Other Kinases

Inhibitors

Cat No Product Name / Activity
5097 A12B4C3
Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor
5123 BMX-IN-1
Potent and irreversible BMX inhibitor
5382 C16
PKR inhibitor
6558 CP 43
Potent TAOK inhibitor
2755 DCA
Mitochondrial pyruvate dehydrogenase kinase (PDK) inhibitor
6632 ERGi-USU
Rio2 kinase (RIOK2) inhibitor; inhibits ERG protein
6480 GSK 583
Potent RIP2 kinase inhibitor; orally bioavailable and cell permeable
3572 GSK 650394
Serum- and glucocorticoid-regulated kinase (SGK) inhibitor
6492 GSK'872
Potent and selective receptor activating protein kinase 3 (RIP3) inhibitor
5845 JX 06
Potent and selective pyruvate dehydrogenase kinase (PDK) 1/2/3 inhibitor
6229 LP 922761
Potent AAK1 inhibitor; peripherally restricted
5604 MI 14
Potent and selective PI 4-kinase IIIβ inhibitor
4880 ML 281
STK33 inhibitor
5134 MRT 67307 dihydrochloride
Salt inducible kinase (SIK) inhibitor
5780 MRT 68921 dihydrochloride
Potent ULK inhibitor; inhibits autophagy
2324 Necrostatin-1
RIPK1 inhibitor; inhibits necroptosis
5429 NG 25
TGF-β-activated kinase (TAK1) inhibitor
3439 NH 125
Histidine protein kinase inhibitor. Also inhibits CaM kinase III
3960 NVP 231
Potent, selective and reversible CerK inhibitor
3604 (5Z)-7-Oxozeaenol
Potent and selective TAK1 MAPKKK inhibitor
5752 PF 06260933 dihydrochloride
MAP4K4 (HGK) inhibitor; also inhibits MINK and TNIK
4278 PF 431396
Dual FAK/PYK2 inhibitor
6440 PIK 93
Potent PI 4-KIIIβ, PI 3-Kγ, and PI 3-Kα inhibitor
4630 SB 747651A dihydrochloride
Potent MSK1 inhibitor; also inhibits other AGC group kinases
6528 SGC AAK1 1
AAK1 and BMP2K inhibitor; activates Wnt signaling
6564 SGC GAK 1
High affinity cyclin G associated kinase (GAK) inhibitor
5063 SRPIN340
Selective SRPK1 inhibitor
6036 STK16-IN-1
Serine/threonine protein kinase 16 (STK16) inhibitor; also inhibits PI 3Kδ, PI 3Kγ and mTOR kinases
5570 STOCK2S 26016
Lysine deficient protein kinase (WNK) signaling inhibitor
5240 TC-S 7006
Potent and selective Tpl2 (Cot; MAP3K8) inhibitor
3946 TNP
Inhibitor of IP6K; also inhibits IP3K
5271 UNC 3230
Potent and selective PIP5K1C inhibitor; antinociceptive
5413 WH-4-023
Potent salt inducible kinase (SIK) inhibitor; also inhibits Lck and Src
5493 XL 413 hydrochloride
Potent and selective Cdc7 inhibitor
6482 XMU MP 1
Potent and selective MST1/2 inhibitor; orally bioavailable

Substrates

Cat No Product Name / Activity
2600 Clofarabine
Deoxycytidine kinase (dCK) substrate

Other

Cat No Product Name / Activity
4082 Anti-PIKFyve
Antibody recognizing PIKfyve
6524 TL 12-186
Multikinase degrading PROTAC
6525 TL 13-27
Negative control for TL 12-186