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Displaying Products by Catalog Number (1500 - 1599)

Cat. No. Product Name / Activity
1500 BQ 788 sodium salt
Selective ETB antagonist
1504 Milrinone
PDE3 inhibitor
1505 Mycophenolic acid
Inosine monophosphatase dehydrogenase (IMPDH) inhibitor
1506 Terazosin hydrochloride
α1 and α2B antagonist (α1 > α2B). Orally active
1507 FR 122047 hydrochloride
Cyclooxygenase (COX-1) inhibitor
1508 GW 9662
Selective covalent PPARγ antagonist
1509 TMS
Cytochrome P450 1B1 inhibitor
1510 Ozagrel hydrochloride
Selective thromboxane A2 synthetase inhibitor
1511 SR 59230A hydrochloride
Potent and selective β3 antagonist
1512 SB 205384
GABAA modulator; slows current decay
1513 CGP 7930
Positive allosteric modulator of GABAB receptors
1514 CGP 13501
Positive allosteric modulator of GABAB receptors
1515 17-AAG
Selective Hsp90 inhibitor
1516 SDZ 21009
β-adrenoceptor antagonist; also 5-HT1A and 5-HT1B antagonist
1518 5-Iodo-A-85380 dihydrochloride
High affinity α4β2 and α6β2 subtype-selective nAChR agonist
1519 Quinelorane hydrochloride
D2 and D3 agonist
1520 Hypericin
Inhibits tyrosine kinases
1521 LY 233053
Competitive NMDA antagonist
1523 LY 215840
5-HT2/5-HT7 antagonist
1524 LY 288513
Selective CCK2 antagonist
1526 Mevastatin
HMG-CoA reductase inhibitor
1527 5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative
Precursor to 5-Iodo-A-85380 (Cat. No. 1518)
1529 SNC 162
Potent, selective non-peptide δ agonist
1530 Lovastatin
Potent HMG-CoA reductase inhibitor
1531 Icilin
Activates a novel cold receptor. Cooling agent
1534 A 68930 hydrochloride
Potent and selective D1-like agonist
1535 Hemokinin 1 (mouse)
Endogenous, high affinity and selective NK1 agonist
1539 β-Pompilidotoxin
Slows neuronal Na+ channel inactivation
1540 DCPIB
Blocker of VRAC/ICl, swell
1541 HA14-1
Bcl-2 inhibitor. Induces apoptosis
1542 Splitomicin
Sir2p inhibitor
1543 (S)-CPW 399
Subtype-selective weakly desensitizing AMPA agonist
1544 (±)-Bay K 8644
CaV1.x activator
1545 (R)-(+)-Bay K 8644
CaV1.x blocker; (R)-(+)-enantiomer of (±)-Bay K 8644; also TMEM176B inhibitor
1546 (S)-(-)-Bay K 8644
CaV1.x activator; (S)-(-)-enantiomer of (±)-Bay K 8644
1547 NSC 95397
Selective Cdc25 dual specificity phosphatase inhibitor
1548 Cantharidin
Protein phosphatase 1 and 2A inhibitor
1549 CD 437
RARγ-selective agonist
1550 SC 560
Cyclooxygenase-1 (COX-1) inhibitor
1551 STO-609 acetate
Selective CaM kinase kinase inhibitor
1552 UFP-101
Potent, selective silent antagonist for NOP
1554 Piceatannol
Inhibits TNF-induced NF-κB activation
1555 AG 825
Selective ErbB2 inhibitor
1558 Tracazolate hydrochloride
Allosteric modulator of GABAA receptors
1559 Roxindole hydrochloride
Dopamine D2 autoreceptor agonist. Also has affinity for D3, D4, 5-HT1A receptors and the 5-HT transporter
1560 CTAP
Potent and selective μ antagonist
1561 (S)-SNAP 5114
GABA uptake inhibitor
1562 Angiotensin (1-7)
Vasorelaxant peptide
1563 Angiotensin I (human, mouse, rat)
Endogenous precursor to angiotensin II (Cat. No. 1158)
1565 JIP-1 (153-163)
JNK-selective inhibitor peptide
1566 [(pF)Phe4]Nociceptin(1-13)NH2
Potent, selective nociceptin receptor agonist
1567 Thiolutin
Bacterial RNA polymerase inhibitor
1568 NADA
Endogenous CB1 agonist; also vanilloid agonist and inhibitor of FAAH and AMT
1570 (-)-Cannabidiol
Natural cannabinoid; GPR55 antagonist, weak CB1 antagonist, CB2 inverse agonist and AMT inhibitor
1571 Cucurbitacin I
Selective inhibitor of STAT3/JAK2 signaling
1577 L-R4W2
TRPV1 antagonist peptide
1578 CTOP
Potent and selective μ antagonist
High affinity selective A3 agonist
1580 Purvalanol A
Cdk inhibitor; potently inhibits cdk1, cdk2 and cdk5
1581 Purvalanol B
Selective cdk inhibitor; potently inhibits cdk1, cdk2 and cdk5
1582 Neurokinin B (human, porcine)
Endogenous tachykinin peptide
1584 MRS 1706
Potent and selective A2B inverse agonist
1586 SKF 83566 hydrobromide
Potent and selective D1-like antagonist; also inhibits adenylyl cyclase 2
1587 Ro 32-0432 hydrochloride
Potent, orally active PKC inhibitor
1588 Indatraline hydrochloride
Potent 5-HT uptake inhibitor; also inhibits dopamine and noradrenalin uptake
1589 Radicicol
Hsp90 inhibitor. Antifungal antibiotic
1590 [Arg14,Lys15]Nociceptin
Highly potent and selective NOP agonist
1591 NBI 27914 hydrochloride
Selective non-peptide CRF1 antagonist
1592 SCH 79797 dihydrochloride
Potent, selective non-peptide PAR1 antagonist
1594 Ro 25-6981 maleate
GluN2B-selective NMDA antagonist
1596 pep4c
Inactive control peptide for pep2m (Cat. No. 1595)
1597 pep2-SVKI
Peptide inhibitor of GluA2 subunit binding to GRIP, ABP and PICK1; increases AMPA current amplitude
1599 pep2-EVKI
Peptide inhibitor of GluA2 subunit binding to PICK1

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