GABAA Receptor Modulators
| Cat. No. | Product Name / Activity |
|---|---|
| 3653 | Allopregnanolone |
| Positive allosteric modulator of GABAA receptors | |
| 1513 | CGP 7930 |
| Positive allosteric modulator of GABAA and GABAB receptors | |
| 3679 | DS2 |
| Positive allosteric modulator of GABAA receptors; displays subunit selectivity | |
| 3113 | Etifoxine hydrochloride |
| GABAA potentiator; anxiolytic | |
| 1471 | Etomidate |
| GABA-mimetic; selectively interacts with β2- and β3-subunit containing GABAA receptors | |
| 2867 | Flupirtine maleate |
| GABAA modulator; also indirect NMDA antagonist and Kv7 channel activator | |
| 2531 | Ganaxolone |
| Potent positive allosteric modulator of GABAA receptors | |
| 1295 | Loreclezole hydrochloride |
| Subtype-selective GABAA modulator | |
| 4949 | MaxiPost |
| Negative modulator of GABAA receptors; also potassium channel modulator | |
| 3652 | Pregnanolone |
| Postitive allosteric modulator of GABAA receptors | |
| 5376 | Pregnenolone sulfate sodium salt |
| GABAA inhibitor; displays some subunit selectivity; NMDA potentiator; also activates TRPM3 channels | |
| 6334 | THDOC |
| Positive modulator of GABAA receptors; endogenous neurosteroid | |
| 3620 | Topiramate |
| Positive allosteric modulator of GABAA receptors; GluK1 antagonist; also inhibits carbonic anhydrase (CA) II and IV |
GABA Scientific Review
Our GABA review gives an overview of the structure and function of the GABA receptors, as well as highlighting pharmacological ligands for their study.
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