MRS 4062 triethylammonium salt

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Cat.No. 4261 - MRS 4062 triethylammonium salt | C18H26N3O15P3.4(C2H5)3N | CAS No. 1309871-50-8
Description: Selective P2Y4 receptor agonist
Chemical Name: N4-Phenylpropoxycytidine-5'-O-triphosphate tetra(triethylammonium) salt
Purity: ≥99% (HPLC)
Datasheet
Citations (1)
Reviews
Literature

Biological Activity

Selective P2Y4 receptor agonist (EC50 values are 23, 640, and 740 nM for hP2Y4, hP2Y2 and hP2Y6 respectively).

Technical Data

M. Wt 1022.09
Formula C18H26N3O15P3.4(C2H5)3N
Storage Store at -20°C
Purity ≥99% (HPLC)
CAS Number 1309871-50-8
PubChem ID 90488925
InChI Key ZCDZFMKRHPANNI-IHQKQWLFSA-N
Smiles O[C@@H]1[C@@H](COP(OP(OP([O-])([O-])=O)([O-])=O)([O-])=O)O[C@@H](N3C(N/C(C=C3)=N\OCCCC2=CC=CC=C2)=O)[C@@H]1O.CC[N+](CC)([H])CC.CC[N+](CC)([H])CC.CC[N+](CC)([H])CC.CC[N+](CC)([H])CC

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

Solubility Soluble in water (supplied pre-dissolved at a concentration of 10mM)

Preparing Stock Solutions

The following data is based on the product molecular weight 1022.09. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 0.98 mL 4.89 mL 9.78 mL
5 mM 0.2 mL 0.98 mL 1.96 mL
10 mM 0.1 mL 0.49 mL 0.98 mL
50 mM 0.02 mL 0.1 mL 0.2 mL

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Product Datasheets

Safety Datasheet

References

References are publications that support the biological activity of the product.

Maruoka et al (2011) Pyrimidine nucleotides with 4-alkyloxyimino and terminal tetraphosphate δ-ester modifications as selective agonists of the P2Y4 receptor. J.Med.Chem. 54 4018 PMID: 21528910


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1 Citation for MRS 4062 triethylammonium salt

Citations are publications that use Tocris products. Selected citations for MRS 4062 triethylammonium salt include:

Ilatovskaya et al (2013) Pharmacological characterization of the P2 receptors profile in the podocytes of the freshly isolated rat glomeruli. Am J Physiol Cell Physiol 305 C1050 PMID: 24048730


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Literature in this Area

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* or download your copy today!

*Please note that Tocris will only send literature to established scientific business / institute addresses.


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