5-HT Transporter Inhibitors

Cat. No. Product Name / Activity
2341 A 80426 mesylate
5-HT uptake inhibitor and α2 antagonist
4456 Amitriptyline hydrochloride
5-HT and NA reuptake inhibitor (SNRI); also TrkA/B agonist
4357 Bicifadine hydrochloride
Noradrenalin, 5-HT and dopamine re-uptake inhibitor
2322 BTS 54-505 hydrochloride
Potent 5-HT and NA reuptake inhibitor (SNRI); active metabolite of sibutramine (Cat. No. 2290)
1427 Citalopram hydrobromide
Highly potent and selective 5-HT uptake inhibitor
0457 Clomipramine hydrochloride
5-HT reuptake inhibitor
2833 Cocaine hydrochloride
Inhibitor of monoamine transporters
4358 Dapoxetine hydrochloride
Selective serotonin reuptake inhibitor (SSRI)
2695 Dexfenfluramine hydrochloride
5-HT reuptake inhibitor; also stimulates 5-HT release
4798 (S)-Duloxetine hydrochloride
Potent 5-HT and NA reuptake inhibitor (SNRI); also blocks dopamine reuptake
4796 Escitalopram oxalate
Selective serotonin reuptake inhibitor (SSRI)
0927 Fluoxetine hydrochloride
5-HT reuptake inhibitor
1033 Fluvoxamine maleate
5-HT reuptake inhibitor
1588 Indatraline hydrochloride
Potent 5-HT uptake inhibitor; also inhibits dopamine and noradrenalin uptake
2545 Lofepramine
5-HT and NA reuptake inhibitor (SNRI)
3350 LY 393558
5-HT reuptake inhibitor; also 5-HT1B and 5-HT1D antagonist
2148 (±)-McN 5652
Potent, orally active 5-HT uptake inhibitor; also inhibits noradrenalin and dopamine uptake in vitro
3027 (±)-MDMA hydrochloride
Inhibitor of 5-HT and dopamine uptake; hallucinogenic
3286 Milnacipran hydrochloride
5-HT and NA reuptake inhibitor (SNRI)
2777 Nefazodone hydrochloride
5-HT uptake inhibitor; also 5-HT2A antagonist; antidepressant
2141 Paroxetine maleate
Highly potent and selective 5-HT uptake inhibitor
2395 Sertraline hydrochloride
5-HT reuptake inhibitor
2290 Sibutramine hydrochloride
5-HT and NA reuptake inhibitor (SNRI)
2175 Tetrabenazine
Potent inhibitor of vesicular monoamine transport; depletes 5-HT stores
2917 Venlafaxine hydrochloride
5-HT and NA reuptake inhibitor (SNRI)
6202 Vilazodone hydrochloride
Potent SSRI and 5-HT1A partial agonist; antidepressant
4194 WY 45233 succinate
5-HT and NA reuptake inhibitor (SNRI)
1767 Zimelidine dihydrochloride
Selective 5-HT uptake inhibitor