Integrin Inhibitors

Cat No Product Name / Activity
2524 A 205804
Selective inhibitor of E-selectin and ICAM-1 expression
4228 A 286982
Potent inhibitor of the LFA-1/ICAM-1 interaction
6058 ATN 161
α5β1 integrin receptor antagonist
3910 BIO 1211
Selective α4β1 (VLA-4) inhibitor
5051 BIO 5192
Highly potent and selective inhibitor of integrin α4β1
4970 BMS 688521
Potent inhibitor of the LFA-1/ICAM interaction
6047 BOP
Dual α9β1/α4β1 integrin inhibitor; preferentially mobilizes HSCs
4724 BTT 3033
Selective inhibitor of integrin α2β1
5870 Cilengitide
Potent and selective inhibitor of integrins αvβ3 and αvβ5
3202 Echistatin, α1 isoform
αVβ3 and glycoprotein IIb/IIIa (integrin αIIbβ3) inhibitor
4725 Eptifibatide
Glycoprotein IIb/IIIa inhibitor; inhibits platelet aggregation
1263 GR 144053 trihydrochloride
Glycoprotein IIb/IIIa (integrin αIIbβ3) receptor antagonist. Antithrombotic
2877 MNS
Glycoprotein IIb/IIIa (αIIbβ3) inhibitor. Also inhibits Src and Syk
4664 Obtustatin
Potent and selective α1β1 inhibitor
4744 P11
Potent antagonist of αvβ3-vitronectin interaction; antiangiogenic
6048 R-BC154
High affinity fluorescent α4β1/α9β1 inhibitor; mobilizes HSCs
3498 RGDS peptide
Integrin binding sequence; inhibits integrin receptor function
4527 TC-I 15
Potent α2β1 inhibitor; displays antithrombotic activity in vivo
3900 TCS 2314
α4β1 (VLA-4) antagonist