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Chlormezanone is a anxiolytic and skeletal muscle relaxant that acts at the benzodiazepine site of GABAA receptors.
Chlormezanone is also offered as part of the Tocriscreen 2.0 Max. Find out more about compound libraries available from Tocris.
|Storage||Store at RT|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
|Solvent||Max Conc. mg/mL||Max Conc. mM|
The following data is based on the product molecular weight 273.73. Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||3.65 mL||18.27 mL||36.53 mL|
|5 mM||0.73 mL||3.65 mL||7.31 mL|
|10 mM||0.37 mL||1.83 mL||3.65 mL|
|50 mM||0.07 mL||0.37 mL||0.73 mL|
References are publications that support the biological activity of the product.
Ervin and Cooper (1988) Use of conditioned taste aversion as a conflict model: effects of anxiolytic drugs. J.Pharmacol.Exp.Ther. 245 137 PMID: 2896235
Simiand et al (1989) Comparative study in mice of tetrazepam and other centrally active skeletal muscle relaxants. Arch.Int.Pharmacodyn.Ther. 297 272 PMID: 2567153
Merck Index 12 2155
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Keywords: Chlormezanone, Chlormezanone supplier, Skeletal, muscle, relaxant, GABAA, Receptors, benzodiazepine, PAM, 0456, Tocris Bioscience
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