All Products

Displaying Products by Catalog Number (4700 - 4799)

Cat. No. Product Name / Activity
4701 EC 144
High affinity, potent and selective Hsp90 inhibitor
4703 3-Deazaneplanocin A hydrochloride
EZH2 histone methyltransferase inhibitor
4708 TC LPA5 4
LPA5 receptor antagonist
4709 RuBi GABA trimethylphosphine
Caged GABA; inhibits neural activity
4710 PF 06465469
Potent ITK inhibitor; also inhibits BTK
4711 Hexa-D-arginine
Furin inhibitor
4712 Salmeterol xinafoate
Long-acting β2 agonist; bronchodilator
4715 JZL 195
Dual FAAH and MAGL inhibitor
4716 A 967079
Selective TRPA1 channel blocker
4719 VU 0463271
Potent and selective KCC2 inhibitor
4720 Entacapone
Potent COMT inhibitor; blocks α-synuclein aggregation
4723 T2AA
PCNA inhibitor
4724 BTT 3033
Selective inhibitor of integrin α2β1
4726 CTA 056
ITK inhibitor
4727 GS 6201
Selective A2B antagonist
4730 PPY A
Potent inhibitor of Abl T315l mutant and wild-type Abl kinases
4731 KY 02111
Inhibits canonical Wnt signaling. Promotes differentiation of human ESCs and iPSCs into cardiomyocytes
4732 ML 204
Selective TRPC4 inhibitor
4735 Quetiapine hemifumarate
5-HT2 antagonist; also D2 antagonist; atypical antipsychotic
4736 WIN 18446
ALDH1A2 inhibitor
4737 CDDO Im
Nrf2 signaling activator
4741 Gadolinium chloride
Stretch-activated calcium channel blocker; calcium-sensing receptor agonist
4745 LIMKi 3
Potent LIM kinase inhibitor; antitumor
4746 ML SA1
Activator of TRPML channels
4748 ML 221
Apelin antagonist
4750 TC Mps1 12
Potent and selective Mps1 kinase inhibitor
4751 FSLLRY-NH2
PAR2 peptide antagonist
4753 AL 8697
Potent and selective p38α inhibitor
4754 AK 7
Selective SIRT2 inhibitor; brain penetrant
4758 Bromosporine
Broad spectrum bromodomain inhibitor
4759 G-36
Selective GPER antagonist
4763 Pyridostatin pentahydrochloride
Stabilizes G-quadruplexes; induces DNA damage and cell cycle arrest
4767 WAY 316606 hydrochloride
Secreted Frizzled-related protein-1 (sFRP-1) inhibitor; increases Wnt signaling
4773 ESI 09
Epac inhibitor
4774 BMS 536924
Dual IR/IGF1R inhibitor
4775 SD 2590 hydrochloride
Potent MMP inhibitor
4776 BIRT 377
Potent negative allosteric modulator of LFA-1
4777 ML 277
Selective KV7.1 (KCNQ1) potassium channel activator; augments IKs current
4778 BETP
Positive allosteric modulator of GLP-1 receptors
4779 GRI 977143
Selective LPA2 receptor non-lipid agonist
4781 ANA 12
TrkB receptor antagonist
4782 Org 25543 hydrochloride
Potent and selective GlyT2 inhibitor
4784 Edaglitazone
Potent and selective PPARγ agonist; antidiabetic
4786 PD 0332991 isethionate
Potent cdk4 and cdk6 inhibitor; brain penetrant
4788 NS 11021
KCa1.1 (BK) channel activator
4791 Candesartan
AT1 antagonist
4793 CE3F4
Noncompetitive Epac1 inhibitor
4795 Galloflavin
Lactate dehydrogenase inhibitor; impairs aerobic glycolysis
4796 Escitalopram oxalate
Selective serotonin reuptake inhibitor (SSRI)
4798 (S)-Duloxetine hydrochloride
Potent 5-HT and NA reuptake inhibitor (SNRI); also blocks dopamine reuptake

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