 (Cat. No. 3248)
3312 BzATP triethylammonium salt
Photoaffinity label for ATPase; also P2X7 agonist and P2X1/P2Y1 partial agonist
3313 rac BHFF
Potent and selective postitive allosteric modulator of GABAB receptors
3314 BI 78D3
Selective, competitive JNK inhibitor
3315 RS 25344 hydrochloride
Potent PDE4 inhibitor
3316 PF 670462
Potent and selective CK1ε and CK1δ inhibitor
3317 AZ 11645373
Potent and selective human P2X7 antagonist
3318 SC 514
IKKβ inhibitor; attenuates NF-κB-induced gene expression
3319 ARL 17477 dihydrochloride
Selective nNOS inhibitor
3321 AR-C 66096 tetrasodium salt
Potent and selective P2Y12 antagonist
3322 ZD 9379
Brain penetrant NMDA antagonist; acts at glycine site
3323 AZ 10606120 dihydrochloride
Potent P2X7 receptor antagonist
3324 QS 11
ARFGAP1 inhibitor; modulates Wnt/β-catenin signaling
3325 VU 1545
Positive allosteric modulator of mGlu5 receptors
3326 BGC 20-761
High affinity 5-HT6 antagonist
3327 CID 755673
Selective protein kinase D inhibitor
3328 Desformylflustrabromine hydrochloride
Positive allosteric modulator of α4β2 nAChRs; also muscle-type nAChR inhibitor
3331 NPEC-caged-(1S,3R)-ACPD
Caged (1S,3R)-ACPD
3332 NPEC-caged-LY 379268
Caged version of LY 379268 (Cat. No. 2453)
3333 NDT 9513727
Potent, selective human C5a receptor negative allosteric modulator (NAM)
3335 SU 6668
PDGFR, VEGFR and FGFR inhibitor
3336 A 769662
Potent AMPK activator
3337 CART (55-102) (rat)
Neuromodulatory neuropeptide fragment; satiety factor
3338 CART (55-102) (human)
Neuromodulatory neuropeptide fragment; satiety factor
3339 CART (62-76) (rat, human)
Neuromodulating neuropeptide fragment; inhibits food intake in vivo
3341 JK 184
Alcohol dehydrogenase 7 inhibitor; inhibits downstream Hh signaling pathway
3342 L-798,106
Potent and highly selective EP3 antagonist
3343 Ro 8-4304 hydrochloride
GluN2B-selective NMDA antagonist
3344 SLV 320
Potent and selective A1 antagonist
3346 ATC 0175 hydrochloride
MCH1 antagonist; also 5-HT2B antagonist and 5-HT1A partial agonist
3347 SNAP 94847 hydrochloride
Potent and selective MCH1 antagonist
3348 10Panx
Panx-1 mimetic inhibitory peptide; blocks pannexin-1 gap junctions
3349 Biocytin
Versatile marker for neuroanatomical investigations
3350 LY 393558
Dual 5-HT1B and 5-HT1D antagonist; also 5-HT re-uptake inhibitor
3351 Selexipag
Selective prostacyclin IP1 receptor agonist
3352 JNJ 28871063 hydrochloride
Potent ErbB receptor family inhibitor
3353 PSN 375963 hydrochloride
GPR119 receptor agonist
3354 PF 429242 dihydrochloride
Competitive inhibitor of SREBP site 1 protease
3355 PNU 177864 hydrochloride
Highly selective D3 antagonist
3356 WR 1065 dihydrochloride
p53 activator. Also ROS scavenger
3357 Ellipticine
Antitumor and intercalating agent; inhibits DNA topoisomerase II
3358 MG 101
Calpain inhibitor; activates p53-dependent apoptosis
3360 CGP 52411
EGFR inhibitor. Also inhibits Aβ42 fibril formation
3361 JNJ 17203212
Reversible, competitive and potent TRPV1 antagonist
3362 MIRA-1
Restores mutant p53 activity; proapoptotic
3364 BIX 01294
GLP and G9a inhibitor
3365 Tenovin-1
Protects against MDM2-mediated p53 degradation
3366 WAY 200070
Selective ERβ agonist
3367 AT 101
Downregulates Bcl-2 and Mcl-1; pro-apoptotic
3368 SB 271046 hydrochloride
Selective 5-HT6 antagonist; orally active
3369 AC 55541
Potent and selective PAR2 agonist
3370 AC 264613
PAR2 receptor agonist
3371 TCS OX2 29
Potent and selective OX2 antagonist
3373 Valinomycin
Selective K+ ionophore
3374 Cortistatin 14
Endogenous neuropeptide; binds sst1 - sst5, ghrelin receptor and MRGPRX2
3375 Dolastatin 10 trifluoroacetate
Tubulin polymerization inhibitor
3377 (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
Selective vasopressin V1A antagonist
3378 EIPA
Inhibits TRPP3-mediated currents; also inhibits the Na+/H+ exchanger (NHE)
3379 Phenamil
Inhibits TRPP3-mediated currents; also inhibits epithelial Na+ channels
3380 Benzamil
NCX inhibitor, Deg/ENaC channel blocker; amiloride (Cat. No. 0890) derivative
3381 AM 1172
Anandamide uptake inhibitor; also FAAH inhibitor and CB receptor partial agonist
3383 VU 152100
Positive allosteric modulator of M4 receptors
3384 (Z)-Pugnac
O-GlcNAcase and β-hexosaminidase inhibitor
3385 GW 791343 hydrochloride
P2X7 allosteric modulator
3387 Gedunin
Hsp90 inhibitor; exhibits anticancer and antimalarial activity
3388 Anastrozole
Potent aromatase (CYP19) inhibitor
3389 Bicalutamide
Non-steroidal androgen receptor antagonist
3390 Thymosin β4
Potent actin polymerization regulator
3391 Amyloid β-peptide (42-1) (human)
Inactive control peptide for amyloid β-peptide (1-42) (Cat. No. 1428)
3392 VKGILS-NH2
Control peptide for SLIGKV-NH2 (Cat. No. 3010)
3393 RLLFT-NH2
Control peptide for TFLLR-NH2 (Cat. No. 1464)
3394 LRGILS-NH2
Control peptide for SLIGRL-NH2 (Cat. No. 1468)
3395 Lestaurtinib
JAK2, FLT3 and TrkA inhibitor; also inhibits AurA and AurB
3396 Desmopressin
Synthetic vasopressin analog; V1B and V2 agonist
3397 LY 2365109 hydrochloride
Potent and selective GlyT1 inhibitor
3399 Myelin Basic Protein (87-99)
Major antigenic component implicated in the pathophysiology of multiple sclerosis

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