Free Fatty Acid Receptors

More Information »Free Fatty Acid (FFA) receptors are a group of Gq/11 protein-coupled receptors currently classified into FFA1, FFA2, FFA3 and FFA4 subtypes. FFA receptors are concentrated in pancreatic islet cells, immune cells and in the brain and are important in immunity and metabolism.

Free Fatty Acid Receptor Products

Agonists
Cat.No.
Product Name / Activity
5789 AM 4668
Potent FFA1 (GPR40) agonist
5035 AS 2034178
Selective FFA1 (GPR40) agonist
4642 4-CMTB
FFA2 agonist; also exhibits positive allosteric modulatory activity
4581 Grifolic acid
Selective partial FFA4 (GPR120) agonist
5257 GSK 137647
Potent and selective FFA4 (GPR120) agonist
2649 GW 9508
Potent and selective FFA1 (GPR40) agonist
4615 MEDICA 16
FFA1 (GPR40) agonist; also inhibits ATP citrate lyase
4601 TUG 891
Potent and selective FFA4 (GPR120) agonist
6001 ZQ 16
Selective GPR84 agonist
Antagonists
Cat.No.
Product Name / Activity
5256 AH 7614
Selective FFA4 (GPR120) antagonist
5903 CATPB
FFA2 antagonist/inverse agonist
5357 DC 260126
FFA1 (GPR40) antagonist
5621 GLPG 0974
Potent FFA2 antagonist
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GPCR Product Listing

GPCR Product Listing

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