GABAA Receptor Modulators

Cat. No. Product Name / Activity
3972 AA 29504
Positive allosteric modulator of GABAA receptors
3653 Allopregnanolone
Positive allosteric modulator of GABAA receptors
0881 Chlormethiazole hydrochloride
Potentiates GABAA receptor function
3679 DS2
Positive allosteric modulator of GABAA receptors; displays subunit selectivity
3113 Etifoxine hydrochloride
GABAA potentiator; anxiolytic
1471 Etomidate
GABA-mimetic; selectively interacts with β2- and β3-subunit containing GABAA receptors
2867 Flupirtine maleate
GABAA modulator; also indirect NMDA antagonist and Kv7 channel activator
2531 Ganaxolone
Potent positive allosteric modulator of GABAA receptors
1295 Loreclezole hydrochloride
Subtype-selective GABAA modulator
4949 MaxiPost
Negative modulator of GABAA receptors; also potassium channel modulator
4410 Ocinaplon
GABAA modulator; anxiolytic
2738 Org 20599
Positive allosteric modulator of GABAA receptors; direct agonist at higher concentrations
2681 17-PA
Antagonist of neurosteroid potentiation and direct gating of GABAA
3652 Pregnanolone
Postitive allosteric modulator of GABAA receptors
5376 Pregnenolone sulfate sodium salt
GABAA inhibitor; displays some subunit selectivity; NMDA potentiator; also activates TRPM3 channels
0830 Primidone
Potentiates GABAA receptor function
6192 PZ-II-029
α6β3γ2-selective GABAA positive allosteric modulator
1512 SB 205384
GABAA modulator; slows current decay
6334 THDOC
Positive modulator of GABAA receptors; endogenous neurosteroid
3620 Topiramate
Positive allosteric modulator of GABAA receptors; GluK1 antagonist; also inhibits carbonic anhydrase (CA) II and IV
1558 Tracazolate hydrochloride
Allosteric modulator of GABAA receptors
2734 U 89843A
Positive allosteric modulator of GABAA receptors
2733 U 90042
GABAA ligand
3048 Valerenic acid
Positive allosteric modulator of GABAA receptors