Purinergic (P2X) Receptor Antagonists

Cat. No. Product Name / Activity
6493 A 317491 sodium salt
Selective, high affinity P2X3 and P2X2/3 receptor antagonist; antinociceptive
2972 A 438079 hydrochloride
Competitive P2X7 antagonist
3701 A 740003
Potent and selective P2X7 antagonist
4473 A 804598
Potent and selective P2X7 antagonist
4232 A 839977
Potent P2X7 antagonist
3323 AZ 10606120 dihydrochloride
Potent P2X7 receptor antagonist
3317 AZ 11645373
Potent and selective human P2X7 antagonist
3579 5-BDBD
Potent and selective P2X4 antagonist
5545 BX 430
Selective P2X4 allosteric antagonist
0845 Evans Blue tetrasodium salt
Selective P2X purinergic antagonist; also non-NMDA iGluR antagonist; inhibits L-glutamate uptake into synaptic vesicles
5299 JNJ 47965567
Potent and selective P2X7 antagonist; brain penetrant
1277 KN-62
Non-competitive P2X7 antagonist
1240 NF 023
Selective, competitive P2X1 antagonist
2548 NF 110
Potent P2X3 antagonist
2450 NF 157
Selective P2Y11/P2X1 antagonist
1199 NF 279
Potent and selective P2X1 antagonist
1391 NF 449
Highly selective P2X1 antagonist
0625 PPADS tetrasodium salt
Non-selective P2 antagonist
0683 iso-PPADS tetrasodium salt
P2X antagonist
1309 PPNDS
Potent, selective P2X1 antagonist
2188 Ro 0437626
Selective P2X1 antagonist
4391 Ro 51
Potent P2X3, P2X2/3 antagonist
3052 RO-3
Selective P2X3 and P2X2/3 antagonist
1472 Suramin hexasodium salt
Non-selective P2 antagonist
4386 TC-P 262
Selective P2X3, P2X2/3 antagonist
2464 TNP-ATP triethylammonium salt
Potent, selective P2X antagonist