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Biological Activity for Repaglinide
Repaglinide is a Kir6 (KATP) channel blocker that binds with high affinity for SUR1 when co-expressed with Kir6.2 (Kd = 0.42 nM). Antidiabetic glucose regulator with hypoglycaemic effect in vivo.
Compound Libraries for Repaglinide
Technical Data for Repaglinide
|Storage||Store at +4°C|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Solubility Data for Repaglinide
|Solvent||Max Conc. mg/mL||Max Conc. mM|
Preparing Stock Solutions for Repaglinide
The following data is based on the product molecular weight 452.59. Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||2.21 mL||11.05 mL||22.1 mL|
|5 mM||0.44 mL||2.21 mL||4.42 mL|
|10 mM||0.22 mL||1.1 mL||2.21 mL|
|50 mM||0.04 mL||0.22 mL||0.44 mL|
References for Repaglinide
References are publications that support the biological activity of the product.
Mark and Grell (1997) Hypoglycaemic effects of the novel antidiabetic agent repagl. in rats and dogs. Br.J.Pharmacol. 121 1597 PMID: 9283692
Hansen et al (2005) Kir6.2-dependent high-affinity repagl. binding to β-cell KATP channels. Br.J.Pharmacol. 144 551 PMID: 15678092
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Keywords: Repaglinide, Repaglinide supplier, K+, channel, pore, blockers, KATP, Blocks, SUR1, KIR6, Kir6.2, sulphonylurea, receptor, inward, rectifier, AG-EE, 623ZW, Inward, Potassium, Channels, 3805, Tocris Bioscience
Citations for Repaglinide
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Currently there are no citations for Repaglinide. Do you know of a great paper that uses Repaglinide from Tocris? Please let us know.
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Literature in this Area
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