Other Proteases
Other Protease Inhibitors |
|
|---|---|
| Cat. No. | Product Name / Activity |
| 5402 | 6bK |
| Insulin degrading enzyme (IDE) inhibitor | |
| 5175 | AEBSF |
| Broad spectrum, irreversible inhibitor of serine proteases | |
| 5491 | Aliskiren hemifumarate |
| Potent renin inhibitor; antihypertensive | |
| 2511 | APC 366 |
| Tryptase inhibitor | |
| 4139 | Aprotinin |
| Competitive serine protease inhibitor | |
| 1637 | Argatroban |
| Potent thrombin inhibitor | |
| 3193 | Camostat mesylate |
| Orally active protease inhibitor; inhibits entry of SARS-Cov-2 into lung cells | |
| 2512 | CGS 35066 |
| Endothelin-converting enzyme (ECE) inhibitor | |
| 0460 | Cinanserin hydrochloride |
| 3C-like proteinase inhibitor; also selective 5-HT2 antagonist; antiviral | |
| 3501 | Decanoyl-RVKR-CMK |
| Subtilisin/Kex2p-like proprotein convertase inhibitor | |
| 4524 | EGCG |
| β-secretase (BACE) inhibitor; inhibits amyloid assembly | |
| 1798 | Gabexate mesylate |
| Serine protease inhibitor; inhibits thrombin, trypsin, kallikrein and plasmin | |
| 6272 | KYP 2047 |
| High affinity prolyl oligopeptidase inhibitor; anti-angiogenic, neuroprotective and brain penetrant | |
| 2627 | L-685,458 |
| High affinity SPP inhibitor; also potent γ-secretase inhibitor | |
| 1167 | Leupeptin hemisulfate |
| Inhibits trypsin-like/cysteine proteases | |
| 7081 | LY 2886721 Hydrochloride |
| Potent and selective β-secretase (BACE) inhibitor | |
| 4848 | MI 2 (MALT1 inhibitor) |
| MALT1 inhibitor | |
| 3081 | Nafamostat mesylate |
| Serine protease inhibitor; inhibits tryptase | |
| 6423 | Pep 2-8 |
| Potent PCSK9 inhibitor | |
| 3354 | PF 429242 dihydrochloride |
| Competitive inhibitor of SREBP site 1 protease | |
| 6333 | Phosphoramidon disodium salt |
| Neutral endopeptidase and endothelin converting enzyme inhibitor | |
| 4486 | PMSF |
| Non-selective protease inhibitor; also blocks anandamide metabolism | |
| 5772 | Sacubitril calcium |
| Membrane metallo-endopeptidase (neprilysin) inhibitor prodrug; orally bioavailable | |
| 6658 | Telaprevir |
| Hepatitis C virus (HCV) protease NS3/4A inhibitor | |
| 4954 | UAMC 00039 dihydrochloride |
| Dipeptidyl peptidase II (DPP-II) inhibitor | |
| 7659 | Verubecestat |
| BACE1 and BACE2 inhibitor | |
| 5563 | VTP 27999 trifluoroacetate |
| Highly potent and selective renin inhibitor | |
| 4645 | Z-VRPR-FMK trifluoroacetate salt |
| Irreversible MALT1 inhibitor | |
Substrates |
|
| Cat. No. | Product Name / Activity |
| 3791 | Hemopressin (human, mouse) |
| Bioactive substrate for endopeptidase 24.15, neurolysin and ACE | |