All Products

Displaying Products by Catalog Number (4700 - 4799)

Cat. No. Product Name / Activity
4701 EC 144
High affinity, potent and selective Hsp90 inhibitor
4703 3-Deazaneplanocin A hydrochloride
EZH2 histone methyltransferase inhibitor
4708 TC LPA5 4
LPA5 receptor antagonist
4709 RuBi GABA trimethylphosphine
Caged GABA; inhibits neural activity
4710 PF 06465469
Potent ITK inhibitor; also inhibits BTK
4711 Hexa-D-arginine
Furin inhibitor
4712 Salmeterol xinafoate
Long-acting β2 agonist; bronchodilator
4715 JZL 195
Dual FAAH and MAGL inhibitor
4716 A 967079
Selective TRPA1 channel blocker
4719 VU 0463271
Potent and selective KCC2 inhibitor
4720 Entacapone
Potent COMT inhibitor; blocks α-synuclein aggregation
4723 T2AA
PCNA inhibitor
4724 BTT 3033
Selective inhibitor of integrin α2β1
4726 CTA 056
ITK inhibitor
4727 GS 6201
Selective A2B antagonist
4730 PPY A
Potent inhibitor of Abl T315l mutant and wild-type Abl kinases
4731 KY 02111
Inhibits canonical Wnt signaling. Promotes differentiation of human ESCs and iPSCs into cardiomyocytes
4732 ML 204
Selective TRPC4 inhibitor
4735 Quetiapine hemifumarate
5-HT2 antagonist; also D2 antagonist; atypical antipsychotic
4736 WIN 18446
ALDH1A2 inhibitor
4737 CDDO Im
Nrf2 signaling activator
4741 Gadolinium chloride
Stretch-activated calcium channel blocker; calcium-sensing receptor agonist
4745 LIMKi 3
Potent LIM kinase inhibitor; antitumor
4746 ML SA1
Activator of TRPML channels
4748 ML 221
Apelin antagonist
4750 TC Mps1 12
Potent and selective Mps1 kinase inhibitor
PAR2 peptide antagonist
4753 AL 8697
Potent and selective p38α inhibitor
4754 AK 7
Selective SIRT2 inhibitor; brain penetrant
4758 Bromosporine
Broad spectrum bromodomain inhibitor
4759 G-36
Selective GPER antagonist
4763 Pyridostatin pentahydrochloride
Stabilizes G-quadruplexes; induces DNA damage and cell cycle arrest
4767 WAY 316606 hydrochloride
Secreted Frizzled-related protein-1 (sFRP-1) inhibitor; increases Wnt signaling
4773 ESI 09
Epac inhibitor
4774 BMS 536924
Dual IR/IGF1R inhibitor
4775 SD 2590 hydrochloride
Potent MMP inhibitor
4776 BIRT 377
Potent negative allosteric modulator of LFA-1
4777 ML 277
Selective KV7.1 (KCNQ1) potassium channel activator; augments IKs current
4778 BETP
Positive allosteric modulator of GLP-1 receptors
4779 GRI 977143
Selective LPA2 receptor non-lipid agonist
4781 ANA 12
TrkB receptor antagonist
4782 Org 25543 hydrochloride
Potent and selective GlyT2 inhibitor
4784 Edaglitazone
Potent and selective PPARγ agonist; antidiabetic
4786 PD 0332991 isethionate
Potent cdk4 and cdk6 inhibitor; brain penetrant
4788 NS 11021
KCa1.1 (BK) channel activator
4791 Candesartan
AT1 antagonist
4793 CE3F4
Noncompetitive Epac1 inhibitor
4795 Galloflavin
Lactate dehydrogenase inhibitor; impairs aerobic glycolysis
4796 Escitalopram oxalate
Selective serotonin reuptake inhibitor (SSRI)
4798 (S)-Duloxetine hydrochloride
Potent 5-HT and NA reuptake inhibitor (SNRI); also blocks dopamine reuptake

Tocris Products Alphabetically by Name