GABAA Receptor Modulators

Cat. No. Product Name / Activity
3972 AA 29504
Positive allosteric modulator of GABAA receptors
3653 Allopregnanolone
Positive allosteric modulator of GABAA receptors
3679 DS2
Positive allosteric modulator of GABAA receptors; displays subunit selectivity
3113 Etifoxine hydrochloride
GABAA potentiator; anxiolytic
1471 Etomidate
GABA-mimetic; selectively interacts with β2- and β3-subunit containing GABAA receptors
2867 Flupirtine maleate
GABAA modulator; also indirect NMDA antagonist and Kv7 channel activator
2531 Ganaxolone
Potent positive allosteric modulator of GABAA receptors
1295 Loreclezole hydrochloride
Subtype-selective GABAA modulator
4949 MaxiPost
Negative modulator of GABAA receptors; also potassium channel modulator
4410 Ocinaplon
GABAA modulator; anxiolytic
2738 Org 20599
Positive allosteric modulator of GABAA receptors; direct agonist at higher concentrations
2681 17-PA
Antagonist of neurosteroid potentiation and direct gating of GABAA
3652 Pregnanolone
Postitive allosteric modulator of GABAA receptors
5376 Pregnenolone sulfate sodium salt
GABAA inhibitor; displays some subunit selectivity; NMDA potentiator; also activates TRPM3 channels
6192 PZ-II-029
α6β3γ2-selective GABAA positive allosteric modulator
1512 SB 205384
GABAA modulator; slows current decay
6334 THDOC
Positive modulator of GABAA receptors; endogenous neurosteroid
3620 Topiramate
Positive allosteric modulator of GABAA receptors; GluK1 antagonist; also inhibits carbonic anhydrase (CA) II and IV
1558 Tracazolate hydrochloride
Allosteric modulator of GABAA receptors
2734 U 89843A
Positive allosteric modulator of GABAA receptors