TRPV Channel Antagonists
| Cat. No. | Product Name / Activity |
|---|---|
| 5781 | A 425619 |
| Potent TRPV1 antagonist | |
| 4319 | A 784168 |
| Potent and selective TRPV1 antagonist | |
| 4330 | AMG 21629 |
| Potent and selective TRPV1 antagonist | |
| 5995 | AMG 517 |
| Potent TRPV1 antagonist | |
| 2316 | AMG 9810 |
| Potent and selective TRPV1 competitive antagonist | |
| 3875 | BCTC |
| TRPV1 antagonist | |
| 0464 | Capsazepine |
| TRPV antagonist; also activator of ENaCδ | |
| 7199 | (±)-Eriodictyol |
| Potent TRPV1 antagonist; also antioxidant; activates Nrf2/ARE signaling | |
| 5106 | GSK 2193874 |
| Potent and selective TRPV4 antagonist; orally active | |
| 4100 | HC 067047 |
| Potent and selective TRPV4 antagonist | |
| 3361 | JNJ 17203212 |
| Reversible, competitive and potent TRPV1 antagonist | |
| 3746 | RN 1734 |
| Selective TRPV4 antagonist | |
| 5678 | RN 9893 hydrochloride |
| Potent and selective TRPV4 antagonist | |
| 1439 | Ruthenium Red |
| Blocks capsaicin-activated cation channels | |
| 1615 | SB 366791 |
| Potent and selective TRPV1 competitive antagonist | |
| 6990 | SET 2 |
| Selective TRPV2 antagonist | |
| 1098 | Tranilast |
| Antiallergic; inhibits TRPV2-mediated responses | |
| 6831 | TRPV3 74a |
| Selective TRPV3 antagonist; brain penetrant |
Pain Research Product Guide
Our Pain guide highlights over 280 products for Pain research.
Request copyRequest PDFPain Life Science Poster
Written by Grant D. Nicol and Michael R. Vasko
Our Peripheral Sensitization poster gives a summary of the excitatory and inhibitory signaling pathways involved in modulation of peripheral sensitization.
Request copyDownload PDF