Cat. No. | Product Name / Activity |
---|---|
5781 | A 425619 |
Potent TRPV1 antagonist | |
4319 | A 784168 |
Potent and selective TRPV1 antagonist | |
4330 | AMG 21629 |
Potent and selective TRPV1 antagonist | |
5995 | AMG 517 |
Potent TRPV1 antagonist | |
2316 | AMG 9810 |
Potent and selective TRPV1 competitive antagonist | |
3875 | BCTC |
TRPV1 antagonist | |
0464 | Capsazepine |
TRPV antagonist; also activator of ENaCδ | |
7199 | (±)-Eriodictyol |
Potent TRPV1 antagonist; also antioxidant; activates Nrf2/ARE signaling | |
5106 | GSK 2193874 |
Potent and selective TRPV4 antagonist; orally active | |
4100 | HC 067047 |
Potent and selective TRPV4 antagonist | |
3361 | JNJ 17203212 |
Reversible, competitive and potent TRPV1 antagonist | |
3746 | RN 1734 |
Selective TRPV4 antagonist | |
5678 | RN 9893 hydrochloride |
Potent and selective TRPV4 antagonist | |
1439 | Ruthenium Red |
Blocks capsaicin-activated cation channels | |
1615 | SB 366791 |
Potent and selective TRPV1 competitive antagonist | |
6990 | SET 2 |
Selective TRPV2 antagonist | |
1098 | Tranilast |
Antiallergic; inhibits TRPV2-mediated responses | |
6831 | TRPV3 74a |
Selective TRPV3 antagonist; brain penetrant |