All Products

Displaying Products by Catalog Number (5600 - 5699)

Cat. No. Product Name / Activity
5600 BA 1
Potent bombesin agonist
5601 DMXAA
mSTING agonist; induces antitumor immunological responses
5602 6877002
CD40-TRAF6 interaction inhibitor
5603 (-)-JQ1
Negative control for (+)-JQ1
5604 MI 14
Potent and selective PI 4-kinase IIIβ inhibitor
5605 CINPA 1
Potent CAR antagonist
5606 LOC14
High affinity protein disulfide isomerase (PDI) modulator
5607 GNF 7
Ras signaling inhibitor; inhibits Ack1 and GCK
5608 BS 181 dihydrochloride
Selective cdk7 inhibitor
5609 DFHBI
GFP fluorophore mimic for imaging RNA in living cells; activated by binding Spinach2 and Broccoli aptamers
5610 DFHBI 1T
GFP fluorophore mimic for imaging RNA in living cells; activated by binding Spinach2 and Broccoli aptamers
5611 Salvinorin B
Activator of κ-opioid DREADD (KORD)
5613 AZD 9272
Potent and selective mGlu5 antagonist; brain penetrant
5614 AZD 2066
mGlu5 antagonist; orally bioavailable and brain penetrant
5615 AZD 3147
Potent and selective dual mTORC1 and 2 inhibitor; orally bioavailable
5617 AZD 1480
Potent and selective JAK2 inhibitor; antiangiogenic
5619 N-Acetylcysteine amide
Glutathione (GSH) precursor; neuroprotective
5620 BDY FL-X, SE
Green BDY (BODIPY® or boron-dipyrromethene) fluorescent dye for the labeling of amines; supplied as NHS ester
5621 GLPG 0974
Potent FFA2 (GPR43) antagonist
5622 HTH 01-015
Potent and selective NUAK1 inhibitor
5625 ML 334
Inhibitor of Keap1- Nrf2 interaction
5626 SR 7826
Potent and selective LIMK inhibitor; antitumor
5631 LDN 193188
Inhibitor of phosphatidylcholine transfer protein (PC-TP)
5632 AZ Dyrk1B 33
Potent and selective Dyrk1B kinase inhibitor
5633 MRS 2905
Potent and selective P2Y14 receptor agonist
5635 GSK 2801
Selective BAZ2A and BAZ2B inhibitor
5636 GS 143
β-TrCP1 ligase inhibitor
5641 MSC 2032964A
Potent and selective ASK1 inhibitor; orally bioavailable
5642 CMPD101
Potent and selective GRK2/3 inhibitor
5646 EML 425
Reversible and non-competitive CBP/p300 inhibitor
5648 Hydroxychloroquine sulfate
Autophagy inhibitor; also TLR9 inhibitor
5650 SAR 216471 hydrochloride
Potent P2Y12 antagonist; orally available
5651 ONO 6818
High affinity and selective human neutrophil elastase 1 (HNE1) inhibitor; orally active
5653 JW 74
Wnt pathway inhibitor
5654 BMS 265246
Cdk inhibitor; potently inhibits cdk1 and cdk2
5655 GN 44028
Potent HIF-1α inhibitor
5656 DY 268
Potent FXR antagonist
5658 AR-C 141990 hydrochloride
MCT1 inhibitor
5659 AmmTX3
KV4 channel blocker
5660 NVP CXCR2 20
Potent and selective CXCR2 antagonist
5661 666-15
Potent and selective CREB inhibitor
5664 O4I2
Oct3/4 inducer; induces expression of pluripotent-associated genes
5665 IRAK1/4 Inhibitor I
IRAK4 and IRAK1 inhibitor
5666 JNJ 63533054
Potent and selective GPR139 agonist
5667 YK 3-237
SIRT1 activator
5668 VUF 11222
High affinity non-peptide CXCR3 agonist
5671 SB 332235
Potent CXCR2 antagonist
5672 GSK 319347A
Potent and selective IKKε inhibitor
5673 GW 2580
Selective cFMS kinase inhibitor; orally bioavailable
5674 GW 501516
Potent and selective PPARδ agonist
5675 AZ PFKFB3 26
Potent and selective PFKFB3 inhibitor
5676 Guangxitoxin 1E
Potent Kv2.1 and Kv2.2 channel blocker
5677 RFRP-1 (human)
Potent NPFF receptor agonist
5678 RN 9893 hydrochloride
Potent and selective TRPV4 antagonist
5679 N-Acetylpuromycin
Downregulates SnoN and Ski protein expression; promotes TGF-β signaling
5680 Vatalanib succinate
Potent VEGFR inhibitor; also aromatase inhibitor
5681 N106
Activator of SUMO-activating enzyme, E1 ligase
5682 OSU 03012
PDPK1 (PDK1) inhibitor; inhibits Akt signaling
5683 MMAE
Potent dolastatin 10 analog; antitumor
5684 Naloxone 3-glucuronide carbonic acid salt
Naloxone conjugate
5687 Centrinone
High affinity and selective PLK4 inhibitor
5690 Centrinone B
High affinity and selective PLK4 inhibitor
5692 ITH 12575
Mitochondrial Na+/Ca2+ exchange (mNCX) inhibitor
5693 VU 0409551
Selective positive allosteric modulator of mGlu5 receptors; brain penetrant and orally bioavailable
5694 GSK 2033
Potent LXR antagonist
5695 Eggmanone
Potent and selective PDE4 inhibitor; suppresses hedgehog signaling
5697 PMX 53c
Negative control for PMX 53 (Cat. No. 5473)
5698 1-Methyl-D-tryptophan
Indoleamine 2,3-dioxygenase (IDO) inhibitor
5699 IP7e
Potent Nurr1 activator

Tocris Products Alphabetically by Name