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Displaying Products by Catalog Number (5600 - 5699)

Cat. No. Product Name / Activity
5601 DMXAA
mSTING agonist; induces antitumor immunological responses
5602 6877002
CD40-TRAF6 interaction inhibitor
5603 (-)-JQ1
Negative control for (+)-JQ1
5604 MI 14
Potent and selective PI 4-kinase IIIβ inhibitor
5607 GNF 7
Ras signaling inhibitor; inhibits Ack1 and GCK
5608 BS 181 dihydrochloride
Selective cdk7 inhibitor
5609 DFHBI
GFP fluorophore mimic for imaging RNA in living cells; activated by binding Spinach2 and Broccoli aptamers
5610 DFHBI 1T
GFP fluorophore mimic for imaging RNA in living cells; activated by binding Spinach2 and Broccoli aptamers
5611 Salvinorin B
Activator of κ-opioid DREADD (KORD)
5613 AZD 9272
Potent and selective mGlu5 antagonist; brain penetrant
5614 AZD 2066
mGlu5 antagonist; orally bioavailable and brain penetrant
5617 AZD 1480
Potent and selective JAK2 inhibitor; antiangiogenic
5619 N-Acetylcysteine amide
Glutathione (GSH) precursor; neuroprotective
5621 GLPG 0974
Potent FFA2 (GPR43) antagonist
5622 HTH 01-015
Potent and selective NUAK1 inhibitor
5625 ML 334
Inhibitor of Keap1- Nrf2 interaction
5626 SR 7826
Potent and selective LIMK inhibitor; antitumor
5631 LDN 193188
Inhibitor of phosphatidylcholine transfer protein (PC-TP)
5632 AZ Dyrk1B 33
Potent and selective Dyrk1B kinase inhibitor
5633 MRS 2905
Potent and selective P2Y14 receptor agonist
5636 GS 143
β-TrCP1 ligase inhibitor
5641 MSC 2032964A
Potent and selective ASK1 inhibitor; orally bioavailable
5642 CMPD101
Potent and selective GRK2/3 inhibitor
5646 EML 425
Reversible and non-competitive CBP/p300 inhibitor
5648 Hydroxychloroquine sulfate
Autophagy inhibitor; also TLR9 inhibitor
5651 ONO 6818
High affinity and selective human neutrophil elastase 1 (HNE1) inhibitor; orally active
5653 JW 74
Wnt pathway inhibitor
5654 BMS 265246
Cdk inhibitor; potently inhibits cdk1 and cdk2
5655 GN 44028
Potent HIF-1α inhibitor
5656 DY 268
Potent FXR antagonist
5658 AR-C 141990 hydrochloride
MCT1 inhibitor
5661 666-15
Potent and selective CREB inhibitor
5664 O4I2
Oct3/4 inducer; induces expression of pluripotent-associated genes
5665 IRAK1/4 Inhibitor I
IRAK4 and IRAK1 inhibitor
5666 JNJ 63533054
Potent and selective GPR139 agonist
5668 VUF 11222
High affinity non-peptide CXCR3 agonist
5671 SB 332235
Potent CXCR2 antagonist
5672 GSK 319347A
Potent and selective IKKε inhibitor
5673 GW 2580
Selective cFMS kinase inhibitor; orally bioavailable
5674 GW 501516
Potent and selective PPARδ agonist
5675 AZ PFKFB3 26
Potent and selective PFKFB3 inhibitor
5676 Guangxitoxin 1E
Potent Kv2.1 and Kv2.2 channel blocker
5678 RN 9893 hydrochloride
Potent and selective TRPV4 antagonist
5679 N-Acetylpuromycin
Downregulates SnoN and Ski protein expression; promotes TGF-β signaling
5680 Vatalanib succinate
Potent VEGFR inhibitor; also aromatase inhibitor
5682 OSU 03012
PDPK1 (PDK1) inhibitor; inhibits Akt signaling
5687 Centrinone
High affinity and selective PLK4 inhibitor
5690 Centrinone B
High affinity and selective PLK4 inhibitor
5692 ITH 12575
Mitochondrial Na+/Ca2+ exchange (mNCX) inhibitor
5693 VU 0409551
Selective positive allosteric modulator of mGlu5 receptors; brain penetrant and orally bioavailable
5694 GSK 2033
Potent LXR antagonist
5697 PMX 53c
Negative control for PMX 53 (Cat. No. 5473)
5698 1-Methyl-D-tryptophan
Indoleamine 2,3-dioxygenase (IDO) inhibitor
5699 IP7e
Potent Nurr1 activator

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