Other Kinases

Other Kinase Agonists

Cat. No. Product Name / Activity
6617 LYN 1604 dihydrochloride
Potent UNC-51-like kinase 1 (ULK1) agonist

Other Kinase Inhibitors

Cat. No. Product Name / Activity
5097 A12B4C3
Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor
7283 Apilimod dimesylate
Potent and selective PIKfyve inhibitor
7511 ARN 3236
Potent inhibitor of salt-inducible kinases
7001 AT 7867
Potent p70-S6 kinase inhibitor; also potently inhibits Akt and PKA
7673 BAY 091
Potent and selective PIP4K2A inhibitor
5123 BMX-IN-1
Potent and irreversible BMX inhibitor
5382 C16
PKR inhibitor
7018 CBR-470-1
PGK1 inhibitor; activates Nrf2
6558 CP 43
Potent TAOK inhibitor
2755 DCA
Mitochondrial pyruvate dehydrogenase kinase (PDK) inhibitor
7285 DCLK1-IN-1
Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable
3572 GSK 650394
Serum- and glucocorticoid-regulated kinase (SGK) inhibitor
6976 JNJ 10198409
c-Abl, Lck, c-Src and Fyn kinase inhibitor; also inhibits PDGFRα and PDGFRβ
5845 JX 06
Potent and selective pyruvate dehydrogenase kinase (PDK) 1/2/3 inhibitor
5604 MI 14
Potent and selective PI 4-kinase IIIβ inhibitor
4880 ML 281
STK33 inhibitor
5134 MRT 67307 dihydrochloride
Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor
5780 MRT 68921 dihydrochloride
ULK inhibitor
7927 MSC 1186
Potent and selective SRPK family inhibitor
7371 Neratinib
Potent inhibitor of MST1; also inhibits EGFR and ErbB2 kinases
5429 NG 25
TGF-β-activated kinase (TAK1) inhibitor
3439 NH 125
Histidine protein kinase inhibitor; also inhibits CaM kinase III
3960 NVP 231
Potent, selective and reversible CerK inhibitor
3604 (5Z)-7-Oxozeaenol
Potent and selective TAK1 MAPKKK inhibitor
5752 PF 06260933 dihydrochloride
MAP4K4 (HGK) inhibitor; also inhibits MINK and TNIK
4278 PF 431396
Dual FAK/PYK2 inhibitor
4630 SB 747651A dihydrochloride
Potent MSK1 inhibitor; also inhibits other AGC group kinases
6528 SGC AAK1 1
AAK1 and BMP2K inhibitor; activates Wnt signaling
6564 SGC GAK 1
High affinity cyclin G associated kinase (GAK) inhibitor
5570 STOCK2S 26016
Lysine deficient protein kinase (WNK) signaling inhibitor
6430 Takinib
Potent and selective TAK1/MAP3K7 kinase inhibitor
5240 TC-S 7006
Potent and selective Tpl2 (Cot; MAP3K8) inhibitor
3946 TNP
Inhibitor of IP6K; also inhibits IP3K
5271 UNC 3230
Potent and selective PIP5K1C inhibitor; antinociceptive
6604 VER 246608
Potent and selective pyruvate dehydrogenase kinase (PDK) 1/2/3/4 inhibitor
5413 WH-4-023
Potent salt inducible kinase (SIK) inhibitor; also inhibits Lck and Src
5493 XL 413 hydrochloride
Potent and selective Cdc7 inhibitor
6482 XMU MP 1
Potent and selective MST1/2 inhibitor; orally bioavailable


Cat. No. Product Name / Activity
2600 Clofarabine
Deoxycytidine kinase (dCK) substrate
6018 Nicotinamide Riboside
NAD+ precursor; substrate for nicotinamide riboside kinases

Other Kinase Activators

Cat. No. Product Name / Activity
7980 MTK 458
PINK1 activator
7876 PZ 3022
PanK Activator
7809 TEPP 46
Potent and selective pyruvate kinase M2 (PKM2) allosteric activator


Cat. No. Product Name / Activity
7425 CG 428
Potent tropomyosin receptor kinase (TRK) Degrader
6524 TL 12-186
Multikinase Degrader


Cat. No. Product Name / Activity
7426 CG 428-Neg
Negative control for CG 428 (Cat. No. 7425)
6529 SGC AAK1 1N
Negative control for SGC AAK1 1 (Cat.No. 6528)
6525 TL 13-27
Negative control for TL 12-186 (Cat. No. 6524)


Cat. No. Product Name / Activity
7546 C28
Potent LMTK3 inhibitor